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Discovery of inhibitors of the channel-activating protease prostasin (CAP1/PRSS8) utilizing structure-based design

Academic Article
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Overview

authors

  • Tully, D. C.
  • Vidal, A.
  • Chatterjee, A. K.
  • Williams, J. A.
  • Roberts, M. J.
  • Petrassi, Mike
  • Spraggon, G.
  • Bursulaya, B.
  • Pacoma, R.
  • Shipway, A.
  • Schumacher, A. M.
  • Danahay, H.
  • Harris, J. L.

publication date

  • November 2008

journal

  • Bioorganic & Medicinal Chemistry Letters  Journal

subject areas

  • Combinatorial Chemistry Techniques
  • Crystallography, X-Ray
  • Molecular Mimicry
  • Molecular Structure
  • Protein Conformation
  • Serine Endopeptidases
  • Serine Proteinase Inhibitors
  • Structure-Activity Relationship
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Research

keywords

  • Channel-activating protease
  • ENaC activation
  • Ketoheterocycle inhibitor
  • PRSS8
  • Peptidomimetic
  • Prostasin
  • hCAP
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Identity

International Standard Serial Number (ISSN)

  • 0960-894X

Digital Object Identifier (DOI)

  • 10.1016/j.bmcl.2008.08.029

PubMed ID

  • 18752942
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Additional Document Info

start page

  • 5895

end page

  • 5899

volume

  • 18

issue

  • 22

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