publication_uri | type | publication_title | year | doi | pmid | journal_uri |
http://vivo.scripps.edu/individual/e2n132419 | AcademicArticle | C1-CBP-vancomycin: Impact of a vancomycin C-terminus trimethylammonium cation on pharmacological properties and insights into its newly introduced mechanism of action | 2020 | 10.1021/acs.joc.9b02314 | 31670958 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/e2n371614 | AcademicArticle | Next-Generation Total Synthesis of Vancomycin | 2020 | 10.1021/jacs.0c07433 | 32885969 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n317190 | AcademicArticle | Precise Targeted Cleavage of a r(CUG) Repeat Expansion in Cells by Using a Small-Molecule-Deglycobleomycin Conjugate | 2020 | 10.1021/acschembio.0c00036 | http://vivo.scripps.edu/individual/endnote153903 | |
http://vivo.scripps.edu/individual/e2n108497 | AcademicArticle | Vancomycin C-Terminus Guanidine Modifications and Further Insights into an Added Mechanism of Action Imparted by a Peripheral Structural Modification | 2020 | 10.1021/acsinfecdis.0c00258 | 32598127 | http://vivo.scripps.edu/individual/e2n233249 |
http://vivo.scripps.edu/individual/e2n181332 | AcademicArticle | Total synthesis and stereochemical assignment of streptide | 2019 | 10.1021/jacs.9b09067 | 31577142 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n373958 | AcademicArticle | A small molecule drug conjugate (SMDC) of DUPA and a duocarmycin built on the solid phase | 2019 | 10.1039/c9md00279k | http://vivo.scripps.edu/individual/endnote55555 | |
http://vivo.scripps.edu/individual/e2n170510 | AcademicArticle | N-acyl pyrazoles: effective and tunable inhibitors of serine hydrolases | 2019 | 10.1016/j.bmc.2019.03.020 | 30879861 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/e2n319448 | AcademicArticle | Ultra-potent vinblastine analogues improve on-target activity of the parent microtubulin-targeting compound | 2019 | 10.1016/j.bmcl.2019.03.036 | 30952593 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n321823 | AcademicArticle | Triarylaminium radical cation promoted coupling of catharanthine with vindoline: diastereospecific synthesis of anhydrovinblastine and reaction scope | 2019 | 10.1021/jacs.9b06968 | 31442047 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n72523 | AcademicArticle | Exploration of the site-specific nature and generalizability of a trimethylammonium salt modification on vancomycin: A-ring derivatives | 2019 | 10.1016/j.tet.2019.02.008 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/e2n91509 | AcademicArticle | SAR studies of 4-acyl-1,6-dialkylpiperazin-2-one arenavirus cell entry inhibitors | 2019 | 10.1016/j.bmcl.2019.08.024 | 31537423 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n185220 | AcademicArticle | Resveratrol trimer enhances gene delivery to hematopoietic stem cells by reducing antiviral restriction at endosomes | 2019 | 10.1182/blood.2019000040 | 31416800 | http://vivo.scripps.edu/individual/endnote304227 |
http://vivo.scripps.edu/individual/e2n193601 | AcademicArticle | Structural basis of TLR2/TLR1 activation by the synthetic agonist diprovocim | 2019 | 10.1021/acs.jmedchem.8b01583 | 30829478 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e2n185787 | AcademicArticle | Inverse electron demand Diels-Alder reactions of heterocyclic azadienes, 1-aza-1,3-butadienes, cyclopropenone ketals and related systems. A retrospective | 2019 | 10.1021/acs.joc.9b00834 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e2n71244 | AcademicArticle | Synthesis, characterization, and rapid cycloadditions of 5-nitro-1,2,3-triazine | 2018 | 10.1021/acs.orglett.8b00825 | 29659291 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/e2n131232 | AcademicArticle | Diprovocims: A new and exceptionally potent class of toll-like receptor agonists | 2018 | 10.1021/jacs.8b09223 | 30272974 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n132606 | AcademicArticle | Duocarmycin SA, a potent antitumor antibiotic, sensitizes glioblastoma cells to proton radiation | 2018 | 10.1016/j.bmcl.2018.04.008 | 29650288 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n195020 | AcademicArticle | Adjuvant effect of the novel TLR1/TLR2 agonist Diprovocim synergizes with anti-PD-L1 to eliminate melanoma in mice | 2018 | 10.1073/pnas.1809232115 | 30150374 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/e2n54849 | AcademicArticle | High expression of class III β-tubulin has no impact on functional cancer cell growth inhibition of a series of key vinblastine analogs | 2018 | 10.1016/j.bmcl.2018.02.006 | 29439899 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n61286 | AcademicArticle | N-terminus alkylation of vancomycin: ligand binding affinity, antimicrobial activity, and site-specific nature of quaternary trimethylammonium salt modification | 2018 | 10.1021/acsinfecdis.8b00152 | 30067012 | http://vivo.scripps.edu/individual/e2n233249 |
http://vivo.scripps.edu/individual/e2n250703 | AcademicArticle | Peripheral modifications of [Ψ[CH2NH]Tpg4]vancomycin with added synergistic mechanisms of action provide durable and potent antibiotics | 2017 | 10.1073/pnas.1704125114 | 28559345 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/e2n251033 | AcademicArticle | Design of benzoxathiazin-3-one 1,1-dioxides as a new class of irreversible serine hydrolase inhibitors: Discovery of a uniquely selective PNPLA4 inhibitor | 2017 | 10.1021/jacs.7602985 | 28498651 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n143800 | AcademicArticle | Direct synthesis of β-aminoenals through reaction of 1,2,3-triazine with secondary amines | 2017 | 10.1021/acs.orglett.7b01543 | 28657329 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/e2n239190 | AcademicArticle | Vinblastine 20 ' amides: synthetic analogues that maintain or improve potency and simultaneously overcome Pgp-derived efflux and resistance | 2017 | 10.1021/acs.jmedchem.7b00958 | 28857558 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e2n261608 | AcademicArticle | The difference a single atom can make: synthesis and design at the chemistry-biology interface | 2017 | 10.1021/acs.joc.7b02088 | 28945374 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/e2n66041 | AcademicArticle | Total synthesis of a key series of vinblastines modified at C4 that define the importance and surprising trends in activity | 2017 | 10.1039/c6sc04146a | 28194270 | http://vivo.scripps.edu/individual/endnote149552 |
http://vivo.scripps.edu/individual/e2n61617 | AcademicArticle | Total syntheses of vancomycin-related glycopeptide antibiotics and key analogues | 2017 | 10.1021/acs.chemrev.6b00820 | 28437097 | http://vivo.scripps.edu/individual/endnote51983 |
http://vivo.scripps.edu/individual/e2n281853 | AcademicArticle | FAAH inhibitor OL-135 disrupts contextual, but not auditory, fear conditioning in rats | 2016 | 10.1016/j.bbr.2016.04.014 | 27083303 | http://vivo.scripps.edu/individual/endnote70642 |
http://vivo.scripps.edu/individual/e2n137683 | AcademicArticle | Synthesis of a potent vinblastine: rationally designed added benign complexity | 2016 | 10.1021/jacs.6b04330 | 27356080 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n144750 | AcademicArticle | Small-molecule fusion inhibitors bind the pH-sensing stable signal peptide-GP2 subunit interface of the Lassa virus Envelope glycoprotein | 2016 | 10.1128/jvi.00597-16 | 27194767 | http://vivo.scripps.edu/individual/endnote197644 |
http://vivo.scripps.edu/individual/e2n53616 | AcademicArticle | Synthesis and evaluation of duocarmycin SA analogs incorporating the methyl 1,2,8,8a-tetrahydrocyclopropa c imidazolo 4,5-e indol-4-one-6-carboxylat e (CImI) alkylation subunit | 2016 | 10.1016/j.bmc.2016.04.050 | 27221071 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/e2n122422 | AcademicArticle | TLR4/MD-2 activation by a synthetic agonist with no similarity to LPS | 2016 | 10.1073/pnas.1525639113 | 26831104 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/e2n330271 | AcademicArticle | Tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition cascade of 1,3,4-oxadiazoles: initial scope and applications | 2016 | 10.1021/acs.accounts.5b00510 | 26813287 | http://vivo.scripps.edu/individual/endnote122847 |
http://vivo.scripps.edu/individual/e2n254668 | AcademicArticle | Ultrapotent vinblastines in which added molecular complexity further disrupts the target tubulin dimer-dimer interface | 2016 | 10.1073/pnas.1611405113 | 27512044 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/e2n305180 | AcademicArticle | Catalysis of heterocyclic azadiene cycloaddition reactions by solvent hydrogen bonding: concise total synthesis of methoxatin | 2016 | 10.1021/jacs.6b05438 | 27571404 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n14106 | AcademicArticle | Discovery and structure-activity relationships of the neoseptins: a new class of toll-like receptor-4 (TLR4) agonists | 2016 | 10.1021/acs.jmedchem.6b00177 | 27050713 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e2n252643 | AcademicArticle | Total synthesis of (-)-vindoline and (+)-4-epi-vindoline based on a 1,3,4-oxadiazole tandem intramolecular 4+2 / 3+2 cycloaddition cascade initiated by an allene dienophile | 2015 | 10.1021/acs.orglett.5b02818 | 26457536 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/e2n330409 | AcademicArticle | A five-membered lactone prodrug of CBI-based analogs of the duocarmycins | 2015 | 10.1016/j.tetlet.2014.11.038 | 26069351 | http://vivo.scripps.edu/individual/endnote225462 |
http://vivo.scripps.edu/individual/e2n171836 | AcademicArticle | Comprehensive analysis of structure-activity relationships of a-ketoheterocycles as sn-1-diacylglycerol lipase a inhibitors | 2015 | 10.1021/acs.jmedchem.5b01627 | 26584396 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e2n330974 | AcademicArticle | Total synthesis of vinblastine, related natural products, and key analogues and development of inspired methodology suitable for the systematic study of their structure-function properties | 2015 | 10.1021/ar500400w | 25586069 | http://vivo.scripps.edu/individual/endnote122847 |
http://vivo.scripps.edu/individual/e2n98348 | AcademicArticle | Target-based screen against a periplasmic serine protease that regulates intrabacterial pH homeostasis in Mycobacterium tuberculosis | 2015 | 10.1021/cb500746z | 25457457 | http://vivo.scripps.edu/individual/endnote153903 |
http://vivo.scripps.edu/individual/e2n229404 | AcademicArticle | Total synthesis of (-)-kopsinine and ent-(+)-kopsinine | 2015 | 10.1016/j.tet.2014.07.094 | 26074629 | http://vivo.scripps.edu/individual/endnote9731 |
http://vivo.scripps.edu/individual/e2n267911 | AcademicArticle | Cycloadditions of 1,2,3-triazines bearing C5-electron donating substituents: robust pyrimidine synthesis | 2015 | 10.1021/acs.orglett.5b01870 | 26172042 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/e2n147302 | AcademicArticle | Total syntheses and initial evaluation of [?[C(-S)NH]Tpg(4)]vancomycin, [?[C(-NH)NH]Tpg(4)]vancomycin, [?[CH2NH]Tpg(4)]vancomycin, and their (4-Chlorobiphenyl)methyl derivatives: synergistic binding pocket and peripheral modifications for the glycopeptide antibiotics | 2015 | 10.1021/jacs.5b01008 | 25750995 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n173008 | AcademicArticle | Total synthesis of dihydrolysergic acid and dihydrolysergol: development of a divergent synthetic strategy applicable to rapid assembly of D-ring analogs | 2015 | 10.1016/j.tet.2015.05.093 | 26273113 | http://vivo.scripps.edu/individual/endnote9731 |
http://vivo.scripps.edu/individual/e2n309155 | AcademicArticle | When sugar is not so sweet | 2015 | 10.1126/science.aad3298 | http://vivo.scripps.edu/individual/endnote276633 | |
http://vivo.scripps.edu/individual/e10n5254 | AcademicArticle | Insights into the mechanism of streptonigrin-induced protein arginine deiminase inactivation | 2014 | 10.1016/j.bmc.2013.12.064 | 24440480 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/e11n218192 | AcademicArticle | Design, synthesis, and characterization of alpha-ketoheterocycles that additionally target the cytosolic port Cys269 of fatty acid amide hydrolase | 2014 | 10.1021/jm401820q | 24456116 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e11n28879 | AcademicArticle | Total syntheses of (-)-kopsifoline D and (-)-deoxoapodine: divergent total synthesis via late-stage key strategic bond formation | 2014 | 10.1021/ja500548e | 24499015 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e11n53454 | AcademicArticle | Total syntheses of (-)-pyrimidoblamic acid and P-3A | 2014 | 10.1021/ja412298c | 24410439 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e12n212983 | AcademicArticle | alpha-Ketoheterocycle inhibitors of fatty acid amide hydrolase: exploration of conformational constraints in the acyl side chain | 2014 | 10.1016/j.bmc.2014.03.013 | 24690529 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/e14n12278 | AcademicArticle | Enzymatic glycosylation of vancomycin aglycon: completion of a total synthesis of vancomycin and N- and C-terminus substituent effects of the aglycon substrate | 2014 | 10.1021/ol501568t | 24954524 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/e14n54464 | AcademicArticle | Discovery libraries targeting the major enzyme classes: the serine hydrolases | 2014 | 10.1016/j.bmcl.2014.06.063 | 25037918 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e14n33648 | AcademicArticle | Inhibition of adenovirus replication by a trisubstituted piperazin-2-one derivative | 2014 | 10.1016/j.antiviral.2014.05.010 | 24907427 | http://vivo.scripps.edu/individual/endnote251700 |
http://vivo.scripps.edu/individual/e2n259165 | AcademicArticle | Total synthesis of Psi C(=NH)NH Tpg(4) vancomycin and its ((4)-chlorobiphenyl)methyl derivative: impact of peripheral modifications on vancomycin analogues redesigned for dual D-Ala-D-Ala and D-Ala-D-Lac binding | 2014 | 10.1021/ja507009a | 25211770 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n187406 | AcademicArticle | Asymmetric synthesis of a CBI-based cyclic N-acyl O-amino phenol duocarmycin prodrug | 2014 | 10.1021/jo501839x | 25247380 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/e2n52915 | AcademicArticle | Cycloadditions of noncomplementary substituted 1,2,3-triazines | 2014 | 10.1021/ol502436n | 25222918 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/e1n6514 | AcademicArticle | A remarkable series of vinblastine analogues displaying enhanced activity and an unprecedented tubulin binding steric tolerance: C20' urea derivatives | 2013 | 10.1021/jm3015684 | 23244701 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e1n121557 | AcademicArticle | Rational design of fatty acid amide hydrolase inhibitors that act by covalently bonding to two active site residues | 2013 | 10.1021/ja4014997 | 23581831 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e3n124417 | AcademicArticle | Probing the role of the vancomycin E-ring aryl chloride: selective divergent synthesis and evaluation of alternatively substituted E-ring analogues | 2013 | 10.1021/jm4004494 | 23617725 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e3n283144 | AcademicArticle | Efficacious cyclic N-acyl O-amino phenol duocarmycin prodrugs | 2013 | 10.1021/jm400413r | 23627265 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/e4n127234 | AcademicArticle | NMR-assisted computational studies of peptidomimetic inhibitors bound in the hydrophobic pocket of HIV-1 glycoprotein 41 | 2013 | 10.1007/s10822-013-9662-6 | 23893342 | http://vivo.scripps.edu/individual/endnote51058 |
http://vivo.scripps.edu/individual/e4n287897 | AcademicArticle | Biological and structural evaluation of 10R- and 10S-methylthio-DDACTHF reveals a new role for sulfur in inhibition of glycinamide ribonucleotide transformylase | 2013 | 10.1021/bi4005182 | 23869564 | http://vivo.scripps.edu/individual/endnote165634 |
http://vivo.scripps.edu/individual/e4n72372 | AcademicArticle | Investigation into the functional impact of the vancomycin C-ring aryl chloride | 2013 | 10.1016/j.bmcl.2013.06.080 | 23880541 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e6n70136 | AcademicArticle | Transannular Diels-Alder/1,3-dipolar cycloaddition cascade of 1,3,4-oxadiazoles: total synthesis of a unique set of vinblastine analogues | 2013 | 10.1021/oI402549n | 24087969 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/e6n376933 | AcademicArticle | Potent vinblastine C20' ureas displaying additionally improved activity against a vinblastine-resistant cancer cell line | 2013 | 10.1021/ml400281w | 24223237 | http://vivo.scripps.edu/individual/endnote225139 |
http://vivo.scripps.edu/individual/e6n2464 | AcademicArticle | Evaluation of a reductively activated duocarmycin prodrug against murine and human solid cancers | 2013 | 10.4161/cbt.24348 | 23760495 | http://vivo.scripps.edu/individual/endnote374839 |
