articles
- A SNAP-tag fluorogenic probe mimicking the chromophore of the red fluorescent protein Kaede. 17:1906-1915. 2019
- A designed protein binding-pocket to control excited-state intramolecular proton transfer fluorescence. 17:1076-1080. 2019
- Binding orientation and reactivity of alkyl α,ω-dibromides in water-soluble cavitands. 17:5279-5282. 2019
- Chemical composition of DNA-encoded libraries, past present and future. 17:4676-4688. 2019
- Identification of a lysine 4-hydroxylase from the glidobactin biosynthesis and evaluation of its biocatalytic potential. 17:1736-1739. 2019
- Rational design of a function-based selection method for genetically encoding acylated lysine derivatives. 17:6127-6130. 2019
- Stereoselective functionalization of platensimycin and platencin by sulfa-Michael/aldol reactions. 17:4261-4272. 2019
- The structure-based traceless specific fluorescence labeling of the smoothened receptor. 17:6136-6142. 2019
- Using reversible non-covalent and covalent bonds to create assemblies and equilibrating molecular networks that survive 5 molar urea. 17:2081-2086. 2019
- Vinylogous acyl triflates as an entry point to α,β-disubstituted cyclic enones via Suzuki-Miyaura cross-coupling. 17:1796-1799. 2019
- An asymmetric Mannich reaction of α-diazocarbonyl compounds and N-sulfonyl cyclic ketimines catalyzed by complexes generated from chiral and achiral phosphines with gold(i). 16:2923-2931. 2018
- Chemoenzymatic macrocycle synthesis using resorcylic acid lactone thioesterase domains. 16:5771-5779. 2018
- Chiral NHC-catalyzed 1,3-dipolar 3+2 cycloaddition of azomethine imines with alpha-chloroaldehydes for the synthesis of bicyclic pyrazolidinones. 16:4433-4438. 2018
- Design, synthesis, and biological evaluation of C7-functionalized DMXAA derivatives as potential human-STING agonists 2018
- Glycosylation of a model proto-RNA nucleobase with non-ribose sugars: implications for the prebiotic synthesis of nucleosides. 16:1263-1271. 2018
- Tandem Diels-Alder/oxidation-aromatization reactions involving 2-styrylchromones and arynes. 16:6077-6085. 2018
- Transition-metal-free synthesis of polysubstituted pyrrole derivatives via cyclization of methyl isocyanoacetate with aurone analogues. 16:5422-5426. 2018
- Asymmetric synthesis of vinylogous β-amino acids and their incorporation into mixed backbone oligomers. 15:3255-3264. 2017
- Base-catalyzed diastereoselective trimerization of trifluoroacetone. 15:5131-5134. 2017
- Construction of tetrahydropyranoquinoline derivatives via an asymmetric organocatalytic aza-Michael-IED/HAD cascade reaction. 15:9630-9637. 2017
- Engineering a periplasmic binding protein for amino acid sensors with improved binding properties. 15:8761-8769. 2017
- Stevens rearrangement of thioethers with arynes: a facile access to multi-substituted β-keto thioethers. 15:2716-2720. 2017
- The design and synthesis of an α-Gal trisaccharide epitope that provides a highly specific anti-Gal immune response. 15:2979-2992. 2017
- Weinreb amide directed cross-coupling reaction between electron-deficient alkenes catalyzed by a rhodium catalyst. 15:1236-1244. 2017
- A mild preparation of alkynes from alkenyl triflates. 14:5591-5594. 2016
- Assessment of reagents for selenocysteine conjugation and the stability of selenocysteine adducts. 14:5141-5147. 2016
- Chemoenzymatic synthesis and utilization of a SAM analog with an isomorphic nucleobase. 14:6189-6192. 2016
- Cyclopropenation of internal alkynylsilanes and diazoacetates catalyzed by copper(I) N-heterocyclic carbene complexes. 14:1742-1747. 2016
- Enantioselective polyene cyclizations. 14:5454-5467. 2016
