Scripps VIVO scripps research logo

  • Index
  • Log in
  • Home
  • People
  • Organizations
  • Research
  • Events
Search form

Publication list

publication_uri type publication_title year doi pmid journal_uri
http://vivo.scripps.edu/individual/e2n323827 AcademicArticle Reducing limitation in probe design: the development of a diazirine-compatible Suzuki-Miyaura cross coupling reaction 2019 10.1021/acsmedchemlett.8b00403 30655947 http://vivo.scripps.edu/individual/endnote225139
http://vivo.scripps.edu/individual/e2n16207 AcademicArticle Discovery of MK-1832, a Kv1.5 inhibitor with improved selectivity and pharmacokinetics 2017 10.1016/j.bmc1.2016.12.054 28131713 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n362331 AcademicArticle Benzoxazolinone aryl sulfonamides as potent, selective Na(v)1.7 inhibitors with in vivo efficacy in a preclinical pain model 2017 10.1016/j.bmcl.2017.04.040 28465103 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n36200 AcademicArticle Synthesis and optimization of N-heterocyclic pyridinones as catechol-O-methyltransferase (COMT) inhibitors 2016 10.1016/j.bmcl.2016.03.095 27133481 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n336092 AcademicArticle Synthesis and evaluation of heterocyclic catechol mimics as inhibitors of catechol-O-methyltransferase (COMT) 2015 10.1021/ml500502d 25815153 http://vivo.scripps.edu/individual/endnote225139
http://vivo.scripps.edu/individual/e2n262575 AcademicArticle Characterization of non-nitrocatechol pan and isoform specific catechol-O-methyltransferase inhibitors and substrates 2012 10.1021/cn200109w 22860182 http://vivo.scripps.edu/individual/endnote309398
http://vivo.scripps.edu/individual/e2n119346 AcademicArticle Design, synthesis, and evaluation of novel 3,6-diaryl-4-aminoalkoxyquinolines as selective agonists of somatostatin receptor subtype 2 2011 10.1021/jm101501b 21395312 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e2n166711 AcademicArticle High concentration electrophysiology-based fragment screen: discovery of novel acid-sensing ion channel 3 (ASIC3) inhibitors 2011 10.1016/j.bmcl.2010.12.115 21257308 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n350618 AcademicArticle Synthesis and evaluation of 5-fluoro-2-aryloxazolo 5,4-b pyridines as beta-amyloid PET ligands and identification of MK-3328 2011 10.1021/ml200018n 24900338 http://vivo.scripps.edu/individual/endnote225139
http://vivo.scripps.edu/individual/e2n18588 AcademicArticle (18)F Fluoroazabenzoxazoles as potential amyloid plaque PET tracers: synthesis and in vivo evaluation in rhesus monkey 2011 10.1016/j.nucmedbio.2011.04.004 21741254 http://vivo.scripps.edu/individual/endnote340909
http://vivo.scripps.edu/individual/e2n314616 AcademicArticle The synthesis and preclinical evaluation in rhesus monkey of F-18 MK-6577 and C-11 CMPyPB glycine transporter 1 positron emission tomography radiotracers 2011 10.1002/syn.20842 http://vivo.scripps.edu/individual/endnote384899
http://vivo.scripps.edu/individual/e2n133619 AcademicArticle Recent progress in the discovery of non-sarcosine based GlyT1 inhibitors 2010 10.2174/156802610790410974 20166956 http://vivo.scripps.edu/individual/endnote373615
http://vivo.scripps.edu/individual/e2n135201 AcademicArticle Discovery of N-{[1-(propylsulfonyl)-4-pyridin-2-ylpiperidin-4-yl]methyl}benzamides as novel, selective and potent GlyT1 inhibitors 2009 10.1016/j.bmcl.2008.12.115 19179073 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n121970 AcademicArticle Discovery of GlyT1 inhibitors with improved pharmacokinetic properties 2009 10.1016/j.bmcl.2009.01.015 19181525 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n281366 AcademicArticle Controlled derivatization of polyhalogenated quinolines utilizing selective cross-coupling reactions 2008 10.1016/j.tetlet.2008.03.040 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/e2n26929 AcademicArticle Novel indole-3-sulfonamides as potent HIV non-nucleoside reverse transcriptase inhibitors (NNRTIs) 2008 10.1016/j.bmcl.2007.11.085 18083561 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n130520 AcademicArticle Recent progress in the discovery of selective, non-peptide ligands of somatostatin receptors 2008 18600562 http://vivo.scripps.edu/individual/endnote227606
http://vivo.scripps.edu/individual/endnote337664 AcademicArticle Rational design, synthesis, and evaluation of key analogues of CC-1065 and the duocarmycins 2007 10.1021/ja073989z 17948994 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n83902 AcademicArticle Synthesis and SAR of GlyT1 inhibitors derived from a series of N-((4-(morpholine-4-carbonyl)-1-(propylsulfonyl)piperidin-4-yl)methyl)benzamides 2006 10.1016/j.bmcl.2006.08.131 16987662 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n120231 AcademicArticle Convenient preparation of substituted 5-aminooxazoles via a microwave-assisted Cornforth rearrangement 2006 10.1016/j.tet.2005.12.065 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/e2n278056 AcademicArticle Identification of potent agonists of photoreceptor-specific nuclear receptor (NR2E3) and preparation of a radioligand 2006 10.1016/j.bmcl.2006.07.056 16879962 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n185122 AcademicArticle Progress in the preparation and testing of glycine transporter type-1 (GlyT1) inhibitors 2006 10.2174/156802606778249784 17017963 http://vivo.scripps.edu/individual/endnote373615