http://vivo.scripps.edu/individual/e8n253951 | AcademicArticle | A fundamental relationship between hydrophobic properties and biological activity for the duocarmycin class of DNA-alkylating antitumor drugs: hydrophobic-binding-driven bonding | 2013 | 10.1021/jm400665c | 23944748 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/enote10848 | AcademicArticle | A Pd(0)-mediated indole (macro)cyclization reaction | 2013 | 10.1021/ja3121394 | 23298368 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/enote337642 | AcademicArticle | Total synthesis of kopsinine | 2013 | 10.1021/ol303573f | 23391149 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/enote74874 | AcademicArticle | Total synthesis and evaluation of vinblastine analogues containing systematic deep-seated modifications in the vindoline subunit ring system: Core redesign | 2013 | 10.1021/jm3014376 | 23252481 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/enote245789 | AcademicArticle | Hypervalent iodine(III)-promoted intermolecular C-C coupling of vindoline with β-ketoesters and related substrates | 2013 | 10.1021/ol400135n | 23421318 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/enote202853 | AcademicArticle | A novel, unusually efficacious duocarmycin carbamate prodrug that releases no residual byproduct | 2012 | 10.1021/jm300330b | 22650244 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/enote26088 | AcademicArticle | Total synthesis of [Psi[C(═S)NH]Tpg4]vancomycin aglycon, [Psi[C(═NH)NH]Tpg4]vancomycin aglycon, and related key compounds: reengineering vancomycin for dual D-Ala-D-Ala and D-Ala-D-Lac binding | 2012 | 10.1021/ja209937s | 22188323 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/enote227473 | AcademicArticle | Fe(III)/NaBH4-mediated free radical hydrofluorination of unactivated alkenes | 2012 | 10.1021/ja3063716 | 22860624 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/enote308105 | AcademicArticle | The fatty acid amide hydrolase (FAAH) inhibitor PF-3845 acts in the nervous system to reverse LPS-induced tactile allodynia in mice | 2012 | 10.1111/j.1476-5381.2011.01445.x | 21506952 | http://vivo.scripps.edu/individual/endnote298379 |
http://vivo.scripps.edu/individual/enote47534 | AcademicArticle | New insights into the mechanism and an expanded scope of the Fe(III)-mediated vinblastine coupling reaction | 2012 | 10.1021/ja306229x | 22856867 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/enote11607 | AcademicArticle | Silver(I)-promoted conversion of thioamides to amidines: divergent synthesis of a key series of vancomycin aglycon residue 4 amidines that clarify binding behavior to model ligands | 2012 | 10.1021/ja302808p | 22568755 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/enote19581 | AcademicArticle | Divergent total syntheses of (-)-aspidospermine and (+)-spegazzinine | 2012 | 10.1021/ol300599p | 22480368 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/enote249169 | AcademicArticle | Iron(III)/NaBH4-mediated additions to unactivated alkenes: synthesis of novel 20'-vinblastine analogues | 2012 | 10.1021/ol300173v | 22369097 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/enote22938 | AcademicArticle | Discovery of HIV fusion inhibitors targeting gp41 using a comprehensive α-helix mimetic library | 2012 | 10.1016/j.bmcl.2012.02.062 | 22424973 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/enote194170 | AcademicArticle | α-Ketoheterocycle-based inhibitors of Fatty Acid Amide Hydrolase (FAAH) | 2012 | 10.1021/cn2001206 | 22639704 | http://vivo.scripps.edu/individual/endnote309398 |
http://vivo.scripps.edu/individual/enote97165 | AcademicArticle | Redesign of glycopeptide antibiotics: back to the future | 2012 | 10.1021/cb300007j | 22330049 | http://vivo.scripps.edu/individual/endnote153903 |
http://vivo.scripps.edu/individual/enote134419 | AcademicArticle | Comprehensive peptidomimetic libraries targeting protein-protein interactions | 2012 | 10.1021/ar300025n | 22799570 | http://vivo.scripps.edu/individual/endnote122847 |
http://vivo.scripps.edu/individual/e2n350794 | AcademicArticle | Tetrahedron Young Investigator Award 2011: Carolyn R. Bertozzi | 2011 | 10.1016/j.bmcl.2011.08.013 | 21840475 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/e2n169388 | AcademicArticle | Recent advances in medicinal chemistry | 2011 | 10.1016/j.bmcl.2011.04.019 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote198465 | AcademicArticle | Reversible competitive α-ketoheterocycle inhibitors of fatty acid amide hydrolase containing additional conformational constraints in the acyl side chain: orally active, long-acting analgesics | 2011 | 10.1021/jm101597x | 21428410 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote338926 | AcademicArticle | Scope of the inverse electron demand Diels-Alder reactions of 1,2,3-triazine | 2011 | 10.1021/ol2007428 | 21488676 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/endnote304212 | AcademicArticle | A redesigned vancomycin engineered for dual D-Ala-D-ala And D-Ala-D-Lac binding exhibits potent antimicrobial activity against vancomycin-resistant bacteria | 2011 | 10.1021/ja207142h | 21823662 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote18737 | AcademicArticle | Inverse electron demand Diels-Alder reactions of 1,2,3-triazines: Pronounced substituent effects on reactivity and cycloaddition scope | 2011 | 10.1021/ja204856a | 21736324 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote59552 | AcademicArticle | 10 '-fluorovinblastine and 10 '-fluorovincristine: synthesis of a key series of modified vinca alkaloids | 2011 | 10.1021/ml200236a | 22247789 | http://vivo.scripps.edu/individual/endnote225139 |
http://vivo.scripps.edu/individual/endnote93884 | AcademicArticle | Design, synthesis, and validation of a β-turn mimetic library targeting protein-protein and peptide-receptor interactions | 2011 | 10.1021/ja201878v | 21609016 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote167443 | AcademicArticle | The discovery and development of inhibitors of fatty acid amide hydrolase (FAAH) | 2011 | 10.1016/j.bmcl.2011.06.096 | 21764305 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote45392 | AcademicArticle | A specific interaction of small molecule entry inhibitors with the envelope glycoprotein complex of the Junin hemorrhagic fever arenavirus | 2011 | 10.1074/jbc.M110.196428 | 21159779 | http://vivo.scripps.edu/individual/endnote308813 |
http://vivo.scripps.edu/individual/endnote326586 | AcademicArticle | Asymmetric synthesis of 1,2,9,9a-tetrahydrocyclopropa[c]benzo[e]indol-4-one (CBI) | 2011 | 10.1021/jo102136w | 21192653 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote385145 | AcademicArticle | Synthesis and stereochemical determination of complestatin A and B (neuroprotectin A and B) | 2011 | 10.1021/ja208570q | 21991993 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote188397 | AcademicArticle | Fluoride-mediated capture of a noncovalent bound state of a reversible covalent enzyme inhibitor: X-ray crystallographic analysis of an exceptionally potent α-ketoheterocycle inhibitor of fatty acid amide hydrolase | 2011 | 10.1021/ja110877y | 21355555 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n63311 | Report | Optimization and characterization of a pan protein arginine deiminase (PAD) inhibitor | 2010 | 23833800 | http://vivo.scripps.edu/individual/e2n193384 | |
http://vivo.scripps.edu/individual/e7n125296 | AcademicArticle | Methods to characterize the effect of DNA-modifying compounds on nucleosomal DNA | 2010 | 10.1007/978-1-60327-418-0_11 | 19997884 | http://vivo.scripps.edu/individual/enote13799 |
http://vivo.scripps.edu/individual/endnote59228 | AcademicArticle | Total synthesis, assignment of the relative and absolute stereochemistry, and structural reassignment of phostriecin (aka Sultriecin) | 2010 | 10.1021/ja9097252 | 20108904 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote179882 | AcademicArticle | Intramolecular 1+2 and 3+2 cycloaddition reactions of cyclopropenone ketals | 2010 | 10.1021/ja103933n | 20527885 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote130386 | AcademicArticle | Total synthesis of (+)-fendleridine (aspidoalbidine) and (+)-1-acetylaspidoalbidine | 2010 | 10.1021/ja908819q | 20148585 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote116035 | AcademicArticle | Synthesis and evaluation of duocarmycin SA analogs incorporating the methyl 1,2,8,8a-tetrahydrocyclopropa[c]oxazolo[2,3-e]indol-4-one-6-carboxylate (COI) alkylation subunit | 2010 | 10.1016/j.bmcl.2010.01.145 | 20171886 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote27945 | AcademicArticle | Total synthesis and evaluation of a key series of C5-substituted vinblastine derivatives | 2010 | 10.1021/ja1027748 | 20518465 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote191718 | AcademicArticle | Fatty acid amide signaling molecules | 2010 | 10.1016/j.bmcl.2010.08.048 | 20817522 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote350214 | AcademicArticle | Synthesis and evaluation of selected key methyl ether derivatives of vancomycin aglycon | 2010 | 10.1021/jm100946e | 20853900 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote95806 | AcademicArticle | Identification of broad-based HIV-1 protease inhibitors from combinatorial libraries | 2010 | 10.1042/bj20091645 | 20507280 | http://vivo.scripps.edu/individual/endnote277207 |
http://vivo.scripps.edu/individual/endnote346786 | AcademicArticle | X-ray crystallographic analysis of alpha-ketoheterocycle inhibitors bound to a humanized variant of fatty acid amide hydrolase | 2010 | 10.1021/jm9012196 | 19924997 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote970 | AcademicArticle | Catharanthine C16 substituent effects on the biomimetic coupling with vindoline: preparation and evaluation of a key series of vinblastine analogues | 2010 | 10.1016/j.bmcl.2010.09.091 | 20932748 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote214314 | AcademicArticle | Synthesis and evaluation of a series of C5'-substituted duocarmycin SA analogs | 2010 | 10.1016/j.bmcl.2010.03.078 | 20381346 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote271946 | AcademicArticle | Total synthesis and evaluation of phostriecin and key structural analogues | 2010 | 10.1021/jo1010203 | 20669916 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote273289 | AcademicArticle | Asymmetric total synthesis of vindorosine, vindoline, and key vinblastine analogues | 2010 | 10.1021/ja106284s | 20809620 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote132574 | AcademicArticle | Total synthesis of lycogarubin C and lycogalic acid | 2010 | 10.1021/ol100146b | 20148525 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/endnote227188 | AcademicArticle | Asymmetric total synthesis of vindoline | 2010 | 10.1021/ja910695e | 20187641 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote207911 | AcademicArticle | Synthesis and characterization of a cyclobutane duocarmycin derivative incorporating the 1,2,10,11-tetrahydro-9H-cyclobuta[c]benzo[e]indol-4-one (CbBI) alkylation subunit | 2010 | 10.1021/ja106986f | 20839806 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote152852 | AcademicArticle | Small molecule peptidomimetic inhibitors of importin α/β mediated nuclear transport | 2010 | 10.1016/j.bmc.2010.08.038 | 20869252 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote345470 | AcademicArticle | Total synthesis of complestatin: development of a Pd(0)-mediated indole annulation for macrocyclization | 2010 | 10.1021/ja102304p | 20469945 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote12499 | AcademicArticle | Design, synthesis, and evaluation of duocarmycin O-amino phenol prodrugs subject to tunable reductive activation | 2010 | 10.1021/jm1010397 | 20942408 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote225419 | AcademicArticle | Intramolecular Diels-Alder reactions of cyclopropenone ketals | 2010 | 10.1021/ol101375a | 20614867 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/endnote70870 | AcademicArticle | Binding and inactivation mechanism of a humanized fatty acid amide hydrolase by alpha-ketoheterocycle inhibitors revealed from cocrystal structures | 2009 | 10.1021/ja902694n | 19722626 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote240008 | AcademicArticle | Synthesis and preliminary evaluation of duocarmycin analogues incorporating the 1,2,11,11a-tetrahydrocyclopropa c naphtho 2,3-e indol-4-one (CNI) and 1,2,11,11a-tetrahydrocyclopropa c naphtho 1,2-e indol-4-one (iso-CNI) alkylation subunits | 2009 | 10.1016/j.tet.2009.02.065 | 20161204 | http://vivo.scripps.edu/individual/endnote9731 |
http://vivo.scripps.edu/individual/endnote245024 | AcademicArticle | Total synthesis of chloropeptin II (complestatin) and chloropeptin I | 2009 | 10.1021/ja907193b | 19839632 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote168002 | AcademicArticle | Blockade of endocannabinoid-degrading enzymes attenuates neuropathic pain | 2009 | 10.1124/jpet.109.155465 | 19502530 | http://vivo.scripps.edu/individual/endnote398496 |
http://vivo.scripps.edu/individual/endnote330326 | AcademicArticle | Characterization of lassa virus cell entry inhibitors: Determination of the active enantiomer by asymmetric synthesis | 2009 | 10.1016/j.bmcl.2009.04.098 | 19428249 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote13131 | AcademicArticle | Structure-activity relationship studies of fostriecin, cytostatin, and key analogs, with PP1, PP2A, PP5, and( beta12-beta13)-chimeras (PP1/PP2A and PP5/PP2A), provide further insight into the inhibitory actions of fostriecin family inhibitors | 2009 | 10.1124/jpet.109.155630 | 19592665 | http://vivo.scripps.edu/individual/endnote398496 |
http://vivo.scripps.edu/individual/endnote178581 | AcademicArticle | Synthesis and evaluation of vancomycin aglycon analogues that bear modifications in the N-terminal D-leucyl amino acid | 2009 | 10.1021/jm801549b | 19209892 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote358052 | AcademicArticle | Synthesis of the chlorofusin cyclic peptide | 2009 | 10.1016/j.tet.2008.09.029 | 20047009 | http://vivo.scripps.edu/individual/endnote9731 |
http://vivo.scripps.edu/individual/endnote251334 | AcademicArticle | Functional and biochemical analysis of a key series of ramoplanin analogues | 2009 | 10.1016/j.bmcl.2009.09.001 | 19783144 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote247413 | AcademicArticle | Total synthesis and evaluation of iso-duocarmycin SA and iso-yatakemycin | 2009 | 10.1021/ja808108q | 19154178 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote98126 | AcademicArticle | Total synthesis of vinblastine, vincristine, related natural products, and key structural analogues | 2009 | 10.1021/ja809842b | 19292450 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote208457 | AcademicArticle | Design, synthesis, and evaluation of an α-helix mimetic library targeting protein-protein interactions | 2009 | 10.1021/ja810025g | 19334711 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote83423 | AcademicArticle | Total synthesis of vindoline and related alkaloids | 2009 | 10.5059/yukigoseikyokaishi.67.123 | http://vivo.scripps.edu/individual/endnote219041 | |
http://vivo.scripps.edu/individual/endnote207343 | AcademicArticle | Small molecule inhibitors of Myc/Max dimerization and Myc-induced cell transformation | 2009 | 10.1016/j.bmcl.2009.09.044 | 19800226 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote163987 | AcademicArticle | The isolation, total synthesis and structure elucidation of chlorofusin, a natural product inhibitor of the p53-mDM2 protein-protein interaction | 2009 | 10.1039/b821676b | 19642417 | http://vivo.scripps.edu/individual/endnote292459 |
http://vivo.scripps.edu/individual/endnote12643 | AcademicArticle | Discovery of inhibitors of aberrant gene transcription from libraries of DNA binding molecules: Inhibition of LEF-1-mediated gene transcription and oncogenic transformation | 2009 | 10.1021/ja809083d | 19216569 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote236543 | AcademicArticle | Evaluation of chlorofusin, its seven chromophore diastereomers, and key analogues | 2009 | 10.1016/j.tetlet.2009.01.081 | 20161293 | http://vivo.scripps.edu/individual/endnote225462 |
http://vivo.scripps.edu/individual/endnote308874 | AcademicArticle | Fundamental relationships between structure, reactivity, and biological activity for the duocarmycins and CC-1065 | 2009 | 10.1021/jm9006214 | 19639994 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote37487 | AcademicArticle | Synthesis and evaluation of a thio analogue of duocarmycin SA | 2009 | 10.1016/j.bmcl.2009.10.063 | 19879753 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote183205 | AcademicArticle | Endocannabinoid modulation of scratching response in an acute allergenic model: a new prospective neural therapeutic target for pruritus | 2009 | 10.1124/jpet.108.150136 | 19168707 | http://vivo.scripps.edu/individual/endnote398496 |
http://vivo.scripps.edu/individual/endnote310690 | AcademicArticle | CSI-FID: high throughput label-free detection of DNA binding molecules | 2009 | 10.1016/j.bmcl.2009.04.097 | 19435662 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote208131 | AcademicArticle | Direct coupling of catharanthine and vindoline to provide vinblastine: Total synthesis of (+)- and ent-(-)-vinblastine | 2008 | 10.1021/ja078192m | 18081297 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote164175 | AcademicArticle | Unique small molecule entry inhibitors of hemorrhagic fever arenaviruses | 2008 | 10.1074/jbc.M802089200 | 18474596 | http://vivo.scripps.edu/individual/endnote308813 |
http://vivo.scripps.edu/individual/endnote320240 | AcademicArticle | Structural features of the (+)-Yatakemycin/d(GACTAATTGAC)-(GTCAATTAGTC) complex: Quantum mechanical calculation of NMR parameters as a tool for the characterization of ligand/DNA Interactions | 2008 | 10.1002/ejoc.200701212 | http://vivo.scripps.edu/individual/endnote282598 | |