- Flexibility is important for inhibition of the MDM2/p53 protein-protein interaction by cyclic β-hairpins. 14:10386-10393. 2016
- Scalable procedure for the fragmentation of hydroperoxides mediated by copper and iron tetrafluoroborate salts. 14:6197-6200. 2016
- Selective inhibition of p97 by chlorinated analogues of dehydrocurvularin. 14:5918-5921. 2016
- Thermodynamic origin of α-helix stabilization by side-chain cross-links in a small protein. 14:5768-5773. 2016
- A concise synthesis of single components of partially sulfated oligomannans. 13:11550-11560. 2015
- Copper-catalysed cross-coupling: an untapped potential. 13:4816-4827. 2015
- Cyanine polyene reactivity: scope and biomedical applications. 13:7584-7598. 2015
- Functional chromatographic technique for natural product isolation. 13:2255-2259. 2015
- Receptor-templated stapling of intrinsically disordered peptide ligands. 13:4183-4189. 2015
- Synthesis and application of a dual chiral [2.2]paracyclophane-based N-heterocyclic carbene in enantioselective β-boration of acyclic enones. 13:10691-10698. 2015
- Solid phase synthesis of 1,3,4-oxadiazin-5 (6R)-one and 1,3,4-oxadiazol-2-one scaffolds from acyl hydrazides. 13:59-63. 2015
- Comparison of backbone modification in protein β-sheets by α→γ residue replacement and α-residue methylation. 12:5375-5381. 2014
- Multivalent glycosylated nanoparticles for studying carbohydrate-protein interactions. 12:5563-5573. 2014
- Protein backbone engineering as a strategy to advance foldamers toward the frontier of protein-like tertiary structure. 12:8796-8802. 2014
- Synthesis of sesquiterpene-inspired derivatives designed for covalent binding and their inhibition of the NF-κB pathway. 12:370-375. 2014
- The mechanism of the NHC catalyzed aza-Morita-Baylis-Hillman reaction: insights into a new substrate-catalyzed bimolecular pathway. 12:2176-2179. 2014
- Folded alkyl chains in water-soluble capsules and cavitands. 12:6561-6563. 2014
- Methods to enable the design of bioactive small molecules targeting RNA. 12:1029-1039. 2014
- Support of academic synthetic chemistry using separation technologies from the pharmaceutical industry. 12:2161-2166. 2014
- Chemoenzymatic synthesis and in situ application of S-adenosyl-L-methionine analogs. 11:7606-7610. 2013
- Copper(II)-catalyzed trifluoromethylation of N-aryl imines. 11:6242-6245. 2013
- Synthesis of acylguanidine zanamivir derivatives as neuraminidase inhibitors and the evaluation of their bio-activities. 11:3943-3948. 2013
- Chemical approaches for detection and destruction of nerve agents. 11:3936-3942. 2013
- Synthesis and biological evaluation of new paclitaxel analogs and discovery of potent antitumor agents. 11:4154-4163. 2013
- Synthesis of libraries of peptidomimetic compounds containing a 2-oxopiperazine unit in the main chain. 11:2088-2092. 2013
- A cucurbit[8]uril sponge. 10:8587-8589. 2012
- Alkadienyl and alkenyl itaconic acids (ceriporic acids G and H) from the selective white-rot fungus Ceriporiopsis subvermispora: a new class of metabolites initiating ligninolytic lipid peroxidation. 10:6432-6442. 2012
- Binding trimethyllysine and other cationic guests in water with a series of indole-derived hosts: large differences in affinity from subtle changes in structure. 10:6885-6892. 2012
- Construction of highly functional α-amino nitriles via a novel multicomponent tandem organocatalytic reaction: a facile access to α-methylene γ-lactams. 10:2214-2217. 2012
- Discovery of an entropically-driven small molecule streptavidin binder from nucleic acid-encoded libraries. 10:1502-1505. 2012
- Gas extrusion in natural products total synthesis. 10:8383-8392. 2012
