publication_uri | type | publication_title | year | doi | pmid | journal_uri |
http://vivo.scripps.edu/individual/e2n323827 | AcademicArticle | Reducing limitation in probe design: the development of a diazirine-compatible Suzuki-Miyaura cross coupling reaction | 2019 | 10.1021/acsmedchemlett.8b00403 | 30655947 | http://vivo.scripps.edu/individual/endnote225139 |
http://vivo.scripps.edu/individual/e2n16207 | AcademicArticle | Discovery of MK-1832, a Kv1.5 inhibitor with improved selectivity and pharmacokinetics | 2017 | 10.1016/j.bmc1.2016.12.054 | 28131713 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n362331 | AcademicArticle | Benzoxazolinone aryl sulfonamides as potent, selective Na(v)1.7 inhibitors with in vivo efficacy in a preclinical pain model | 2017 | 10.1016/j.bmcl.2017.04.040 | 28465103 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n36200 | AcademicArticle | Synthesis and optimization of N-heterocyclic pyridinones as catechol-O-methyltransferase (COMT) inhibitors | 2016 | 10.1016/j.bmcl.2016.03.095 | 27133481 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n336092 | AcademicArticle | Synthesis and evaluation of heterocyclic catechol mimics as inhibitors of catechol-O-methyltransferase (COMT) | 2015 | 10.1021/ml500502d | 25815153 | http://vivo.scripps.edu/individual/endnote225139 |
http://vivo.scripps.edu/individual/e2n262575 | AcademicArticle | Characterization of non-nitrocatechol pan and isoform specific catechol-O-methyltransferase inhibitors and substrates | 2012 | 10.1021/cn200109w | 22860182 | http://vivo.scripps.edu/individual/endnote309398 |
http://vivo.scripps.edu/individual/e2n119346 | AcademicArticle | Design, synthesis, and evaluation of novel 3,6-diaryl-4-aminoalkoxyquinolines as selective agonists of somatostatin receptor subtype 2 | 2011 | 10.1021/jm101501b | 21395312 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e2n166711 | AcademicArticle | High concentration electrophysiology-based fragment screen: discovery of novel acid-sensing ion channel 3 (ASIC3) inhibitors | 2011 | 10.1016/j.bmcl.2010.12.115 | 21257308 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n350618 | AcademicArticle | Synthesis and evaluation of 5-fluoro-2-aryloxazolo 5,4-b pyridines as beta-amyloid PET ligands and identification of MK-3328 | 2011 | 10.1021/ml200018n | 24900338 | http://vivo.scripps.edu/individual/endnote225139 |
http://vivo.scripps.edu/individual/e2n18588 | AcademicArticle | (18)F Fluoroazabenzoxazoles as potential amyloid plaque PET tracers: synthesis and in vivo evaluation in rhesus monkey | 2011 | 10.1016/j.nucmedbio.2011.04.004 | 21741254 | http://vivo.scripps.edu/individual/endnote340909 |
http://vivo.scripps.edu/individual/e2n314616 | AcademicArticle | The synthesis and preclinical evaluation in rhesus monkey of F-18 MK-6577 and C-11 CMPyPB glycine transporter 1 positron emission tomography radiotracers | 2011 | 10.1002/syn.20842 | http://vivo.scripps.edu/individual/endnote384899 | |
http://vivo.scripps.edu/individual/e2n133619 | AcademicArticle | Recent progress in the discovery of non-sarcosine based GlyT1 inhibitors | 2010 | 10.2174/156802610790410974 | 20166956 | http://vivo.scripps.edu/individual/endnote373615 |
http://vivo.scripps.edu/individual/e2n135201 | AcademicArticle | Discovery of N-{[1-(propylsulfonyl)-4-pyridin-2-ylpiperidin-4-yl]methyl}benzamides as novel, selective and potent GlyT1 inhibitors | 2009 | 10.1016/j.bmcl.2008.12.115 | 19179073 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n121970 | AcademicArticle | Discovery of GlyT1 inhibitors with improved pharmacokinetic properties | 2009 | 10.1016/j.bmcl.2009.01.015 | 19181525 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n281366 | AcademicArticle | Controlled derivatization of polyhalogenated quinolines utilizing selective cross-coupling reactions | 2008 | 10.1016/j.tetlet.2008.03.040 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/e2n26929 | AcademicArticle | Novel indole-3-sulfonamides as potent HIV non-nucleoside reverse transcriptase inhibitors (NNRTIs) | 2008 | 10.1016/j.bmcl.2007.11.085 | 18083561 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n130520 | AcademicArticle | Recent progress in the discovery of selective, non-peptide ligands of somatostatin receptors | 2008 | 18600562 | http://vivo.scripps.edu/individual/endnote227606 | |
http://vivo.scripps.edu/individual/endnote337664 | AcademicArticle | Rational design, synthesis, and evaluation of key analogues of CC-1065 and the duocarmycins | 2007 | 10.1021/ja073989z | 17948994 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n83902 | AcademicArticle | Synthesis and SAR of GlyT1 inhibitors derived from a series of N-((4-(morpholine-4-carbonyl)-1-(propylsulfonyl)piperidin-4-yl)methyl)benzamides | 2006 | 10.1016/j.bmcl.2006.08.131 | 16987662 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n120231 | AcademicArticle | Convenient preparation of substituted 5-aminooxazoles via a microwave-assisted Cornforth rearrangement | 2006 | 10.1016/j.tet.2005.12.065 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/e2n278056 | AcademicArticle | Identification of potent agonists of photoreceptor-specific nuclear receptor (NR2E3) and preparation of a radioligand | 2006 | 10.1016/j.bmcl.2006.07.056 | 16879962 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n185122 | AcademicArticle | Progress in the preparation and testing of glycine transporter type-1 (GlyT1) inhibitors | 2006 | 10.2174/156802606778249784 | 17017963 | http://vivo.scripps.edu/individual/endnote373615 |