http://vivo.scripps.edu/individual/endnote230198 | AcademicArticle | Correlation of inhibitor effects on enzyme activity and thermal stability for the integral membrane protein fatty acid amide hydrolase | 2008 | 10.1016/j.bmcl.2008.06.086 | 18644727 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote9193 | AcademicArticle | Yatakemycin: Total synthesis, DNA alkylation, and biological properties | 2008 | 10.1039/b705665f | 18389136 | http://vivo.scripps.edu/individual/endnote292459 |
http://vivo.scripps.edu/individual/endnote277167 | AcademicArticle | Glycinamide ribonucleotide transformylase (GAR Tfase) as a target for cancer therapy | 2008 | 10.1358/dof.2008.33.11.1247542 | http://vivo.scripps.edu/individual/endnote288580 | |
http://vivo.scripps.edu/individual/endnote37163 | AcademicArticle | Disruption of the MYC transcriptional function by a small-molecule antagonist of MYC/MAX dimerization | 2008 | 18288422 | http://vivo.scripps.edu/individual/endnote100285 | |
http://vivo.scripps.edu/individual/endnote115125 | AcademicArticle | Optimization of the central heterocycle of alpha-ketoheterocycle inhibitors of fatty acid amide hydrolase | 2008 | 10.1021/jm800136b | 18630870 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote286204 | AcademicArticle | Asymmetric synthesis of inhibitors of glycinamide ribonucleotide transformylase | 2008 | 10.1021/jm800555h | 18686942 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote121561 | AcademicArticle | An additional spirocyclization for duocarmycin SA | 2008 | 10.1021/ja806593w | 19554689 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote184462 | AcademicArticle | Optimization of alpha-ketooxazole inhibitors of fatty acid amide hydrolase | 2008 | 10.1021/jm701210y | 18247553 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote371316 | AcademicArticle | Exploration of a fundamental substituent effect of α-ketoheterocycle enzyme inhibitors: Potent and selective inhibitors of fatty acid amide hydrolase | 2008 | 10.1016/j.bmcl.2008.06.084 | 18639454 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote59043 | AcademicArticle | Total synthesis of chlorofusin, its seven chromophore diastereomers, and key partial structures | 2008 | 10.1021/ja8012819 | 18712872 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote179836 | AcademicArticle | Structure-based design, synthesis, evaluation, and crystal structures of transition state analogue inhibitors of inosine monophosphate cyclohydrolase | 2007 | 10.1074/jbc.M607293200 | 17324932 | http://vivo.scripps.edu/individual/endnote308813 |
http://vivo.scripps.edu/individual/endnote267198 | AcademicArticle | Potent and selective alpha-ketoheterocycle-based inhibitors of the anandamide and oleamide catabolizing enzyme, fatty acid amide hydrolase | 2007 | 10.1021/jm0611509 | 17279740 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote62332 | AcademicArticle | Alanine scan of [L-Dap2]ramoplanin A2 aglycon: Assessment of the importance of each residue | 2007 | 10.1021/ja068573k | 17592838 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote198424 | AcademicArticle | Structure-activity relationships of alpha-ketooxazole inhibitors of fatty acid amide hydrolase | 2007 | 10.1021/jm061414r | 17559203 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote65252 | AcademicArticle | A unique class of duocarmycin and CC-1065 analogues subject to reductive activation | 2007 | 10.1021/ja075398e | 18020335 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote206989 | AcademicArticle | An in vitro and in vivo disconnect uncovered through high-throughput identification of botulinum neurotoxin A antagonists | 2007 | 10.1073/pnas.0611213104 | 17293454 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote324261 | AcademicArticle | Total synthesis, stereochemical reassignment, and absolute configuration of chlorofusin | 2007 | 10.1021/ja073264v | 17637057 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote200449 | AcademicArticle | Systematic exploration of the structural features of yatakemycin impacting DNA alkylation and biological activity | 2007 | 10.1021/ja072777z | 17691783 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote190245 | AcademicArticle | Total synthesis of (-)- and ent-(+)-4-desacetoxy-5-desethylvindoline | 2007 | 10.3987/COM-06-S(K)8 | http://vivo.scripps.edu/individual/endnote14559 | |
http://vivo.scripps.edu/individual/endnote337664 | AcademicArticle | Rational design, synthesis, and evaluation of key analogues of CC-1065 and the duocarmycins | 2007 | 10.1021/ja073989z | 17948994 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote258157 | AcademicArticle | Delineation of a fundamental alpha-ketoheterocycle substituent effect for use in the design of enzyme inhibitors | 2006 | 10.1021/ja064522b | 17061864 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote5493 | AcademicArticle | Total synthesis of (-)- and ent-(+)-vindorosine: Tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition of 1,3,4-oxadiazoles | 2006 | 10.1002/anie.200503024 | 16355429 | http://vivo.scripps.edu/individual/endnote319084 |
http://vivo.scripps.edu/individual/endnote244550 | AcademicArticle | Total synthesis of cytostatin | 2006 | 10.3987/COM-06-S(W)13 | http://vivo.scripps.edu/individual/endnote14559 | |
http://vivo.scripps.edu/individual/endnote182395 | AcademicArticle | Asymmetric total synthesis of (+)- and ent-(-)-yatakemycin and duocarmycin SA: evaluation of yatakemycin key partial structures and its unnatural enantiomer | 2006 | 10.1021/ja064228j | 17147378 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote203649 | AcademicArticle | Discovery of a potent, nonpolyglutamatable inhibitor of glycinamide ribonucleotide transformylase | 2006 | 10.1021/jm0601147 | 16686541 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote66316 | AcademicArticle | The mechanism of action of ramoplanin and enduracidin | 2006 | 10.1039/b515328j | 16880924 | http://vivo.scripps.edu/individual/endnote93661 |
http://vivo.scripps.edu/individual/endnote246390 | AcademicArticle | Total synthesis of (-)- and ent-(+)-vindoline and related alkaloids | 2006 | 10.1021/ja061256t | 16895428 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote206198 | AcademicArticle | Total synthesis and evaluation of [Ψ[CH(2)NH]Tpg(4)]vancomycin aglycon: reengineering vancomycin for dual D-Ala-D-Ala and D-Ala-D-Lac binding | 2006 | 10.1021/ja0572912 | 16506767 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote159164 | AcademicArticle | Diastereoselective Diels-Alder reactions of N-sulfonyl-1-aza-1,3-butadienes with optically active enol ethers: An asymmetric variant of the 1-azadiene Diels-Alder reaction | 2006 | 10.1021/ja0571646 | 16492042 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote17487 | AcademicArticle | Total synthesis of piericidin A1 and B1 and key analogues | 2006 | 10.1021/ja0632862 | 16953619 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote187884 | AcademicArticle | Alkylation of duplex DNA in nucleosome core particles by duocarmycin SA and yatakemycin | 2006 | 10.1038/nchembio761 | 16415862 | http://vivo.scripps.edu/individual/endnote16708 |
http://vivo.scripps.edu/individual/endnote19183 | AcademicArticle | Two novel 1,2,4,5-tetrazines that participate in inverse electron demand Diels-Alder reactions with an unexpected regioselectivity | 2006 | 10.1021/jo051832o | 16388634 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote394364 | AcademicArticle | Intramolecular Diels-Alder/1,3-dipolar cycloaddition cascade of 1,3,4-oxadiazoles | 2006 | 10.1021/ja0612549 | 16895427 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote19249 | AcademicArticle | Total synthesis and evaluation of cytostatin, its C10-C11 diastereomers, and additional key analogues: Impact on PP2A inhibition | 2006 | 10.1021/ja066477d | 17177422 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/e2n328144 | AcademicArticle | Bioorganic & Medicinal Chemistry Letters Symposia-in-Print | 2005 | 10.1016/j.bmcl.2005.07.002 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote136021 | AcademicArticle | Discovery of a potent, selective, and efficacious class of reversible alpha-ketoheterocycle inhibitors of fatty acid amide hydrolase effective as analgesics | 2005 | 10.1021/jm049614v | 15771430 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote120777 | AcademicArticle | Chemistry and biology of ramoplanin: A lipoglycodepsipeptide with potent antibiotic activity | 2005 | 10.1021/cr030106n | 15700952 | http://vivo.scripps.edu/individual/endnote51983 |
http://vivo.scripps.edu/individual/endnote258061 | AcademicArticle | Elucidation of fatty acid amide hydrolase inhibition by potent alpha-ketoheterocycle derivatives from Monte Carlo simulations | 2005 | 10.1021/ja055438j | 16332087 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote287545 | AcademicArticle | Design, synthesis, and biological evaluation of 10-methanesulfonyl-DDACTHF, 10-methanesulfonyl-5-DACTHF, and 10-methylthio-DDACTHF as potent inhibitors of GAR Tfase and the de novo purine biosynthetic pathway | 2005 | 10.1016/j.bmc.2004.12.004 | 15848770 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote289349 | AcademicArticle | Synthesis and biological evaluation of α- and γ-carboxamide derivatives of 10-CF3CO-DDACTHF | 2005 | 10.1016/j.bme.2004.11.050 | 15848771 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote125136 | AcademicArticle | Discovery of an exceptionally potent and selective class of fatty acid amide hydrolase inhibitors enlisting proteome-wide selectivity screening: concurrent optimization of enzyme inhibitor potency and selectivity | 2005 | 10.1016/j.bmcl.2004.12.085 | 15713400 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote67107 | AcademicArticle | Heterocyclic sulfoxide and sulfone inhibitors of fatty acid amide hydrolase | 2005 | 10.1016/j.bmcl.2004.10.025 | 15582420 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote92329 | AcademicArticle | Total synthesis of piericidin A1 and B1 | 2005 | 10.1021/ja055041f | 16277503 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote63204 | AcademicArticle | Discovery of aicar tfase inhibitors that disrupt requisite enzyme dimerization | 2005 | 10.1016/j.bcml.2005.03.094 | 15911265 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote50866 | AcademicArticle | Potent reversal of multidrug resistance by ningalins and its use in drug combinations against human colon carcinoma xenograft in nude mice | 2005 | 10.1007/s00280-005-1019-y | 15875185 | http://vivo.scripps.edu/individual/endnote235495 |
http://vivo.scripps.edu/individual/endnote291060 | AcademicArticle | Synthesis and biological evaluation of N-{4- 5-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-2-(2,2,2-trifluoro acetyl)pentyl)benzoyl}-L-glutamic acid as a potential inhibitor of GAR Tfase and the de novo purine biosynthetic pathway | 2005 | 10.1016/j.bme.2004.11.049 | 15848772 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote294251 | AcademicArticle | Total synthesis of (-)- and ent-(+)-vindoline | 2005 | 10.1021/o1051975x | 16178578 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/endnote238354 | AcademicArticle | Total synthesis of ningalin D | 2005 | 10.1021/ja0526416 | 16045367 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote251755 | AcademicArticle | Total synthesis of natural (-)- and ent-(+)-4-desacetoxy-6,7-dihydrovindorosine and natural and ent-minovine: Oxadiazole tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition reaction | 2005 | 10.1021/ol050017s | 15704939 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/endnote9036 | AcademicArticle | Sequence-selective DNA recognition: natural products and nature's lessons | 2004 | 10.1016/j.chembiol.2003.08.012 | 15610844 | http://vivo.scripps.edu/individual/endnote342045 |
http://vivo.scripps.edu/individual/endnote304860 | AcademicArticle | A fluorescent intercalator displacement assay for establishing DNA binding selectivity and affinity | 2004 | 10.1021/ar030113y | 14730995 | http://vivo.scripps.edu/individual/endnote122847 |
http://vivo.scripps.edu/individual/endnote144263 | AcademicArticle | A powerful selection assay for mixture libraries of DNA alkylating agents | 2004 | 10.1021/ja0477930 | 15281804 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote76671 | AcademicArticle | Total synthesis, structure revision, and absolute configuration of (+)-yatakemycin | 2004 | 10.1021/ja0472735 | 15237994 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote8937 | AcademicArticle | Total synthesis and examination of three key analogues of ramoplanin: a lipoglycodepsipeptide with potent antibiotic activity | 2004 | 10.1021/ja039671y | 14746470 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote282893 | AcademicArticle | Dissecting ramoplanin: mechanistic analysis of synthetic ramoplanin analogues as a guide to the design of improved antibiotics | 2004 | 10.1021/ja047879t | 15198592 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote79055 | AcademicArticle | A human single-chain antibody specific for integrin alpha(3)beta(1) capable of cell internalization and delivery of antitumor agents | 2004 | 10.1016/j.chembiol.2004.04.018 | 15271348 | http://vivo.scripps.edu/individual/endnote342045 |
http://vivo.scripps.edu/individual/endnote173920 | AcademicArticle | Establishing the parabolic relationship between reactivity and activity for derivatives and analogues of the duocarmycin and CC-1065 alkylation subunits | 2004 | 10.1021/ja038162t | 14709069 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote332968 | AcademicArticle | Reversible inhibitors of fatty acid amide hydrolase that promote analgesia: evidence for an unprecedented combination of potency and selectivity | 2004 | 10.1124/jpet.104.069401 | 15229230 | http://vivo.scripps.edu/individual/endnote398496 |
http://vivo.scripps.edu/individual/endnote310066 | AcademicArticle | Total synthesis and structure of the ramoplanin A1 and A3 aglycons: two minor components of the ramoplanin complex | 2004 | 10.1073/pnas.0401419101 | 15175429 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote267028 | AcademicArticle | Effective asymmetric synthesis of 1,2,9,9a-tetrahydrocyclopropa c benzo e indol-4-one (cbi) | 2004 | 10.1021/jo035465x | 15049620 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote296935 | AcademicArticle | Energetic preferences for alpha,beta versus beta,gamma unsaturation | 2004 | 10.1021/jo049365y | 15287795 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote288887 | AcademicArticle | Synthesis and evaluation of N-aryl and N-alkenyl CBI derivatives | 2004 | 10.1016/j.bmc.2004.08.032 | 15498660 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote231971 | AcademicArticle | Total synthesis of the ristocetin aglycon | 2004 | 10.1021/ja039795a | 15053621 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote301033 | AcademicArticle | Multidrug resistance reversal activity of permethyl ningalin B amide derivatives | 2004 | 10.1016/j.bmcl.2004.10.002 | 15546712 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote352787 | AcademicArticle | Synthesis of the chlorofusin cyclic peptide: assignment of the asparagine stereochemistry | 2003 | 10.1021/ol036083g | 14682761 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/endnote93713 | AcademicArticle | Comprehensive high-resolution analysis of hairpin polyamides utilizing a fluorescent intercalator displacement (FID) assay | 2003 | 10.1016/s0968-0896(03)00455-3 | 13129584 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote357622 | AcademicArticle | Synthesis and inverse electron demand Diels-Alder reactions of 3,6-bis(3,4-dimethoxybenzoyl)-1,2,4,5-tetrazine | 2003 | 10.1021/jo020713v | 12713365 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote35698 | AcademicArticle | Multidrug resistance reversal activity of key ningalin analogues | 2003 | 10.1016/s0960-894x(03)00294-4 | 12729663 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote62339 | AcademicArticle | 10-(2-benzoxazolcarbonyl)-5,10-dideaza-acyclic-5,6,7,8-tetrahydrofolic acid: a potential inhibitor of GAR transformylase and AICAR transformylase | 2003 | 10.1016/s0968-0896(03)00457-7 | 13129586 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote201679 | AcademicArticle | Synthesis of the (S,S,S)-diastereomer of the 15-membered biaryl ring system of RP 66453 | 2003 | 10.1016/s0040-4039(03)00856-6 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote160952 | AcademicArticle | NMR structure of the (+)-CPI-indole/d(GACTAATTGAC)-d(GTCAATTAGTC) covalent complex | 2003 | 10.1002/cbic.200300642 | 14613110 | http://vivo.scripps.edu/individual/e2n264100 |