- Synthetic approaches to a chiral 4-amino-3-hydroxy piperidine with pharmaceutical relevance. 10:5253-5257. 2012
- Bicyclic core estrogens as full antagonists: Synthesis, biological evaluation and structure-activity relationships of estrogen receptor ligands based on bridged oxabicyclic core arylsulfonamides. 10:8692-8700. 2012
- Exploring the self-assembly of glycopeptides using a diphenylalanine scaffold. 9:5755-5761. 2011
- Protein assembly directed by synthetic molecular recognition motifs. 9:7296-7299. 2011
- Synthesis of serine-based glycolipids as potential TLR4 activators. 9:2492-2504. 2011
- Impact of sugar stereochemistry on natural killer T cell stimulation by bacterial glycolipids. 9:7659-7662. 2011
- Mechanism-based crosslinking as a gauge for functional interaction of modular synthases. 8:1769-1772. 2010
- Preparation of FRET reporters to support chemical probe development. 8:4601-4606. 2010
- Selective inhibition of ADAR2-catalyzed editing of the serotonin 2c receptor pre-mRNA by a helix-threading peptide. 8:4898-4904. 2010
- Synthetic studies on the mycolactone core. 8:5159-5165. 2010
- Combinatorial approach toward synthesis of small molecule libraries as bacterial transglycosylase inhibitors. 8:2586-2593. 2010
- In water, on water, and by water: Mimicking nature's aldolases with organocatalysis and water. 8:4043-4050. 2010
- N-methylcysteine-mediated total chemical synthesis of ubiquitin thioester. 8:2392-2396. 2010
- Regioselective synthesis of di-c-glycosylflavones possessing anti-inflammation activities. 8:4451-4462. 2010
- Intramolecular azide-alkyne [3 + 2] cycloaddition: versatile route to new heterocyclic structural scaffolds. 7:1921-1930. 2009
- Dynamic polythioesters via ring-opening polymerization of 1,4-thiazine-2,5-diones. 7:2878-2884. 2009
- New development of glycan arrays. 7:2247-2254. 2009
- The pyridinone-methide elimination. 7:4825-4828. 2009
- Synthesis and evaluation of novel pyridine based PLG tripeptidomimetics. 6:1647-1654. 2008
- A systems perspective to digital structures in molecular analysis. 5:214-222. 2007
- Sialic acid and N-acyl sialic acid analog production by fermentation of metabolically and genetically engineered Escherichia coli. 5:1903-1909. 2007
- A deep cavitand catalyzes the Diels-Alder reaction of bound maleimides. 5:3631-3636. 2007
- Geometry in digital molecular arrays. 4:3052-3055. 2006
- One-pot chemo-enzymatic synthesis of reporter-modified proteins. 4:44-46. 2006
- Microtiter plate based chemistry and in situ screening: A useful approach for rapid inhibitor discovery. 4:1446-1457. 2006
- Sigma-chelation-directed C-H functionalizations using Pd(II) and Cu(II) catalysts: Regioselectivity, stereoselectivity and catalytic turnover. 4:4041-4047. 2006
- Synthesis of iso-epoxy-amphidinolide n and des-epoxy-caribenolide i structures. Initial forays. 4:2119-2157. 2006
- Synthesis of iso-epoxy-amphidinolide n and des-epoxy-caribenolide i structures. Revised strategy and final stages. 4:2158-2183. 2006
- α- and β-Stilbenosides as base-pair surrogates in DNA hairpins. 4:314-322. 2006
- New aminocyclitols as modulators of glucosylceramide metabolism. 3:1195-1201. 2005
- Preferred dimerization of tetra-tolyl- and tetra-tosylurea derivatives of flexible and rigidified calix[4]arenes. 2:3080-3084. 2004
- The ins and outs of molecular encapsulation. 2:3051-3059. 2004
- Metabolic engineering - a genetic toolbox for small molecule organic synthesis. 1:1-4. 2003
- Molecular screening on a compact disc. 1:3244-3249. 2003
- Discovery and optimization of non-steroidal FXR agonists from natural product-like libraries. 1:908-920. 2003
- HIV-1 protease: Mechanism and drug discovery. 1:5-14. 2003