http://vivo.scripps.edu/individual/e2n311209 | AcademicArticle | Potent antagonists of the Kv1.5 potassium channel: synthesis and evaluation of analogous N,N-diisopropyl-2-(pyridine-3-yl)acetamides | 2006 | 10.1016/j.bmcl.2006.08.054 | 16949818 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n382599 | AcademicArticle | Convenient and general microwave-assisted protocols for the expedient synthesis of heterocycles | 2006 | 10.3987/REV-06-SR(W)1 | http://vivo.scripps.edu/individual/endnote14559 | |
http://vivo.scripps.edu/individual/e2n95645 | AcademicArticle | Progress towards validating the NMDA receptor hypofunction hypothesis of schizophrenia | 2006 | 10.2174/156802606777057599 | 16719816 | http://vivo.scripps.edu/individual/endnote373615 |
http://vivo.scripps.edu/individual/endnote244550 | AcademicArticle | Total synthesis of cytostatin | 2006 | 10.3987/COM-06-S(W)13 | http://vivo.scripps.edu/individual/endnote14559 | |
http://vivo.scripps.edu/individual/endnote19249 | AcademicArticle | Total synthesis and evaluation of cytostatin, its C10-C11 diastereomers, and additional key analogues: Impact on PP2A inhibition | 2006 | 10.1021/ja066477d | 17177422 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n209827 | AcademicArticle | Recent advances in positive allosteric modulators of metabotropic glutamate receptors | 2005 | 16022181 | http://vivo.scripps.edu/individual/endnote227606 | |
http://vivo.scripps.edu/individual/e2n243194 | AcademicArticle | Accelerating lead development by microwave-enhanced medicinal chemistry | 2005 | 10.1016/j.ddtec.2005.05.002 | 24981843 | http://vivo.scripps.edu/individual/e9n63592 |
http://vivo.scripps.edu/individual/e2n365916 | AcademicArticle | Applications of microwave-assisted organic synthesis on the multigram scale | 2005 | 16312146 | http://vivo.scripps.edu/individual/endnote227606 | |
http://vivo.scripps.edu/individual/e2n28747 | AcademicArticle | General microwave-assisted protocols for the expedient synthesis of quinoxalines and heterocyclic pyrazines | 2004 | 10.1016/j.tetlet.2004.04.144 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/e2n61318 | AcademicArticle | Efficient synthesis of imidazoles from aldehydes and 1,2-diketones using microwave irradiation | 2004 | 10.1021/ol049682b | 15101765 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/endnote163232 | AcademicArticle | DNA alkylation properties of yatakemycin | 2003 | 10.1021/ja035984h | 12952479 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote322034 | AcademicArticle | Mechanisms of in situ activation for DNA-targeting antitumor agents | 2002 | 10.1021/cr010046q | 12105933 | http://vivo.scripps.edu/individual/endnote51983 |
http://vivo.scripps.edu/individual/endnote114633 | AcademicArticle | Intramolecular Diels-Alder and tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition reactions of 1,3,4-oxadiazoles | 2002 | 10.1021/ja027533n | 12236743 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote46956 | AcademicArticle | Total synthesis of anhydrolycorinone utilizing sequential intramolecular Diels-Alder reactions of a 1,3,4-oxadiazole | 2002 | 10.1021/jo030437k | 12375965 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote277003 | AcademicArticle | Metal cation complexation and activation of reversed CPyi analogues of CC-1065 and duocarmycin SA: Partitioning the effects of binding and catalysis | 2001 | 10.1021/ja010769r | 11562212 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote238936 | AcademicArticle | Combinatorial synthesis and discovery of an antibiotic compound - an experiment suitable for high school and undergraduate laboratories | 2001 | http://vivo.scripps.edu/individual/endnote193577 | ||
http://vivo.scripps.edu/individual/endnote182597 | AcademicArticle | Synthesis and evaluation of 1,2,8, 8a-Tetrahydrocyclopropa[c]pyrrolo[3,2-e]indol-4(5H)-one, the parent alkylation subunit of CC-1065 and the duocarmycins: impact of the alkylation subunit substituents and its implications for DNA alkylation catalysis | 2000 | 10.1021/jo000297j | 10866627 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote239483 | AcademicArticle | A new method of in situ activation for a novel class of DNA alkylating agents: tunable metal cation complexation and activation | 2000 | 10.1021/ja000653f | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote123072 | AcademicArticle | Total synthesis of Amaryllidaceae alkaloids utilizing sequential intramolecular heterocyclic azadiene Diels-Alder reactions of an unsymmetrical 1,2,4,5-tetrazine | 2000 | 10.1021/jo0012546 | 11149859 | http://vivo.scripps.edu/individual/endnote171323 |