http://vivo.scripps.edu/individual/endnote89489 | AcademicArticle | A new and improved method for deglycosidation of glycopeptide antibiotics exemplified with vancomycin, ristocetin, and ramoplanin | 2003 | 10.1016/s0960-894x(03)00051-9 | 12643936 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote108126 | AcademicArticle | High-resolution assessment of protein DNA binding affinity and selectivity utilizing a fluorescent intercalator displacement (FID) assay | 2003 | 10.1016/j.bmcl.2003.06.002 | 14552784 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote399934 | AcademicArticle | Synthesis of isochrysohermidin-distamycin hybrids | 2003 | 10.1021/jo034326c | 12816485 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote165310 | AcademicArticle | Synthesis and evaluation of methyl ether derivatives of the vancomycin, teicoplanin, and ristocetin aglycon methyl esters | 2003 | 10.1016/s0960-894x(03)00513-4 | 14611861 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote43335 | AcademicArticle | Determination of binding affinities of triplex forming oligonucleotides using a fluorescent intercalator displacement (FID) assay | 2003 | 10.1016/j.bmcl.2003.07.005 | 14552783 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote63515 | AcademicArticle | Solution-phase synthesis of combinatorial libraries designed to modulate protein-protein or protein-DNA interactions | 2003 | 10.1016/s0968-0896(03)00031-2 | 12659745 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote206837 | AcademicArticle | Discovering potent and selective reversible inhibitors of enzymes in complex proteomes | 2003 | 10.1038/nbt826 | 12740587 | http://vivo.scripps.edu/individual/endnote208688 |
http://vivo.scripps.edu/individual/endnote7829 | AcademicArticle | Fundamental role of the fostriecin unsaturated lactone and implications for selective protein phosphatase inhibition | 2003 | 10.1021/ja038672n | 14677930 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote210880 | AcademicArticle | Synthesis and X-ray analysis of an unprecedented and stable 2-aza-4,4-spirocyclopropacyclohexadienone | 2003 | 10.1021/ol035000t | 12841785 | http://vivo.scripps.edu/individual/endnote341245 |
http://vivo.scripps.edu/individual/endnote163232 | AcademicArticle | DNA alkylation properties of yatakemycin | 2003 | 10.1021/ja035984h | 12952479 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote147585 | AcademicArticle | Design, synthesis and biological evaluation of 10-CF3CO-DDACTHF analogues and derivatives as inhibitors of GAR Tfase and the de novo purine biosynthetic pathway | 2003 | 10.1016/s0968-0896(03)00458-9 | 13129587 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote292242 | AcademicArticle | Total synthesis of the ramoplanin a2 and ramoplanose aglycon | 2003 | 10.1021/ja0212314 | 12580615 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote275708 | AcademicArticle | Establishment of substituent effects in the DNA binding subunit of CBI analogues of the duocarmycins and CC-1065 | 2003 | 10.1016/s0968-0896(03)00194-9 | 12901927 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote180327 | AcademicArticle | Synthesis and evaluation of duocarmycin and CC-1065 analogues incorporating the 1,2,9,9a-tetrahydrocyclopropa c benz e -3-azaindol-4-one (CBA) alkylation subunit | 2003 | 10.1021/jo035119f | 14604371 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote172922 | AcademicArticle | Design, synthesis, and biological evaluation of simplified alpha-keto heterocycle, trifluoromethyl ketone, and formyl substituted folate analogues as potential inhibitors of GAR transformylase and AICAR transformylase | 2003 | 10.1016/s0968-0896(03)00456-5 | 13129585 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote359072 | AcademicArticle | Rational design, synthesis, evaluation, and crystal structure of a potent inhibitor of human GAR Tfase: 10-(trifluoroacetyl)-5,10-dideazaacyclic-5,6,7,8-tetrahydrofolic acid | 2003 | 10.1021/bi034219c | 12755606 | http://vivo.scripps.edu/individual/endnote165634 |
http://vivo.scripps.edu/individual/endnote79506 | AcademicArticle | Solution-phase combinatorial libraries: modulating cellular signaling by targeting protein-protein or protein-DNA interactions | 2003 | 10.1002/anie.200300574 | 14502729 | http://vivo.scripps.edu/individual/endnote319084 |
http://vivo.scripps.edu/individual/endnote331747 | AcademicArticle | Partitioning the loss in vancomycin binding affinity for D-Ala-D-Lac into lost H-bond and repulsive lone pair contributions | 2003 | 10.1021/ja035901x | 12889959 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote343214 | AcademicArticle | Small-molecule antagonists of Myc/Max dimerization inhibit Myc-induced transformation of chicken embryo fibroblasts | 2002 | 10.1073/pnas.062036999 | 11891322 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote4164 | AcademicArticle | Preparation of the 14-membered L,L-cycloisodityrosine subunit of RP 66453 | 2002 | 10.1016/s0040-4039(01)02194-3 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote262372 | AcademicArticle | Erythropoietin mimetics derived from solution phase combinatorial libraries | 2002 | 10.1021/ja0118789 | 11804483 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote94295 | AcademicArticle | Synthesis and DNA binding properties of iminodiacetic acid-linked polyamides: characterization of cooperative extended 2 : 1 side-by-side parallel binding | 2002 | 10.1021/ja026588m | 12207521 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote322034 | AcademicArticle | Mechanisms of in situ activation for DNA-targeting antitumor agents | 2002 | 10.1021/cr010046q | 12105933 | http://vivo.scripps.edu/individual/endnote51983 |
http://vivo.scripps.edu/individual/endnote109717 | AcademicArticle | Synthesis and evaluation of vancomycin and vancomycin aglycon analogues that bear modifications in the residue 3 asparagine | 2002 | 10.1016/s0960-894x(02)00130-0 | 11965380 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote317615 | AcademicArticle | Inhibitors of cell migration that inhibit intracellular paxillin/alpha a binding: A well-documented use of positional scanning libraries | 2002 | 10.1016/s1074-5521(02)00246-6 | 12445772 | http://vivo.scripps.edu/individual/endnote342045 |
http://vivo.scripps.edu/individual/endnote314513 | AcademicArticle | Solution-phase parallel synthesis of a pharmacophore library of hun-7293 analogues: a general chemical mutagenesis approach to defining structure-function properties of naturally occurring cyclic (depsi)peptides | 2002 | 10.1021/ja020166v | 11996584 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote276137 | AcademicArticle | Synthesis and DNA binding properties of saturated distamycin analogues | 2002 | 10.1016/s0960-894x(02)00467-5 | 12182879 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote73363 | AcademicArticle | Fostriecin: Chemistry and biology | 2002 | 12369868 | http://vivo.scripps.edu/individual/endnote178003 | |
http://vivo.scripps.edu/individual/endnote46956 | AcademicArticle | Total synthesis of anhydrolycorinone utilizing sequential intramolecular Diels-Alder reactions of a 1,3,4-oxadiazole | 2002 | 10.1021/jo030437k | 12375965 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote188582 | AcademicArticle | Total synthesis of the ramoplanin a2 and ramoplanose aglycon | 2002 | 10.1021/ja020237q | 11996568 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote114633 | AcademicArticle | Intramolecular Diels-Alder and tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition reactions of 1,3,4-oxadiazoles | 2002 | 10.1021/ja027533n | 12236743 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote384272 | AcademicArticle | Crystal structures of human GAR Tfase at low and high pH and with substrate β-GAR | 2002 | 10.1021/bi020522m | 12450384 | http://vivo.scripps.edu/individual/endnote165634 |
http://vivo.scripps.edu/individual/endnote268759 | AcademicArticle | The DNA phosphate backbone is not involved in catalysis of the duocarmycin and CC-1065 DNA alkylation reaction | 2002 | 10.1016/s0960-894x(01)00740-5 | 11814783 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote34329 | AcademicArticle | 10-formyl-5,10-dideaza-acyclic-5,6,7,8-tetrahydrofolic acid (10-formyl-DDACTHF): a potent cytotoxic agent acting by selective inhibition of human GAR Tfase and the de novo purine biosynthetic pathway | 2002 | 10.1016/s0968-0896(02)00102-5 | 12057663 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote41441 | AcademicArticle | Total synthesis of (+)-camptothecin | 2002 | 10.1016/s0040-4020(02)00633-6 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/endnote279320 | AcademicArticle | Hairpin versus extended DNA binding of a substituted beta-alanine linked polyamide | 2002 | 10.1021/ja0122039 | 11878968 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote21263 | AcademicArticle | Total syntheses of thiocoraline and be-22179 and assessment of their DNA binding and biological properties | 2001 | 10.1021/ja003602r | 11456568 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote121063 | AcademicArticle | Synthesis and evaluation of a series of C3-substituted CBI analogues of CC-1065 and the duocarmycins | 2001 | 10.1021/jo010309g | 11463270 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote384073 | AcademicArticle | Synthesis, chemical properties, and biological evaluation of CC-1065 and duocarmycin analogues incorporating the 5-methoxycarbonyl-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one alkylation subunit | 2001 | 10.1021/jo001772g | 11281757 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote203640 | AcademicArticle | Disruption of matrix metalloproteinase 2 binding to integrin alpha(v)beta(3) by an organic molecule inhibits angiogenesis and tumor growth in vivo | 2001 | 10.1073/pnas.011343298 | 11134507 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote249578 | AcademicArticle | Identification of a novel class of small-molecule antiangiogenic agents through the screening of combinatorial libraries which function by inhibiting the binding and localization of proteinase MMP2 to integrin alpha(V)beta(3) | 2001 | 10.1021/ja003579+ | 11456699 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote286887 | AcademicArticle | Alpha-Keto heterocycle inhibitors of fatty acid amide hydrolase: carbonyl group modification and alpha-substitution | 2001 | 10.1016/s0960-894x(01)00211-6 | 11412972 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote70838 | AcademicArticle | Substituent effects within the DNA binding subunit of CBI analogues of the duocarmycins and CC-1065 | 2001 | 10.1016/s0960-894x(01)00372-9 | 11454471 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote4989 | AcademicArticle | Thiazole orange as the fluorescent intercalator in a high resolution fid assay for determining DNA binding affinity and sequence selectivity of small molecules | 2001 | 10.1016/s0968-0896(01)00243-7 | 11553493 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote277003 | AcademicArticle | Metal cation complexation and activation of reversed CPyi analogues of CC-1065 and duocarmycin SA: Partitioning the effects of binding and catalysis | 2001 | 10.1021/ja010769r | 11562212 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote242915 | AcademicArticle | Cytokine receptor dimerization and activation: prospects for small molecule agonists | 2001 | 10.1016/s0968-0896(00)00276-5 | 11310589 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote225790 | AcademicArticle | Parallel synthesis and evaluation of 132 (+)-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (CBI) analogues of CC-1065 and the duocarmycins defining the contribution of the DNA-binding domain | 2001 | 10.1021/jo010454u | 11578217 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote138294 | AcademicArticle | A simple, high-resolution method for establishing DNA binding affinity and sequence selectivity | 2001 | 10.1021/ja010041a | 11414820 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote124062 | AcademicArticle | First and second generation total synthesis of the teicoplanin aglycon | 2001 | 10.1021/ja003835i | 11456806 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote111578 | AcademicArticle | Recent advances in bioorganic and medicinal chemistry. Preface. | 2001 | 10.1016/s0960-894x(01)00337-7 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote286284 | AcademicArticle | Vancomycin, teicoplanin, and ramoplanin: Synthetic and mechanistic studies | 2001 | 10.1002/med.1014 | 11579438 | http://vivo.scripps.edu/individual/endnote50744 |
http://vivo.scripps.edu/individual/endnote216314 | AcademicArticle | Asymmetric total synthesis of ent-(-)-roseophilin: Assignment of absolute configuration | 2001 | 10.1021/ja011271s | 11525659 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote128105 | AcademicArticle | Unexpected formation of an epoxide-derived multisubstrate adduct inhibitor on the active site of GAR transformylase | 2001 | 10.1021/bi011482+ | 11695901 | http://vivo.scripps.edu/individual/endnote165634 |
http://vivo.scripps.edu/individual/endnote47587 | AcademicArticle | Behavioral evidence for the interaction of oleamide with multiple neurotransmitter systems | 2001 | 11561096 | http://vivo.scripps.edu/individual/endnote398496 | |
http://vivo.scripps.edu/individual/endnote151661 | AcademicArticle | Alternative synthesis and thermal atropisomerism of a fully functionalized DEFG ring system of teicoplanin | 2001 | 10.1016/s0040-4039(01)01199-6 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote374953 | AcademicArticle | Total synthesis of fostriecin (CI-920) | 2001 | 10.1021/ja010195q | 11457179 | http://vivo.scripps.edu/individual/endnote181842 |
http://vivo.scripps.edu/individual/endnote89251 | AcademicArticle | Total syntheses of thiocoraline and be-22179: Establishment of relative and absolute stereochemistry | 2000 | 10.1021/ja0001660 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote182597 | AcademicArticle | Synthesis and evaluation of 1,2,8, 8a-Tetrahydrocyclopropa[c]pyrrolo[3,2-e]indol-4(5H)-one, the parent alkylation subunit of CC-1065 and the duocarmycins: impact of the alkylation subunit substituents and its implications for DNA alkylation catalysis | 2000 | 10.1021/jo000297j | 10866627 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote357589 | AcademicArticle | Development of a solution-phase synthesis of minor groove binding bis-intercalators based on triostin A suitable for combinatorial synthesis | 2000 | 10.1021/jo000382r | 10987932 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote116495 | AcademicArticle | Total synthesis of distamycin A and 2640 analogues: A solution-phase combinatorial approach to the discovery of new, bioactive DNA binding agents and development of a rapid, high-throughput screen for determining relative DNA binding affinity or DNA binding sequence selectivity | 2000 | 10.1021/ja994192d | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote151989 | AcademicArticle | Design, synthesis, and biological evaluation of fluoronitrophenyl substituted folate analogues as potential inhibitors of GAR transformylase and AICAR transformylase | 2000 | 10.1016/s0960-894x(00)00271-7 | 10888335 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote74082 | AcademicArticle | Exceptionally potent inhibitors of fatty acid amide hydrolase: the enzyme responsible for degradation of endogenous oleamide and anandamide | 2000 | 10.1073/pnas.97.10.5044 | 10805767 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote185537 | AcademicArticle | Total synthesis of the rubrolone aglycon | 2000 | 10.1021/ja002997b | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote265356 | AcademicArticle | Fatty acid amide hydrolase substrate specificity | 2000 | 10.1016/s0960-894x(00)00528-x | 11128635 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote129079 | AcademicArticle | Two comparisons of the performance of positional scanning and deletion synthesis for the identification of active constituents in mixture combinatorial libraries | 2000 | 10.1021/jo9916481 | 10814111 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote229545 | AcademicArticle | Assessment of solution-phase positional scanning libraries based on distamycin A for the discovery of new DNA binding agents | 2000 | 10.1016/s0968-0896(00)00137-1 | 11003149 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote266305 | AcademicArticle | Synthesis and evaluation of a novel bleomycin A(2) analogue: Continuing assessment of the linker domain | 2000 | 10.1016/s0040-4039(00)01633-6 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote217191 | AcademicArticle | Asymmetric synthesis of orthogonally protected L-threo-beta-hydroxyasparagine | 2000 | 10.1021/jo000628s | 11052134 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote317012 | AcademicArticle | A new class of highly cytotoxic diketopiperazines | 2000 | 10.1016/s0960-894x(00)00152-9 | 10843206 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote162686 | AcademicArticle | Selective metal cation activation of a DNA alkylating agent: Synthesis and evaluation of methyl 1,2,9,9a-Tetrahydrocyclopropa c pyrido 3,2-e indol-4-one-7-carboxylate (CPyl) | 2000 | 10.1021/jo000177b | 10866626 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote351894 | AcademicArticle | Conformationally restricted analogues designed for selective inhibition of GAR Tfase versus thymidylate synthase or dihydrofolate reductase | 2000 | 10.1016/s0968-0896(00)00051-1 | 10882019 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote20485 | AcademicArticle | The structural basis for in situ activation of DNA alkylation by duocarmycin sa | 2000 | 10.1006/jmbi.2000.3887 | 10903864 | http://vivo.scripps.edu/individual/endnote261742 |