http://vivo.scripps.edu/individual/e2n311209 AcademicArticle Potent antagonists of the Kv1.5 potassium channel: synthesis and evaluation of analogous N,N-diisopropyl-2-(pyridine-3-yl)acetamides 2006 10.1016/j.bmcl.2006.08.054 16949818 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n382599 AcademicArticle Convenient and general microwave-assisted protocols for the expedient synthesis of heterocycles 2006 10.3987/REV-06-SR(W)1 http://vivo.scripps.edu/individual/endnote14559
http://vivo.scripps.edu/individual/e2n95645 AcademicArticle Progress towards validating the NMDA receptor hypofunction hypothesis of schizophrenia 2006 10.2174/156802606777057599 16719816 http://vivo.scripps.edu/individual/endnote373615
http://vivo.scripps.edu/individual/endnote244550 AcademicArticle Total synthesis of cytostatin 2006 10.3987/COM-06-S(W)13 http://vivo.scripps.edu/individual/endnote14559
http://vivo.scripps.edu/individual/endnote19249 AcademicArticle Total synthesis and evaluation of cytostatin, its C10-C11 diastereomers, and additional key analogues: Impact on PP2A inhibition 2006 10.1021/ja066477d 17177422 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n209827 AcademicArticle Recent advances in positive allosteric modulators of metabotropic glutamate receptors 2005 16022181 http://vivo.scripps.edu/individual/endnote227606
http://vivo.scripps.edu/individual/e2n243194 AcademicArticle Accelerating lead development by microwave-enhanced medicinal chemistry 2005 10.1016/j.ddtec.2005.05.002 24981843 http://vivo.scripps.edu/individual/e9n63592
http://vivo.scripps.edu/individual/e2n365916 AcademicArticle Applications of microwave-assisted organic synthesis on the multigram scale 2005 16312146 http://vivo.scripps.edu/individual/endnote227606
http://vivo.scripps.edu/individual/e2n28747 AcademicArticle General microwave-assisted protocols for the expedient synthesis of quinoxalines and heterocyclic pyrazines 2004 10.1016/j.tetlet.2004.04.144 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/e2n61318 AcademicArticle Efficient synthesis of imidazoles from aldehydes and 1,2-diketones using microwave irradiation 2004 10.1021/ol049682b 15101765 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/endnote163232 AcademicArticle DNA alkylation properties of yatakemycin 2003 10.1021/ja035984h 12952479 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote322034 AcademicArticle Mechanisms of in situ activation for DNA-targeting antitumor agents 2002 10.1021/cr010046q 12105933 http://vivo.scripps.edu/individual/endnote51983
http://vivo.scripps.edu/individual/endnote114633 AcademicArticle Intramolecular Diels-Alder and tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition reactions of 1,3,4-oxadiazoles 2002 10.1021/ja027533n 12236743 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote46956 AcademicArticle Total synthesis of anhydrolycorinone utilizing sequential intramolecular Diels-Alder reactions of a 1,3,4-oxadiazole 2002 10.1021/jo030437k 12375965 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote277003 AcademicArticle Metal cation complexation and activation of reversed CPyi analogues of CC-1065 and duocarmycin SA: Partitioning the effects of binding and catalysis 2001 10.1021/ja010769r 11562212 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote238936 AcademicArticle Combinatorial synthesis and discovery of an antibiotic compound - an experiment suitable for high school and undergraduate laboratories 2001 http://vivo.scripps.edu/individual/endnote193577
http://vivo.scripps.edu/individual/endnote182597 AcademicArticle Synthesis and evaluation of 1,2,8, 8a-Tetrahydrocyclopropa[c]pyrrolo[3,2-e]indol-4(5H)-one, the parent alkylation subunit of CC-1065 and the duocarmycins: impact of the alkylation subunit substituents and its implications for DNA alkylation catalysis 2000 10.1021/jo000297j 10866627 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote239483 AcademicArticle A new method of in situ activation for a novel class of DNA alkylating agents: tunable metal cation complexation and activation 2000 10.1021/ja000653f http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote123072 AcademicArticle Total synthesis of Amaryllidaceae alkaloids utilizing sequential intramolecular heterocyclic azadiene Diels-Alder reactions of an unsymmetrical 1,2,4,5-tetrazine 2000 10.1021/jo0012546 11149859 http://vivo.scripps.edu/individual/endnote171323

©2019 The Scripps Research Institute | Terms of Use | Powered by VIVO

  • About
  • Contact Us
  • Support