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Quinolines

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  • 3,5-disubstituted quinolines as novel c-Jun N-terminal kinase inhibitors  Academic Article
  • A new regulatory switch in a JAK protein kinase  Academic Article
  • Activity of piperaquine and other 4-aminoquinoline antiplasmodial drugs against chloroquine-sensitive and resistant blood-stages of Plasmodium falciparum: Role of β-haematin inhibition and drug concentration in vacuolar water- and lipid-phases  Academic Article
  • Chemoproteomics demonstrates target engagement and exquisite selectivity of the clinical phosphodiesterase 10A inhibitor MP-10 in its native environment  Academic Article
  • Combination therapy targeting both tumor-initiating and differentiated cell populations in prostate carcinoma  Academic Article
  • Conformation-induced remote meta-C-H activation of amines  Academic Article
  • Congenital myopathy-causing tropomyosin mutations induce thin filament dysfunction via distinct physiological mechanisms  Academic Article
  • D3 receptor test in vitro predicts decreased cocaine self-administration in rats  Academic Article
  • Design, synthesis, and evaluation of novel 3,6-diaryl-4-aminoalkoxyquinolines as selective agonists of somatostatin receptor subtype 2  Academic Article
  • Determinants of cytochrome P4502C8 substrate binding - structures of complexes with montelukast, troglitazone, felodipine, and 9-cis-retinoic acid  Academic Article
  • Discovery and SAR of muscarinic receptor subtype 1 (M-1) allosteric activators from a molecular libraries high throughput screen. Part 1: 2,5-Dibenzyl-2H-pyrazolo 4,3-c quinolin-3(5H)-ones as positive allosteric modulators  Academic Article
  • Discovery of a drug candidate for GLIS3-associated diabetes  Academic Article
  • Divergent total syntheses of (-)-aspidospermine and (+)-spegazzinine  Academic Article
  • Effects of a 5-lipoxygenase-activating protein inhibitor on biomarkers associated with risk of myocardial infarction - a randomized trial  Academic Article
  • Effects of the slco1b1*15 allele on the pharmacokinetics of pitavastatin  Academic Article
  • Exploiting a water network to achieve enthalpy-driven, bromodomain-selective BET inhibitors  Academic Article
  • Golgicide A reveals essential roles for GBF1 in Golgi assembly and function  Academic Article
  • How thiostrepton was made in the laboratory  Academic Article
  • IL-7/anti-IL-7 mAb complexes augment cytokine potency in mice through association with IgG-Fc and by competition with IL-7R  Academic Article
  • Induction of avian tumor viruses in normal cells by physical and chemical carcinogens  Academic Article
  • Inhibition of dsRNA-induced signaling in hepatitis C virus-infected cells by NS3 protease-dependent and -independent mechanisms  Academic Article
  • Inhibitors of c-jun-n-terminal kinase (jnk)  Academic Article
  • Insights into the mechanism of streptonigrin-induced protein arginine deiminase inactivation  Academic Article
  • Integrated hydrogenated amorphous Si photodiode detector for microfluidic bioanalytical devices  Academic Article
  • Lead optimization of 3-carboxyl-4(1H)-quinolones to deliver orally bioavailable antimalarials  Academic Article
  • Ligand-controlled C(sp(3))-H arylation and olefination in synthesis of unnatural chiral alpha-amino acids  Academic Article
  • Ligand-enabled gamma-C-H olefination and carbonylation: construction of beta-quaternary carbon centers  Academic Article
  • Ligand-enabled methylene C(sp3)-H bond activation with a Pd(II) catalyst  Academic Article
  • Marginal utility of montelukast for persistent asthma  Academic Article
  • Neurochemical evidence that postsynaptic nucleus accumbens D3 receptor stimulation enhances cocaine reinforcement  Academic Article
  • New class of HIV-1 integrase (IN) inhibitors with a dual mode of action  Academic Article
  • New diarylmethylpiperazines as potent and selective nonpeptidic delta opioid receptor agonists with increased in vitro metabolic stability  Academic Article
  • Parallel synthesis of N-biaryl quinolone carboxylic acids as selective M(1) positive allosteric modulators  Academic Article
  • Pd0/PR3-catalyzed arylation of nicotinic and isonicotinic acid derivatives  Academic Article
  • Pharmacological and behavioral profile of N-[(3R)-1-azabicyclo[2.2.2]oct-3-yl]-6-chinolincarboxamide (EVP-5141), a novel α7 nicotinic acetylcholine receptor agonist/serotonin 5-HT3 receptor antagonist  Academic Article
  • Phosphodiesterase 10A regulates alcohol and saccharin self-administration in rats  Academic Article
  • Phospshoinositide 3-kinase (PI3K)/mammalian target of rapamycin (mTOR) dual inhibitors: discovery and structure-activity relationships of a series of quinoline and quinoxaline derivatives  Academic Article
  • Piperaquine resistance is associated with a copy number variation on chromosome 5 in drug-pressured plasmodium falciparum parasites  Academic Article
  • Quinelorane, a dopamine D3/D2 receptor agonist, reduces prepulse inhibition of startle and ventral pallidal GABA efflux: time course studies  Academic Article
  • S1P3-mediated cardiac fibrosis in sphingosine kinase 1 transgenic mice involves reactive oxygen species  Academic Article
  • Screening helix-threading peptides for RNA binding using a thiazole orange displacement assay  Academic Article
  • Selective inhibitors and tailored activity probes for lipoprotein-associated phospholipase A(2)  Academic Article
  • Stereocontrolled synthesis of the quinaldic acid macrocyclic system of thiostrepton  Academic Article
  • Streptonigrin and lavendamycin partial structures - probes for the minimum, potent pharmacophore of streptonigrin, lavendamycin, and synthetic quinoline-5,8-diones  Academic Article
  • Structure-activity relationships of imidazo[4,5-f]quinoline partial structures and analogs. Discovery of pyrazolo[3,4-f]quinoline derivatives as potent immunostimulants  Academic Article
  • Synthesis of artemiside and its effects in combination with conventional drugs against severe murine malaria.  Academic Article
  • Synthesis of small molecule inhibitors of the orphan nuclear receptor steroidogenic factor-1 (NR5A1) based on isoquinolinone scaffolds  Academic Article
  • The PI3K/Akt pathway contributes to arenavirus budding  Academic Article
  • Thiazole orange as the fluorescent intercalator in a high resolution fid assay for determining DNA binding affinity and sequence selectivity of small molecules  Academic Article
  • Total synthesis of thiostrepton, part 2: Construction of the quinaldic acid macrocycle and final stages of the synthesis  Academic Article

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