http://vivo.scripps.edu/individual/endnote369655 | AcademicArticle | Thermal atropisomerism of teicoplanin aglycon derivatives: Preparation of the P,P,P and M,P,P atropisomers of the teicoplanin aglycon via selective equilibration of the DE ring system | 2000 | 10.1021/ja002376i | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote149655 | AcademicArticle | Bifunctional alkylating agents derived from duocarmycin SA: Potent antitumor activity with altered sequence selectivity | 2000 | 10.1016/s0960-894x(00)00042-1 | 10743956 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote233289 | AcademicArticle | Total synthesis of the teicoplanin aglycon | 2000 | 10.1021/ja001663j | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote176668 | AcademicArticle | Synthesis and evaluation of aza HUN-7293 | 2000 | 10.1016/s0960-894x(00)00336-x | 10937737 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote12566 | AcademicArticle | Total synthesis of ningalin B utilizing a heterocyclic azadiene Diels-Alder reaction and discovery of a new class of potent multidrug resistant (MDR) reversal agents | 2000 | 10.1021/jo9916535 | 10789460 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote123072 | AcademicArticle | Total synthesis of Amaryllidaceae alkaloids utilizing sequential intramolecular heterocyclic azadiene Diels-Alder reactions of an unsymmetrical 1,2,4,5-tetrazine | 2000 | 10.1021/jo0012546 | 11149859 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote239483 | AcademicArticle | A new method of in situ activation for a novel class of DNA alkylating agents: tunable metal cation complexation and activation | 2000 | 10.1021/ja000653f | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote112830 | AcademicArticle | Non-amide-based combinatorial libraries derived from N-BOC-iminodiacetic acid: solution-phase synthesis of piperazinone libraries with activity against LEF-1/β-catenin-mediated transcription | 2000 | 10.1002/1522-2675(20000809)83:8<1825::aid-hlca1825>3.0.co;2-4 | http://vivo.scripps.edu/individual/endnote350717 | |
http://vivo.scripps.edu/individual/endnote187932 | AcademicArticle | Total synthesis and comparative evaluation of luzopeptin A-C and quinoxapeptin A-C | 1999 | 10.1021/ja993019e | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote279965 | AcademicArticle | A novel class of CC-1065 and duocarmycin analogues subject to mitomycin-related reductive activation | 1999 | 10.1021/jo991301y | 11674758 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote348860 | AcademicArticle | Total synthesis of luzopeptins A-C | 1999 | 10.1021/ja983925b | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote225088 | AcademicArticle | CBI prodrug analogs of CC-1065 and the duocarmycins | 1999 | http://vivo.scripps.edu/individual/endnote215025 | ||
http://vivo.scripps.edu/individual/endnote353539 | AcademicArticle | Shape-dependent catalysis: Insights into the source of catalysis for the CC-1065 and duocarmycin DNA alkylation reaction | 1999 | 10.1021/ar9800946 | http://vivo.scripps.edu/individual/endnote122847 | |
http://vivo.scripps.edu/individual/endnote45497 | AcademicArticle | N-acylglycine amidation: implications for the biosynthesis of fatty acid primary amides | 1999 | 10.1021/bi982255j | 10079066 | http://vivo.scripps.edu/individual/endnote165634 |
http://vivo.scripps.edu/individual/endnote168914 | AcademicArticle | Total synthesis of quinoxapeptin A-C: Establishment of absolute stereochemistry | 1999 | 10.1002/(sici)1521-3773(19990816)38:16<2424::aid-anie2424>3.0.co;2-9 | 10458810 | http://vivo.scripps.edu/individual/endnote319084 |
http://vivo.scripps.edu/individual/endnote228432 | AcademicArticle | Total synthesis of the vancomycin aglycon | 1999 | 10.1021/ja992577q | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote176165 | AcademicArticle | Trifluoromethyl ketone inhibitors of fatty acid amide hydrolase: a probe of structural and conformational features contributing to inhibition | 1999 | 10.1016/s0960-894x(98)00734-3 | 10021942 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote377764 | AcademicArticle | Total synthesis of phomazarin | 1999 | 10.1021/ja983631q | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote184660 | AcademicArticle | Total synthesis of HUN-7293 | 1999 | 10.1021/ja990918u | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote170614 | AcademicArticle | Solution phase combinatorial synthesis of biaryl libraries employing heterogeneous conditions for catalysis and isolation with size exclusion chromatography for purification | 1999 | 10.1021/jo982234v | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote96922 | AcademicArticle | Resolution of a CPzl precursor, synthesis and biological evaluation of (+) and (-)-NBoc-CPzl: a further validation of the relationship between chemical solvolytic stability and cytotoxicity | 1999 | 10.1016/s0960-894x(99)00533-8 | 10560730 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote218088 | AcademicArticle | Arachidonic acid amide inhibitors of gap junction cell-cell communication | 1999 | 10.1016/s0960-894x(99)00148-1 | 10328303 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote341174 | AcademicArticle | Convergent solution-phase combinatorial synthesis with multiplication of diversity through rigid biaryl and diarylacetylene couplings | 1999 | 10.1021/jo990639p | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote247939 | AcademicArticle | Vancomycin CD and DE macrocyclization and atropisomerism studies | 1999 | 10.1021/jo980880o | 11674087 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote171910 | AcademicArticle | Are the duocarmycin and CC-1065 DNA alkylation reactions acid-catalyzed? Solvolysis pH-rate profiles suggest they are not | 1999 | 10.1021/jo990762g | 11674637 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote62791 | AcademicArticle | Diastereoselective total synthesis of the vancomycin aglycon with ordered atropisomer equilibrations | 1999 | 10.1021/ja990189i | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote35031 | AcademicArticle | Synthesis and evaluation of duocarmycin and CC-1065 analogues containing modifications in the subunit linking amide | 1999 | 10.1021/jo990452y | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote226505 | AcademicArticle | Binding-induced activation of DNA alkylation by duocarmycin SA: Insights from the structure of an indole derivative-DNA adduct | 1999 | 10.1021/ja983556j | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote72941 | AcademicArticle | Total syntheses of ningalin A, lamellarin O, lukianol A, and permethyl storniamide A utilizing heterocyclic azadiene Diels-Alder reactions | 1999 | 10.1021/ja982078+ | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote84645 | AcademicArticle | New insights into inhibitor design from the crystal structure and NMR studies of escherichia coli GAR and 10-formyl-5,8,10-trideazafolic acid | 1999 | 10.1021/bi991888a | 10606510 | http://vivo.scripps.edu/individual/endnote165634 |
http://vivo.scripps.edu/individual/endnote223713 | AcademicArticle | Bleomycin: synthetic and mechanistic studies | 1999 | 10.1002/(sici)1521-3773(19990215)38:4<448::aid-anie448>3.0.co;2-w | http://vivo.scripps.edu/individual/endnote319084 | |
http://vivo.scripps.edu/individual/endnote321743 | AcademicArticle | DNA binding properties of key sandramycin analogues: systematic examination of the intercalation chromophore | 1999 | 10.1016/s0968-0896(98)00206-5 | 10218823 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/e2n367672 | AcademicArticle | Combinatorial chemistry | 1998 | 10.1016/s0960-894x(98)90007-5 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/e7n84380 | AcademicArticle | The first synthesis of a daphnane diterpene: the enantiocontrolled total synthesis of (+)-resiniferatoxin | 1998 | http://vivo.scripps.edu/individual/e7n18490 | ||
http://vivo.scripps.edu/individual/endnote150799 | AcademicArticle | Thermal atropisomerism of aglucovancomycin derivatives: preparation of (M,M,M)- and (P,M,M)-aglucovancomycins | 1998 | 10.1021/ja981928i | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote398787 | AcademicArticle | Solution-phase combinatorial synthesis: Convergent multiplication of diversity via the olefin metathesis reaction | 1998 | 10.1016/s0040-4020(98)00128-8 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/endnote82992 | AcademicArticle | Synthesis of acyclic precursors to (3S,4S)-4-hydroxy-2,3,4,5-tetrahydro-pyridazine-3-carboxylic acid and incorporation into a luzopeptin/quinoxapeptin dipeptide | 1998 | 10.1021/jo980765d | 11672282 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote371226 | AcademicArticle | Heterocyclic and acyclic azadiene Diels-Alder reactions: total synthesis of nothapodytine B | 1998 | 10.1002/jhet.5570350502 | http://vivo.scripps.edu/individual/endnote355769 | |
http://vivo.scripps.edu/individual/endnote211351 | AcademicArticle | An endogenous sleep-inducing compound is a novel competitive inhibitor of fatty acid amide hydrolase | 1998 | 10.1016/s0960-894x(98)00073-0 | 9871570 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote322623 | AcademicArticle | Chemical requirements for inhibition of gap junction communication by the biologically active lipid oleamide | 1998 | 10.1073/pnas.95.9.4810 | 9560184 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote139070 | AcademicArticle | Higher order iminodiacetic acid libraries for probing protein-protein interactions | 1998 | 10.1016/s0960-894x(98)00423-5 | 9873538 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote3246 | AcademicArticle | Design, synthesis, and evaluation of potential GAR and AICAR transformylase inhibitors | 1998 | 10.1016/s0968-0896(98)00040-6 | 9681131 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote233392 | AcademicArticle | Synthesis and evaluation of a carbocyclic analogue of the CC-1065 and duocarmycin alkylation subunits: role of the vinylogous amide and implications on DNA alkylation catalysis | 1998 | 10.1021/jo981698q | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote195891 | AcademicArticle | Synthesis of the vancomycin CDE ring system | 1998 | 10.1016/s0960-894x(98)00110-3 | 9871529 | http://vivo.scripps.edu/individual/endnote119710 |
http://vivo.scripps.edu/individual/endnote103386 | AcademicArticle | Regioselective inverse electron demand Diels-Alder reactions of N-acyl 6-amino-3-(methylthio)-1,2,4,5-tetrazines | 1998 | 10.1021/jo980795g | 11672266 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote240228 | AcademicArticle | NMR studies of Co.deglycoBleomycin A2 green and its complex with d(CCAGGCCTGG) | 1998 | 10.1021/ja972125i | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote282523 | AcademicArticle | Assessment of the role of the bleomycin A(2) pyrimidoblamic acid C4 amino group | 1998 | 10.1021/ja971889v | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote258490 | AcademicArticle | Critical role of the linking amide in CC-1065 and the duocarmycins: implications on the source of DNA alkylation catalysis | 1998 | 10.1021/ja9818093 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote249563 | AcademicArticle | Structural requirements for 5-HT2A and 5-HT1A serotonin receptor potentiation by the biologically active lipid oleamide | 1998 | 10.1073/pnas.95.8.4102 | 9539697 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote216022 | AcademicArticle | Synthesis of key sandramycin analogs: Systematic examination of the intercalation chromophore | 1998 | 10.1016/s0968-0896(97)10014-1 | 9502108 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote312787 | AcademicArticle | Definition of the effect and role of the bleomycin A(2) valerate substituents: preorganization of a rigid, compact conformation implicated in sequence-selective DNA cleavage | 1998 | 10.1021/ja9816640 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote25122 | AcademicArticle | A systematic evaluation of the bleomycin A(2) L-threonine side chain: its role in preorganization of a compact conformation implicated in sequence-selective DNA cleavage | 1998 | 10.1021/ja9816638 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote140851 | AcademicArticle | Oleamide: an endogenous sleep-inducing lipid and prototypical member of a new class of biological signaling molecules | 1998 | 10197045 | http://vivo.scripps.edu/individual/endnote248220 | |
http://vivo.scripps.edu/individual/endnote196859 | AcademicArticle | Higher order iminodiacetic acid libraries for probing protein-protein interactions | 1998 | 10.1016/s0968-0896(98)00128-x | 9784874 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote164535 | AcademicArticle | Synthesis of CC-1065 and duocarmycin analogs via intramolecular aryl radical cyclization of a tethered vinyl chloride | 1998 | 10.1016/s0040-4039(98)00232-9 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote388085 | AcademicArticle | Multistep convergent solution-phase combinatorial synthesis and deletion synthesis deconvolution | 1998 | 10.1021/ja9803557 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote47504 | AcademicArticle | Total synthesis of nothapodytine B and (-)-mappicine | 1998 | 10.1021/ja973007y | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/e7n368030 | AcademicArticle | Solution structures of Co·Bleomycin A2 green and its complex with d(CCAGGCCTGG)2 | 1997 | http://vivo.scripps.edu/individual/e7n18490 | ||
http://vivo.scripps.edu/individual/endnote63378 | AcademicArticle | Total synthesis of (+)-duocarmycin A, epi-(+)-duocarmycin A and their unnatural enantiomers: assessment of chemical and biological properties | 1997 | 10.1021/ja962431g | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote9779 | AcademicArticle | pH dependence of the rate of DNA alkylation for (+)-duocarmycin SA and (+)-CCBI-TMI | 1997 | 10.1016/s0960-894x(96)00605-1 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote351599 | AcademicArticle | Applications of free radicals in organic synthesis | 1997 | http://vivo.scripps.edu/individual/endnote235588 | ||
http://vivo.scripps.edu/individual/endnote57934 | AcademicArticle | Determination of the relative and absolute stereochemistry of fostriecin (CL-920) | 1997 | 10.1021/jo962166h | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote343313 | AcademicArticle | CC-1065/duocarmycin and bleomycin A(2) hybrid agents: lack of enhancement of DNA alkylation by attachment to noncomplementary DNA binding subunits | 1997 | 10.1016/s0968-0896(96)00237-4 | 9061188 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote267204 | AcademicArticle | Preparation and inverse electron demand diels-alder reactions of 3-methoxy-6-methylthio-1,2,4,5-tetrazine | 1997 | 10.1016/s0040-4039(97)00751-x | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote46694 | AcademicArticle | Solution-phase combinatorial synthesis via the olefin metathesis reaction | 1997 | 10.1016/s0960-894x(97)00043-7 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote17378 | AcademicArticle | 10-formyl-5,8,10-trideazafolic acid (10-formyl-TDAF): a potent inhibitor of glycinamide ribonucleotide transformylase | 1997 | 10.1016/s0968-0896(97)00120-x | 9354237 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote168316 | AcademicArticle | Multisubstrate analogue based on 5,8,10-trideazafolate | 1997 | 10.1016/s0968-0896(97)00124-7 | 9354241 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote266407 | AcademicArticle | Synthesis and evaluation of CC-1065 and duocarmycin analogues incorporating the iso-CI and iso-CBI alkylation subunits: impact of relocation of the C-4 carbonyl | 1997 | 10.1021/jo971686p | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote72606 | AcademicArticle | Synthesis of (9R,12S)- and (9S,12S)-cycloisodityrosine and their N-methyl derivatives | 1997 | 10.1021/jo961346o | 11671510 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote228294 | AcademicArticle | Abenzyl 10-formyl-trideazafolic acid (abenzyl 10-formyl-TDAF): an effective inhibitor of glycinamide ribonucleotide transformylase | 1997 | 10.1016/s0968-0896(97)00123-5 | 9354240 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote170972 | AcademicArticle | Catalysis of the CC-1065 and duocarmycin DNA alkylation reaction: DNA binding induced conformational change in the agent results in activation | 1997 | 10.1016/s0968-0896(96)00238-6 | 9061191 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote347473 | AcademicArticle | Synthesis of the vancomycin CD and DE ring systems | 1997 | 10.1021/jo970560p | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote396213 | AcademicArticle | An exceptionally potent analog of sandramycin | 1997 | 10.1016/s0960-894x(97)00129-7 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote265865 | AcademicArticle | N-methyl threonine analogues of deglycobleomycin A(2): Synthesis and evaluation | 1997 | 10.1016/s0968-0896(97)00107-7 | 9313863 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote122835 | AcademicArticle | Duocarmycin SA shortened, simplified, and extended agents: A systematic examination of the role of the DNA binding subunit | 1997 | 10.1021/ja9637208 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote322661 | AcademicArticle | CC-1065 and the duocarmycins: Synthetic studies | 1997 | 10.1021/cr960095g | 11848889 | http://vivo.scripps.edu/individual/endnote51983 |
http://vivo.scripps.edu/individual/endnote129480 | AcademicArticle | Functionalized analogues of 5,8,10-trideazafolate: Development of an enzyme-assembled tight binding inhibitor of GAR Tfase and a potential irreversible inhibitor of AICAR Tfase | 1997 | 10.1016/s0968-0896(97)00122-3 | 9354239 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote22856 | AcademicArticle | High resolution solution structure of a DNA duplex alkylated by the antitumor agent duocarmycin SA | 1997 | 10.1006/jmbi.1997.1223 | 9299351 | http://vivo.scripps.edu/individual/endnote261742 |
http://vivo.scripps.edu/individual/endnote395585 | AcademicArticle | Functionalized analogues of 5,8,10-trideazafolate as potential inhibitors of gar tfase or aicar tfase | 1997 | 10.1016/s0968-0896(97)00121-1 | 9354238 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote270306 | AcademicArticle | The sleep-inducing lipid oleamide deconvolutes gap junction communication and calcium wave transmission in glial cells | 1997 | 10.1083/jcb.139.7.1785 | 9412472 | http://vivo.scripps.edu/individual/endnote322298 |
http://vivo.scripps.edu/individual/endnote52885 | AcademicArticle | Synthesis and evaluation of CC-1065 and duocarmycin analogs incorporating the 1,2,3,4,11,11a-hexahydrocyclopropa c naphtho 2,1-b azepin-6-one (CNA) alkylation subunit: Structural features that govern reactivity and reaction regioselectivity | 1997 | 10.1021/jo9707085 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote180172 | AcademicArticle | Thermal atropisomerism of fully functionalized vancomycin CD, DE, and CDE ring systems | 1997 | 10.1016/s0960-894x(97)10182-2 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote122948 | AcademicArticle | Asymmetric synthesis of the CBI alkylation subunit of the CC-1065 and duocarmycin analogs | 1997 | http://vivo.scripps.edu/individual/endnote302592 | ||
http://vivo.scripps.edu/individual/endnote183242 | AcademicArticle | Reversed and sandwiched analogs of duocarmycin SA: Establishment of the origin of the sequence-selective alkylation of DNA and new insights into the source of catalysis | 1997 | 10.1021/ja9637210 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote203700 | AcademicArticle | Generation of targeted C-2-symmetrical compound libraries by solution-phase combinatorial chemistry | 1997 | 10.1016/s0960-894x(97)00330-2 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/e2n232667 | AcademicArticle | Editorial | 1996 | 10.1016/s0960-894x(96)90241-3 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/e7n301280 | AcademicArticle | Cycloaddition reactions of azadienes, cyclopropenone ketals, and related systems: scope and applications | 1996 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/e7n121566 | AcademicArticle | Alternative synthesis of the cycloisodityrosine subunit of deoxybouvardin, RA-VII, and related agents: reassignment of the stereochemistry of prior intermediates | 1996 | 10.1021/jo9604144 | 11667262 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/e7n289723 | AcademicArticle | Control of chemoselectivity in catalytic rhodium carbenoid reactions through ligand modification. Comments | 1996 | http://vivo.scripps.edu/individual/e7n180816 | ||
http://vivo.scripps.edu/individual/endnote220512 | AcademicArticle | A comparative study of the solvolysis reactivity, regioselectivity, and stereochemistry of the duocarmycin A and SA alkylation subunits | 1996 | 10.1016/0960-894x(96)00346-0 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote339406 | AcademicArticle | Synthesis, chemical properties, and preliminary evaluation of substituted CBI analogs of CC-1065 and the duocarmycins incorporating the 7-cyano-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one alkylation subunit: Hammett quantitation of the magnitude of electronic effects on functional reactivity | 1996 | 10.1021/jo9605298 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote117425 | AcademicArticle | Molecular characterization of an enzyme that degrades neuromodulatory fatty-acid amides | 1996 | 10.1038/384083a0 | 8900284 | http://vivo.scripps.edu/individual/endnote351395 |
http://vivo.scripps.edu/individual/endnote360112 | AcademicArticle | Structure determination of an endogenous sleep-inducing lipid, cis-9-octadecenamide (oleamide): A synthetic approach to the chemical analysis of trace quantities of a natural product | 1996 | 10.1021/ja9532345 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote187755 | AcademicArticle | Demonstration and definition of the noncovalent binding selectivity of agents related to CC-1065 by an affinity cleavage agent: Noncovalent binding coincidental with alkylation | 1996 | 10.1016/0968-0896(96)00073-9 | 8818235 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote182195 | AcademicArticle | Examination of the role of the duocarmycin SA methoxy substituents: Identification of the minimum, fully potent DNA binding subunit | 1996 | 10.1016/0960-894x(96)00401-5 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote19802 | AcademicArticle | Inhibition of oleamide hydrolase catalyzed hydrolysis of the endogenous sleep-inducing lipid cis-9-octadecenamide | 1996 | 10.1021/ja954064z | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote26390 | AcademicArticle | CC-1065 and the duocarmycins: understanding their biological function through mechanistic studies | 1996 | 10.1002/anie.199614381 | http://vivo.scripps.edu/individual/endnote319084 | |
http://vivo.scripps.edu/individual/endnote63617 | AcademicArticle | Synthesis of (9S,12S)-cycloisodityrosine and its unnatural (9R,12S)-diastereomer | 1996 | 10.1016/0960-894x(96)00179-5 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote30964 | AcademicArticle | (-)-Sandramycin: total synthesis and characterization of DNA binding properties | 1996 | 10.1021/ja952799y | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote238056 | AcademicArticle | Novel solution phase strategy for the synthesis of chemical libraries containing small organic molecules | 1996 | 10.1021/ja9530681 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote137025 | AcademicArticle | Key analogues of the tetrapeptide subunit of RA-VII and deoxybouvardin | 1996 | 10.1016/0968-0896(96)00151-4 | 8931929 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote172529 | AcademicArticle | Synthesis and evaluation of deglycobleomycin A(2) analogues containing a tertiary N-methyl amide and simple ester replacement for the L-histidine secondary amide: Direct functional characterization of the requirement for secondary amide metal complexation | 1996 | 10.1016/0968-0896(95)00183-2 | 8814877 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote18327 | AcademicArticle | Synthesis and evaluation of potential N-pi and N-sigma metal chelation sites within the beta-hydroxy-L-histidine subunit of bleomycin A(2): Functional characterization of imidazole N-pi metal complexation | 1996 | 10.1016/0968-0896(95)00184-0 | 8814878 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote394540 | AcademicArticle | A solution-phase strategy for the synthesis of chemical libraries containing small organic molecules: a universal and dipeptide mimetic template | 1996 | 10.1016/0968-0896(96)00069-7 | 8804539 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote289638 | AcademicArticle | Synthesis, X-ray structure, and properties of fluorocyclopropane analogs of the duocarmycins incorporating the 9,9-difluoro-1,2,9,9a-tetrahydrocyclopropa c benzo e indol-4-one (F2CBI) alkylation subunit | 1996 | 10.1021/ja961888n | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote29742 | AcademicArticle | Azadiene Diels-Alder reactions: scope and applications. Total synthesis of natural and ent-fredericamycin A | 1996 | 10.1002/jhet.5570330508 | http://vivo.scripps.edu/individual/endnote355769 | |
http://vivo.scripps.edu/individual/endnote307756 | AcademicArticle | Synthesis of (r)-(4-methoxy-3,5-dihydroxyphenyl)glycine derivatives: The central amino acid of vancomycin and related agents | 1996 | 10.1021/jo960085f | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote267683 | AcademicArticle | Enantioselective total synthesis of (+)-duocarmycin A, epi-(+)-duocarmycin a, and their unnatural enantiomers | 1996 | 10.1021/ja953777e | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote202999 | AcademicArticle | Generalized dipeptidomimetic template: solution phase parallel synthesis of combinatorial libraries | 1996 | 10.1021/ja9539711 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote82719 | AcademicArticle | Synthesis and properties of substituted CBI analogs of CC-1065 and the duocarmycins incorporating the 7-methoxy-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (MCBI) alkylation subunit: magnitude of electronic effects on the functional reactivity | 1996 | 10.1021/jo952033g | 11667041 | http://vivo.scripps.edu/individual/endnote171323 |
http://vivo.scripps.edu/individual/endnote149972 | AcademicArticle | A Hammett correlation for CC-1065 and duocarmycin analogs: magnitude of substituent electronic effects on functional reactivity | 1996 | 10.1016/0960-894x(96)00093-5 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/e7n179688 | AcademicArticle | Total synthesis of (+)- and ent-(-)-duocarmycin SA | 1995 | http://vivo.scripps.edu/individual/e7n257080 | ||
http://vivo.scripps.edu/individual/endnote180960 | AcademicArticle | A modified friedlander condensation for the synthesis of 3-hydroxyquinoline-2-carboxylates | 1995 | 10.1021/jo00127a055 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote322928 | AcademicArticle | CC-1065 CBI analogs - an example of enhancement of DNA alkylation efficiency through introduction of stabilizing electrostatic interactions | 1995 | 10.1016/0968-0896(95)00048-l | 7582940 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote329599 | AcademicArticle | Diastereoselective dieckmann condensation suitable for introduction of the duocarmycin A C6 center - development of a divergent strategy for the total synthesis of duocarmycins A and SA | 1995 | 10.1016/0968-0896(94)00147-u | 8612048 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote183158 | AcademicArticle | An unusually facile SNAr 14-membered biaryl ether macrocyclization reaction suitable for preparation of the cycloisodityrosine subunit of bouvardin, deoxybouvardin and related agents | 1995 | 10.1016/0960-894x(95)00192-v | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote343252 | AcademicArticle | Chemical characterization of a family of brain lipids that induce sleep | 1995 | 10.1126/science.7770779 | 7770779 | http://vivo.scripps.edu/individual/endnote276633 |
http://vivo.scripps.edu/individual/endnote132861 | AcademicArticle | Key synthetic analogs of bleomycin A(2) that directly address the effect and role of the disaccharide - demannosylbleomycin A(2) and alpha-D-mannopyranosyldeglycobleomycin A(2) | 1995 | 10.1021/ja00133a008 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote142239 | AcademicArticle | Key analogs of the tetrapeptide subunit of RA-VII and deoxybouvardin | 1995 | 10.1016/0968-0896(95)00141-7 | 8770383 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote367504 | AcademicArticle | CBI-CDPBO1 and CBI-CDPBI1 - CC-1065 analogs containing deep-seated modifications in the DNA-binding subunit | 1995 | 10.1016/0968-0896(95)00066-p | 7582954 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote245376 | AcademicArticle | Second definitive test of proposed models for the origin of the CC-1065 and duocarmycin DNA alkylation selectivity | 1995 | 10.1021/ja00109a035 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote121527 | AcademicArticle | An efficient synthesis of 1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (CBI) - an enhanced and simplified analog of the CC-1065 and duocarmycin alkylation subunits | 1995 | 10.1021/jo00110a034 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote247922 | AcademicArticle | DNA alkylation properties of CC-1065 and duocarmycin analogs incorporating the 2,3,10,10a-tetrahydrocyclopropa d benzo f quinol-5-one alkylation subunit - identification of subtle structural features that contribute to the regioselectivity of the adenine N3 alkylation reaction | 1995 | 10.1021/ja00152a004 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote211094 | AcademicArticle | Synthesis and evaluation of the fully functionalized bleomycin A(2) metal-binding domain-containing the 2-O-(3-O-carbamoyl-alpha-D-mannopyranosyl)-alpha-L-gulopyranosyl disaccharide | 1995 | 10.1021/ja00133a007 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote347005 | AcademicArticle | Total synthesis of natural and ent-fredericamycin-a | 1995 | 10.1021/ja00153a004 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote353147 | AcademicArticle | 1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one (CBI) analogs of CC-1065 and the duocarmycins: synthesis and evaluation | 1995 | 10.1016/0968-0896(95)00130-9 | 8634824 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote42726 | AcademicArticle | CC-1065 and the duocarmycins - unraveling the keys to a new class of naturally derived DNA alkylating-agents | 1995 | 10.1073/pnas.92.9.3642 | 7731958 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote3861 | AcademicArticle | Synthesis of key analogs of bleomycin A(2) that permit a systematic evaluation of the linker region - identification of an exceptionally prominent role for the L-threonine substituent | 1995 | 10.1016/0968-0896(95)00113-u | 8564421 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote374345 | AcademicArticle | N-desmethyl derivatives of deoxybouvardin and RA-VII: synthesis and evaluation | 1995 | 10.1021/ja00133a010 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote54399 | AcademicArticle | The duocarmycins: synthetic and mechanistic studies | 1995 | 10.1021/ar00049a004 | http://vivo.scripps.edu/individual/endnote122847 | |
http://vivo.scripps.edu/individual/endnote395760 | AcademicArticle | Solution-phase conformational studies of the cyclic peptide RA-VII: lithium-chloride perturbation of the conformational equilibria | 1995 | 10.1021/ja00133a009 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote239998 | AcademicArticle | Total synthesis of granditropone, grandirubrine, imerubrine, and isoimerubrine | 1995 | 10.1021/ja00155a009 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote114077 | AcademicArticle | Synthesis of appropriately functionalized vancomycin CD and DE ring systems | 1995 | 10.1016/0960-894x(95)00543-9 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/e7n266715 | AcademicArticle | Design, synthesis and evaluation of bouvardin, deoxybouvardin and RA-I-XIV pharmacophore analogs | 1994 | 10.1016/s0968-0896(00)82005-2 | 7922127 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/e7n387665 | AcademicArticle | Control of chemoselectivity in catalytic rhodium carbenoid reactions through ligand modification | 1994 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/e7n364678 | AcademicArticle | Molecular basis for sequence selective DNA alkylation by (+)- and ent-(-)-CC-1065 and related agents: alkylation site models that accommodate the offset AT-rich adenine N3 alkylation selectivity | 1994 | 10.1016/S0968-0896(00)82007-6 | 7922122 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote264892 | AcademicArticle | Cerebrodiene: A brain lipid isolated from sleep-deprived cats | 1994 | 10.1073/pnas.91.20.9505 | 7937797 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote233050 | AcademicArticle | Total synthesis of bleomycin A(2) and related agents .4. Synthesis of the disaccharide subunit - 2-O-(3-O-carbamoyl-alpha-D-mannopyranosyl)-L-gulopyranose and completion of the total synthesis of bleomycin a(2) | 1994 | 10.1021/ja00092a014 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote216390 | AcademicArticle | P-quinonemethide analog of the CC-1065 and duocarmycin alkylation subunits | 1994 | 10.1021/jo00096a043 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote319634 | AcademicArticle | Diels-Alder reactions of cyclopropenone ketals - a concise tropolone annulation applicable to rubrolone-C ring introduction | 1994 | 10.1021/jo00091a040 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote16486 | AcademicArticle | Total synthesis and biological properties of novel antineoplastic (chloromethyl)furanoindolines - an asymmetric hydroboration mediated synthesis of the alkylation subunits | 1994 | 10.1021/jm00028a005 | 8295210 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote144893 | AcademicArticle | Design, synthesis, and evaluation of DNA minor-groove binding-agents - the duocarmycins | 1994 | 10.1351/pac199466040837 | http://vivo.scripps.edu/individual/endnote313708 | |
http://vivo.scripps.edu/individual/endnote287904 | AcademicArticle | Chemical and structural comparison of N-BOC-CBQ and N-BOC-CBI - identification and structural origin of an unappreciated but productive stability of the CC-1065 and duocarmycin SA alkylation subunits | 1994 | 10.1021/ja00093a067 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote167157 | AcademicArticle | (+)- and ent-(-)-duocarmycin SA and (+)- and ent-(-)-N-BOC-DSA DNA alkylation properties - alkylation site models that accommodate the offset AT-rich adenine N3 alkylation selectivity of the enantiomeric agents | 1994 | 10.1021/ja00084a004 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote289851 | AcademicArticle | CBI-TMI - synthesis and evaluation of a key analog of the duocarmycins - validation of a direct relationship between chemical solvolytic stability and cytotoxic potency and confirmation of the structural features responsible for the distinguishing behavior of enantiomeric pairs of agents | 1994 | 10.1021/ja00097a006 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote102790 | AcademicArticle | Crossing extreme mechanistic barriers by antibody catalysis: Syn elimination to a cis olefin | 1994 | 10.1021/ja00092a080 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote30738 | AcademicArticle | Role of the CC-1065 and duocarmycin N-2 substituent - validation of a direct relationship between solvolysis chemical-stability and in-vitro biological potency | 1994 | 10.1021/ja00091a088 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote237484 | AcademicArticle | Total synthesis of bouvardin, O-methylbouvardin, and O-methyl-N-9-desmethylbouvardin | 1994 | 10.1021/ja00098a015 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote380868 | AcademicArticle | Design, synthesis, and evaluation of CC-1065 and duocarmycin analogs incorporating the 2,3,10,10a-tetrahydro-1H-cyclopropa d benzo f quinol-5-one (CBQ) alkylation subunit - identification and structural origin of subtle stereoelectronic features that govern reactivity and regioselectivity | 1994 | 10.1021/ja00104a013 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote242802 | AcademicArticle | Total synthesis of bleomycin-A(2) and related agents .1. Synthesis and DNA-binding properties of the extended C-terminus - tripeptide-S, tetrapeptide-S, pentapeptide-S, and related agents | 1994 | 10.1021/ja00092a011 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote118365 | AcademicArticle | Total syntheses of (+)-p-3a, epi-(-)-p-3a, and (-)-desacetamido p-3a | 1994 | 10.1021/ja00080a010 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote45569 | AcademicArticle | Synthesis of a functionalized rigid bicyclo[2.2.1]heptane: a useful hapten for eliciting catalytic antibodies | 1994 | 10.1021/jo00096a064 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote66318 | AcademicArticle | Induction of endonucleolytic DNA fragmentation and apoptosis by the duocarmycins | 1994 | 10.1016/s0960-894x(01)80168-2 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote115977 | AcademicArticle | Inverse electron demand Diels-Alder reactions of heterocyclic azadienes - 4+2 -cycloaddition reaction of amidines with 1,3,5-triazines | 1994 | 10.1021/jo00096a044 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote41313 | AcademicArticle | Total synthesis of bleomycin-A(2) and related agents .2. Synthesis of (-)-pyrimidoblamic acid, epi-(+)-pyrimidoblamic acid, (+)-desacetamidopyrimidoblamic acid, and (-)-descarboxamidopyrimidoblamic acid | 1994 | 10.1021/ja00092a012 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote273598 | AcademicArticle | Total synthesis of bleomycin-A(2) and related agents .3. Synthesis and comparative-evaluation of deglycobleomycin-A(2), epideglycobleomycin-A(2), deglycobleomycin-A(1), and desacetamidodeglycobleomycin, descarboxamidodeglycobleomycin, desmethyldeglycobleomycin, and desimidazolyldeglycobleomycin-A(2) | 1994 | 10.1021/ja00092a013 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/e7n378082 | AcademicArticle | Evaluation of functional analogs of CC-1065 and the duocarmycins incorporating the cross-linking 9a-chloromethyl-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-on e (C2BI) alkylation subunit | 1993 | 10.1016/S0968-0896(00)82100-8 | 8081835 | http://vivo.scripps.edu/individual/endnote193708 |
http://vivo.scripps.edu/individual/endnote188912 | AcademicArticle | Vancomycin and ristocetin models - synthesis via the Ullmann macrocyclization reaction | 1993 | 10.1021/jo00058a024 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote53013 | AcademicArticle | 4pi participation of 1-aza-1,3-butadienes in [4 + 2] cycloaddition reactions: intramolecular Diels-Alder reactions of alpha,beta-unsaturated N-sulfonylimines | 1993 | 10.1021/jo00060a022 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote260958 | AcademicArticle | Design, synthesis, and evaluation of DNA minor-groove binding-agents | 1993 | 10.1351/pac199365061123 | http://vivo.scripps.edu/individual/endnote313708 | |
http://vivo.scripps.edu/individual/endnote366526 | AcademicArticle | Singlet oxygen oxidation of bipyrroles - total synthesis of d,l-isochrysohermidin and meso-isochrysohermidin | 1993 | 10.1021/ja00071a069 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote72459 | AcademicArticle | (-)-sandramycin - total synthesis and preliminary DNA-binding properties | 1993 | 10.1021/ja00077a082 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote66520 | AcademicArticle | CDPI3-enediyne and CDPI3-EDTA conjugates - a new class of DNA cleaving agents | 1993 | 10.1021/jo00063a019 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote345558 | AcademicArticle | Studies on the synthesis of bleomycin-A(2) - observations on a diastereoselective imine addition-reaction for C2-acetamido side-chain introduction | 1993 | 10.1016/0040-4039(93)85008-k | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote266906 | AcademicArticle | D, l- and meso-isochrysohermidin - total synthesis and interstrand DNA cross-linking | 1993 | 10.1021/ja00077a046 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote9911 | AcademicArticle | Total synthesis of streptonigrone | 1993 | 10.1021/ja00076a035 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote115780 | AcademicArticle | Total synthesis of (-)-pyrimidoblamic acid and deglycobleomycin A2 | 1993 | 10.1002/anie.199302731 | http://vivo.scripps.edu/individual/endnote319084 | |
http://vivo.scripps.edu/individual/endnote397602 | AcademicArticle | Total synthesis and preliminary evaluation of (+)-duocarmycin and ent-(-)-duocarmycin SA | 1993 | 10.1021/ja00073a019 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote282808 | AcademicArticle | Reversibility of the duocarmycin-A and SA DNA alkylation reaction | 1993 | 10.1021/ja00074a093 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote293730 | AcademicArticle | K-13 and OF4949 - evaluation of key partial structures and pharmacophore delineation | 1993 | 10.1016/s0960-894x(01)80885-4 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote222276 | AcademicArticle | Total synthesis of cycloisodityrosine, RA-VII, deoxybouvardin, and N29-desmethyl-RA-VII - identification of the pharmacophore and reversal of the subunit functional roles | 1993 | 10.1021/ja00062a004 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote42248 | AcademicArticle | Total synthesis of (+)-piperazinomycin | 1993 | 10.1021/ja00077a047 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/e7n385159 | AcademicArticle | Preparation and Diels-Alder reaction of a reactive, electron-deficient heterocyclic azadiene: dimethyl 1,2,4,5-tetrazine-3,6-dicarboxylate. 1,2-Diazine and pyrrole introduction | 1992 | http://vivo.scripps.edu/individual/endnote12246 | ||
http://vivo.scripps.edu/individual/e7n334975 | AcademicArticle | Total synthesis of (+)-duocarmycin SA | 1992 | 10.1021/ja00051a045 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/e7n71158 | AcademicArticle | Synthesis of N29-desmethyl RA-VII. Identification of the pharmacophore of RA-I-VII and deoxybouvardin and reassignment of the subunit functional roles | 1992 | 10.1021/jo00031a001 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n326895 | AcademicArticle | Synthesis of tri- and tetrapeptide S: the extended C-terminus of bleomycin A2 | 1992 | 10.1021/jo00042a003 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n284662 | AcademicArticle | Synthesis of desacetamidopyrimidoblamic acid and deglyco desacetamidobleomycin A2 | 1992 | 10.1021/jo00042a004 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n373535 | AcademicArticle | Design, synthesis, and evaluation of functional analogs of CC-1065 and the duocarmycins: a study of structural features effecting DNA binding selectivity | 1992 | http://vivo.scripps.edu/individual/e7n385337 | ||
http://vivo.scripps.edu/individual/e7n187986 | AcademicArticle | Synthesis of desacetamido P-3A: 1,3,5-triazine .fwdarw. pyrimidine heteroaromatic azadiene Diels-Alder reaction | 1992 | 10.1021/jo00032a001 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote29754 | AcademicArticle | DNA alkylation properties of enhanced functional analogs of cc-1065 incorporating the 1,2,9,9a-tetrahydrocyclopropa 1,2-c benz 1,2-e indol-4-one (cbi) alkylation subunit | 1992 | 10.1021/ja00040a001 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote386103 | AcademicArticle | P-3A and (-)-desacetamido P-3A - demonstration and study of their effective functional cleavage of duplex DNA | 1992 | 10.1016/s0960-894x(00)80449-7 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote132393 | AcademicArticle | Acyl radicals - intermolecular and intramolecular alkene addition-reactions | 1992 | 10.1021/jo00031a021 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote198417 | AcademicArticle | A convenient and general preparation of n-sulfonylimines | 1992 | 10.1021/jo00043a047 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote267978 | AcademicArticle | Deglyco GABA,gly-desacetamidobleomycin-A2 - a simplified synthetic model for bleomycin-A2 | 1992 | 10.1016/s0960-894x(01)81076-3 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote107076 | AcademicArticle | A concise synthesis of the fredericamycin-a DEF ring-system - 4+2 cycloaddition reactions of 1-aza-1,3-butadienes | 1992 | 10.1021/jo00040a044 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote566 | AcademicArticle | Functional analogs of CC-1065 and the duocarmycins incorporating the 9A-(chloromethyl)-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (C2BI) alkylation subunit - synthesis and preliminary DNA alkylation studies | 1992 | 10.1021/ja00050a012 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote160953 | AcademicArticle | An improved synthesis of 1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (CBI) - a simplified analog of the CC-1065 alkylation subunit | 1992 | 10.1021/jo00036a023 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote311521 | AcademicArticle | A simple method for the purification and isolation of bleomycin-A2 | 1992 | 10.1016/s0960-894x(00)80597-1 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote185465 | AcademicArticle | DNA alkylation properties of enhanced functional analogs of CC-1065 incorporating the 1,2,9,9a-tetrahydrocyclopropa[1,2-c]benz[1,2-e]indol-4-one (CBI) alkylation subunit | 1992 | 10.1016/s0960-894x(00)80407-2 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote113320 | AcademicArticle | Synthesis of the lower subunit of rhizoxin | 1992 | 10.1021/jo00034a010 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote192783 | AcademicArticle | CC-1065 partial structures - enhancement of noncovalent affinity for DNA minor groove binding through introduction of stabilizing electrostatic interactions | 1992 | 10.1021/jo00030a042 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n393042 | AcademicArticle | Total synthesis of calicheamicinone: a solution to the problem of the elusive urethane | 1991 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/e7n251533 | AcademicArticle | Recent advances in bioorganic chemistry. Preface | 1991 | 10.1016/s0040-4020(01)81771-3 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/e7n81503 | AcademicArticle | Solution structure of FKBP, a rotamase enzyme and receptor for FK506 and rapamycin. Atomic structure of FKBP-FK506, an immunophilin-immunosuppressant complex | 1991 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/e7n109651 | AcademicArticle | Duocarmycins: a new class of sequence selective DNA minor groove alkylating agents | 1991 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/endnote344314 | AcademicArticle | Singlet oxygen mediated oxidative decarboxylation of pyrrole-2-carboxylic acids | 1991 | 10.1021/jo00024a045 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote270484 | AcademicArticle | Inverse electron demand Diels-Alder reactions of N-sulfonyl alpha,beta-unsaturated imines - a general-approach to implementation of the 4-pi participation of 1-aza-1,3-butadienes in Diels-Alder reactions | 1991 | 10.1021/ja00005a040 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote158004 | AcademicArticle | Design and synthesis of a conformational analog of deoxybouvardin | 1991 | 10.1021/jo00018a035 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote319162 | AcademicArticle | Intramolecular Ullmann condensation reaction - an effective approach to macrocyclic diaryl ethers | 1991 | 10.1021/jo00005a020 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote41555 | AcademicArticle | Isolation and characterization of the duocarmycin adenine DNA adduct | 1991 | 10.1021/ja00017a042 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote83430 | AcademicArticle | A potent, simple derivative of an analog of the CC-1065 alkylation subunit | 1991 | 10.1016/s0960-894x(01)81090-8 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote101550 | AcademicArticle | Diels-Alder reactions of N-sulfonyl-1-aza-1,3-butadienes: Development of a synthetic approach to the streptonigrone C ring | 1991 | 10.1021/jo00002a077 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote388201 | AcademicArticle | Evaluation of bouvardin, deoxybouvardin, and RA-I - RA-VII partial structures - reassignment of the pharmacophore | 1991 | 10.1016/s0960-894x(01)80815-5 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote196335 | AcademicArticle | Demonstration of a pronounced effect of noncovalent binding selectivity on the (+)-CC-1065 DNA alkylation and identification of the pharmacophore of the alkylation subunit | 1991 | 10.1073/pnas.88.4.1431 | 1847523 | http://vivo.scripps.edu/individual/endnote71945 |
http://vivo.scripps.edu/individual/endnote213657 | AcademicArticle | Total synthesis of (+/-)-cis-trikentrin-A and (+/-)-trans-trikentrin-A - Diels-Alder reactions of heteroaromatic azadienes | 1991 | 10.1021/ja00011a026 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote126154 | AcademicArticle | (+)-CC-1065 DNA alkylation - observation of an unexpected relationship between cyclopropane electrophile reactivity and the intensity of DNA alkylation | 1991 | 10.1021/ja00007a077 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote141476 | AcademicArticle | Total synthesis of deoxybouvardin and RA-VII - macrocyclization via an intramolecular Ullmann reaction | 1991 | 10.1021/ja00004a062 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote140285 | AcademicArticle | Synthesis and preliminary evaluation of the fredericamycin-A ABCDE ring-system | 1991 | 10.1021/jo00006a029 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote60386 | AcademicArticle | Total synthesis of combretastatin D-2 - intramolecular ullmann macrocyclization reaction | 1991 | 10.1021/jo00013a024 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote137621 | AcademicArticle | (+)-CC-1065 DNA alkylation - key studies demonstrating a noncovalent binding selectivity contribution to the alkylation selectivity | 1991 | 10.1021/ja00010a046 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote398001 | AcademicArticle | Synthesis and preliminary evaluation of (+)-CBI-indole2 - an enhanced functional analog of (+)-CC-1065 | 1991 | 10.1016/s0960-894x(00)80243-7 | http://vivo.scripps.edu/individual/endnote119710 | |
http://vivo.scripps.edu/individual/endnote312063 | AcademicArticle | Studies on the synthesis of rubrolone: 4π participation of O-alkyl α,β-unsaturated oximes in intramolecular [4 + 2] cycloaddition reactions | 1991 | 10.1016/0040-4039(91)80554-j | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote46782 | AcademicArticle | An alternative and convenient strategy for generation of substantial quantities of singly 5-32P-end-labeled double-stranded DNA for binding-studies - development of a protocol for examination of functional features of (+)-CC-1065 and the duocarmycins that contribute to their sequence-selective DNA alkylation properties | 1991 | 10.1016/s0040-4020(01)81798-1 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/e2n15447 | AcademicArticle | Tandem free-radical ring expansion and 5-exo-dig 5-hexynyl radical cyclization: a useful approach to fused bicyclic carbocycles | 1990 | 10.1021/jo00307a010 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n237859 | AcademicArticle | Use of methylenecyclopropanone ketals for cyclopentane synthesis. A new efficient thermal [3 + 2] cycloaddition | 1990 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/e7n51727 | AcademicArticle | Polyethylene-bound soluble recoverable palladium(0) catalysts | 1990 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/e7n124651 | AcademicArticle | Photolytic reactions of chromium aminocarbene complexes. Conversion of amides to α-amino acids | 1990 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/e7n209698 | AcademicArticle | Room-temperature, endo-specific 1-aza-1,3-butadiene Diels-Alder reactions: acceleration of the LUMOdiene-controlled [4 + 2] cycloaddition reactions through noncomplementary aza diene substitution | 1990 | 10.1021/jo00297a006 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n108806 | AcademicArticle | Synthesis and preliminary evaluation of agents incorporating the pharmacophore of the duocarmycin/pyrindamycin alkylation subunit: identification of the CC-1065/duocarmycin common pharmacophore | 1990 | 10.1021/jo00302a002 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n262907 | AcademicArticle | The absolute configuration and synthesis of natural (-)-dolastatin 10 | 1990 | http://vivo.scripps.edu/individual/e7n47566 | ||
http://vivo.scripps.edu/individual/e7n280569 | AcademicArticle | Diels-Alder reactions of 1-aza-1,3-butadienes: room temperature, endo-selective LUMOdiene-controlled [4 + 2] cycloaddition reactions of N-sulfonyl-4-(ethoxycarbonyl)-1-aza-1,3-butadienes | 1990 | 10.1021/jo00307a009 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote266256 | AcademicArticle | Synthesis of N-(tert-butyloxycarbonyl)-CBI, CBI, CBI-CBI1, and CBI-CDPI2 - enhanced functional analogs of CC-1065 incorporating the 1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (CBI) left-hand subunit | 1990 | 10.1021/jo00310a013 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote310433 | AcademicArticle | Regiocontrolled nucleophilic-addition to selectively activated para-quinone diimines - alternative preparation of a key intermediate employed in the preparation of the CC-1065 left-hand subunit | 1990 | 10.1021/jo00291a059 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote174449 | AcademicArticle | Synthesis and evaluation of aborted and extended CC-1065 functional analogs - (+)-CPI-PDE-1, and (-)-CPI-PDE-1, (+)-CPI-PDE-1, and (-)-CPI-CDPI1, and (+/-)-CPI-PDE-i1, (+)-CPI-PDE-i1, and (-)-CPI-CDPI3 - preparation of key partial structures and definition of an additional functional-role of the CC-1065 central and right-hand subunits | 1990 | 10.1021/ja00168a002 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote78406 | AcademicArticle | Tandem free-radical alkene addition-reactions of acyl radicals | 1990 | 10.1021/ja00166a043 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote279273 | AcademicArticle | Synthesis and preliminary evaluation of agents incorporating the pharmacophore of the duocarmycin pyrindamycin alkylation subunit - identification of the cc-1065 duocarmycin common pharmacophore | 1990 | 10.1021/jo00302a002 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote47805 | AcademicArticle | Duocarmycin pyrindamycin DNA alkylation properties and identification, synthesis, and evaluation of agents incorporating the pharmacophore of the duocarmycin pyrindamycin alkylation subunit - identification of the CC-1065-duocarmycin common pharmacophore | 1990 | 10.1021/ja00180a048 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote322347 | AcademicArticle | Design and total synthesis of a conformational analog of bouvardin deoxybouvardin | 1990 | http://vivo.scripps.edu/individual/endnote302592 | ||
http://vivo.scripps.edu/individual/endnote62204 | AcademicArticle | Resolution of a CBI precursor and incorporation into the synthesis of (+)-CBI, (+)-CBI-CDPI1, (+)-CBI-CDPI2 - enhanced functional analogs of (+)-CC-1065 - a critical-appraisal of a proposed relationship between electrophile reactivity, DNA-binding properties, and cytotoxic potency | 1990 | 10.1016/s0040-4039(00)94629-x | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote149493 | AcademicArticle | Intramolecular acyl radical alkene addition-reactions - macrocyclization reactions | 1990 | 10.1021/ja00166a044 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote13515 | AcademicArticle | Diels-Alder reactions of azadienes: scope and applications | 1990 | 10.1002/bscb.19900990902 | http://vivo.scripps.edu/individual/endnote204561 | |
http://vivo.scripps.edu/individual/endnote235650 | AcademicArticle | Studies of the total synthesis of fredericamycin-A - preparation of key partial structures and development of an intermolecular alkyne chromium carbene complex benzannulation cyclization approach to the ABCD(E) ring-system | 1990 | 10.1021/jo00293a043 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote84827 | AcademicArticle | Total synthesis of L,L-isodityrosine and isodityrosine-derived agents - K-13, OF4949-III, and OF4949-IV | 1990 | 10.1021/jo00311a019 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote186396 | AcademicArticle | A demonstration of the intrinsic importance of stabilizing hydrophobic binding and noncovalent van der Waals contacts dominant in the noncovalent CC-1065/b-DNA binding | 1990 | 10.1016/0009-2797(90)90107-x | 2406033 | http://vivo.scripps.edu/individual/endnote187913 |
http://vivo.scripps.edu/individual/endnote354821 | AcademicArticle | Synthesis of n-(phenylsulfonyl)-CI, N-((tert-butyloxy)carbonyl)-CI, CI-CDPI1, and CI-CDPI2 - CC-1065 functional analogs incorporating the parent 1,2,7,7a-tetrahydrocycloprop 1,2-c indol-4-one (CI) left-hand subunit | 1990 | 10.1021/ja00169a034 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/e2n323346 | AcademicArticle | Total synthesis of (.+-.)-N-(phenylsulfonyl)- and (.+-.)-N-(tert-butyloxycarbonyl)-CI, (.+-.)-CI-CDPI1, and (.+-.)-CI-CDPI2: CC-1065 functional analogs incorporating the parent 1,2,7,7a-tetrahydrocycloprop[1,2-c]indol-4-one (CI) left-hand subunit | 1989 | 10.1021/jo00267a004 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n296998 | AcademicArticle | Total synthesis of K-13 | 1989 | 10.1021/jo00272a003 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n270787 | AcademicArticle | Diels-Alder reactions of heterocyclic azadienes: development of a strategy for the total synthesis of streptonigrin, lavendamycin, and synthetic quinoline-5,8-quinones | 1989 | 10.1016/B978-0-08-092429-8.50006-4 | http://vivo.scripps.edu/individual/e7n271124 | |
http://vivo.scripps.edu/individual/e7n69344 | AcademicArticle | Phenylselenoesters as effective precursors of acyl radicals for use in intermolecular alkene addition reactions | 1989 | 10.1021/jo00269a001 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n252223 | AcademicArticle | Recent applications of the inverse electron demand Diels-Alder reaction | 1989 | http://vivo.scripps.edu/individual/e7n163765 | ||
http://vivo.scripps.edu/individual/endnote1433 | AcademicArticle | A general-solution to implementing the 4-p participation of 1-aza-1,3-butadienes in Diels-Alder reactions - inverse electron demand Diels-Alder reactions of alpha,beta-unsaturated n-benzenesulfonyl imines | 1989 | 10.1021/ja00186a067 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote173129 | AcademicArticle | Studies on the total synthesis of fredericamycin-a - development of an intermolecular alkyne-chromium carbene complex cyclization approach to the abcde ring-system | 1989 | 10.1016/s0040-4039(01)93705-0 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote345129 | AcademicArticle | Synthesis of isodityrosine | 1989 | 10.1016/s0040-4039(01)93709-8 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote43046 | AcademicArticle | Total synthesis of OF4949-III and OF4949-IV - unusual effects of remote substituents on the rate of macrocyclization reactions | 1989 | 10.1016/s0040-4039(01)93447-1 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote80846 | AcademicArticle | A study of the scope of the 4+2 cyclo-addition reactions of unactivated 1,3-oxazin-6-ones | 1989 | 10.1021/jo00264a041 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote21719 | AcademicArticle | Total synthesis and evaluation of (+/-)-N-(tert-butyloxycarbonyl)-CBI, (+/-)-CBI-CDPI1, and (+/-)-CBI-CDPI2 - CC-1065 functional agents incorporating the equivalent 1,2,9,9a-tetrahydrocycloprop 1,2-c benz 1,2-e indol-4-one (CBI) left-hand subunit | 1989 | 10.1021/ja00198a089 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/e7n140777 | AcademicArticle | A divergent de novo synthesis of carbohydrates based on an accelerated inverse electron demand Diels-Alder reaction of 1-oxa-1,3-butadienes | 1988 | 10.1021/jo00259a040 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n148045 | AcademicArticle | Preparation and inverse-electron-demand Diels-Alder reaction of an electron-deficient heterocyclic azadiene: triethyl 1,2,4-triazine-3,5,6-tricarboxylate and 2,3,6-tricarboethoxypyridine | 1988 | http://vivo.scripps.edu/individual/endnote12246 | ||
http://vivo.scripps.edu/individual/e7n26376 | AcademicArticle | Accelerated inverse electron demand Diels-Alder reactions of 1-oxa-1,3-butadienes: [4 + 2] cycloaddition reactions of beta,gamma-unsaturated alpha-keto esters | 1988 | 10.1021/jo00249a052 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n192828 | AcademicArticle | Acyl radicals: functionalized free radicals for intramolecular cyclization reactions | 1988 | 10.1021/jo00249a053 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote246984 | AcademicArticle | Inverse electron demand Diels-Alder reactions of 2,4,6-tris(ethoxycarbonyl)-1,3,5-triazine and 2,4,6-tris(methylthio)-1,3,5-triazine - pyrimidine introduction | 1988 | 10.1016/s0040-4020(01)85973-1 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/endnote252937 | AcademicArticle | Studies on the total synthesis of bouvardin and deoxybouvardin - cyclic hexapeptide cyclization studies and preparation of key partial structures | 1988 | 10.1021/jo00238a005 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote300165 | AcademicArticle | Oxidative coupling of methyl 6-hydroxyindole-2-carboxylate with primary amines - preparation of 2-substituted methyl pyrrolo 2,3-e benzoxazole-5-carboxylates | 1988 | 10.1021/jo00256a053 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote24237 | AcademicArticle | Total synthesis of (+/-)-n-2-(phenylsulfonyl)-cpi, (+/-)-cc-1065, (+)-cc-1065, ent-(-)-cc-1065, and the precise, functional agents (+/-)-cpi-cdpi2, (+)-cpi-cdpi2, and (-)-cpi-cdpi2 (+/-)-(3br-star,4as-star)-deoxy-cc-1065, (+)-(3br,4as)-deoxy-cc-1065, and (-)-(3bs,4ar)-deoxy-cc-1065 | 1988 | 10.1021/ja00222a043 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote3953 | AcademicArticle | Total synthesis of prodigiosin, prodigiosene, and desmethoxyprodigiosin - Diels-Alder reactions of heterocyclic azadienes and development of an effective palladium(II)-promoted 2,2'-bipyrrole coupling procedure | 1988 | 10.1021/jo00242a013 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote232546 | AcademicArticle | Total synthesis of (+)CPI-CDPI2 and (-)-CPI-CDPI2 - (+)-(3br,4as)-deoxy-CC-1065 and (-)-(3bs,4ar)-deoxy-CC-1065 | 1988 | 10.1021/jo00238a042 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote15051 | AcademicArticle | Preparation and inverse electron demand Diels-Alder reaction of an electron-deficient heterocyclic azadiene - triethyl 1,2,4-triazine-3,5,6-tricarboxylate | 1988 | http://vivo.scripps.edu/individual/endnote12246 | ||
http://vivo.scripps.edu/individual/endnote373062 | AcademicArticle | Inverse electron demand Diels-Alder reactions of 3,6-bis(methylthio)-1,2,4,5-tetrazine - 1,2-diazine introduction and direct implementation of a divergent 1,2,4,5-tetrazine- 1,2-diazine- benzene (indoline indole) Diels-Alder strategy | 1988 | 10.1021/jo00242a014 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote159208 | AcademicArticle | Thermal cyclo-addition reactions of pi-delocalized singlet vinylcarbenes - 3-carbon 1,1-dipoles/1,3-dipoles - the thermal 3-carbon + 2-carbon cyclo-addition | 1988 | 10.1021/jo00250a002 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote13343 | AcademicArticle | Total synthesis of (+)-CC-1065 and ent-(-)-CC-1065 | 1988 | 10.1021/ja00212a067 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/e7n112519 | AcademicArticle | Preparation and inverse electron demand Diels-Alder reaction of an electron-deficient diene: methyl 2-oxo-5,6,7,8-tetrahydro-2H-1-benzopyran-3-carboxylate (2H-1-benzopyran-3-carboxylic acid, 5,6,7,8-tetrahydro-2-oxo-, methyl ester) | 1987 | http://vivo.scripps.edu/individual/endnote12246 | ||
http://vivo.scripps.edu/individual/e7n151037 | AcademicArticle | Preparation and three-carbon + two-carbon cycloaddition of a cyclopropenone ketal: cyclopropenone 1,3-propanediol ketal (4,8-dioxaspiro[2.5]oct-1-ene) | 1987 | http://vivo.scripps.edu/individual/endnote12246 | ||
http://vivo.scripps.edu/individual/endnote39970 | AcademicArticle | Activation and coupling of pyrrole-1-carboxylic acid in the formation of pyrrole N-carbonyl compounds - pyrrole-1-carboxylic acid anhydride | 1987 | 10.1021/jo00387a046 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote58429 | AcademicArticle | Diels-alder reactions of heterocyclic azadienes - total synthesis of pde-i, pde-ii, and pde-i dimer methyl-ester | 1987 | 10.1021/ja00243a027 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote206328 | AcademicArticle | Selectively protected L-dopa derivatives - application of the benzylic hydroperoxide rearrangement | 1987 | 10.1021/jo00232a044 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote31699 | AcademicArticle | Further observations on the Lewis acid-catalyzed benzylic hydroperoxide rearrangement - use of a boron-trifluoride hydrogen-peroxide preformed, aged reagent | 1987 | 10.1016/s0040-4039(00)95902-1 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote215926 | AcademicArticle | Streptonigrin and lavendamycin partial structures. Preparation of 7-amino-2-(2′-pyridyl)quinoline-5,8-quinone-6′-carboxylic acid: a probe for the minimum, potent pharmacophore of the naturally occurring antitumor-antibiotics | 1987 | 10.1002/jhet.5570240504 | http://vivo.scripps.edu/individual/endnote355769 | |
http://vivo.scripps.edu/individual/endnote118849 | AcademicArticle | Streptonigrin and lavendamycin partial structures - probes for the minimum, potent pharmacophore of streptonigrin, lavendamycin, and synthetic quinoline-5,8-diones | 1987 | 10.1021/jm00393a040 | 3656364 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote201544 | AcademicArticle | Indole N-carbonyl compounds - preparation and coupling of indole-1-carboxylic acid anhydride | 1987 | 10.1021/jo00226a044 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote113754 | AcademicArticle | Total synthesis of prodigiosin | 1987 | 10.1016/s0040-4039(00)95451-0 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote365520 | AcademicArticle | Studies on the total synthesis of CC-1065 - preparation of a synthetic, simplified 3-carbamoyl-1,2-dihydro-3h-pyrrolo 3,2-e indole dimer/trimer/tetramer (CDPI dimer/trimer/tetramer) and development of methodology for PDE-I dimer methyl-ester formation | 1987 | 10.1021/jo00384a026 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n396489 | AcademicArticle | Diels-Alder reactions of heterocyclic azadienes: total synthesis of PDE-II methyl ester | 1986 | 10.1021/jo00366a048 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote248573 | AcademicArticle | Thermal-reactions of cyclopropenone ketals - key mechanistic features and scope of the cycloaddition reactions of delocalized singlet vinylcarbenes - 3-carbon 1,1-dipoles 1,3-dipoles | 1986 | 10.1021/ja00281a041 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote310880 | AcademicArticle | Benzylic hydroperoxide rearrangement - observations on a viable and convenient alternative to the Baeyer Villiger rearrangement | 1986 | 10.1021/jo00376a079 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote62135 | AcademicArticle | An improved and divergent introduction of the streptonigrin and lavendamycin quinoline-5,8-quinone AB ring-systems | 1986 | 10.3987/R-1986-04-1067 | http://vivo.scripps.edu/individual/endnote14559 | |
http://vivo.scripps.edu/individual/endnote33353 | AcademicArticle | Diels-Alder reactions of heterocyclic azadienes: scope and applications | 1986 | 10.1021/cr00075a004 | http://vivo.scripps.edu/individual/endnote51983 | |
http://vivo.scripps.edu/individual/endnote289061 | AcademicArticle | Diels-Alder cycloaddition reactions of cyclopropenone ketals: dual participation in inverse electron demand (LUMOdiene controlled) and normal HOMOdiene controlled) Diels-Alder reactions, approaches to the preparation of tropones | 1986 | 10.1016/s0040-4020(01)90567-8 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/endnote88058 | AcademicArticle | Thermal-reactions of cyclopropenone ketals - application of the cycloaddition reactions of delocalized singlet vinylcarbenes - 3-carbon 1,1-dipoles 1,3-dipoles - an alternative synthesis of deacetamidocolchiceine - formal total synthesis of colchicine | 1986 | 10.1021/ja00281a042 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote390618 | AcademicArticle | Diels-Alder cycloadditions of rigid dienophiles: a probe for allylic axial substituent control of the pi-facial selectivity in the Diels-Alder reaction | 1986 | 10.1016/s0040-4039(00)84072-1 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/e7n384434 | AcademicArticle | Thermal, four-carbon + three-carbon cycloaddition reaction of cyclopropenone ketals. Total synthesis of deacetamidocolchiceine: formal total synthesis of colchicine | 1985 | 10.1021/jo00218a042 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote112947 | AcademicArticle | Inverse electron demand Diels-Alder reactions of heterocyclic azadienes - formal total synthesis of streptonigrin | 1985 | 10.1021/ja00306a024 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote65240 | AcademicArticle | Antimicrobial and cytotoxic properties of 9,10-dihydrophenanthrenes: structure activity studies on juncusol | 1985 | 10.1021/jm00148a031 | 4045930 | http://vivo.scripps.edu/individual/endnote266962 |
http://vivo.scripps.edu/individual/endnote282630 | AcademicArticle | Total synthesis of lavendamycin methyl-ester | 1985 | 10.1021/jo00350a070 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote286000 | AcademicArticle | Inverse electron demand Diels-Alder reactions of heterocyclic aza dienes - studies on the total synthesis of lavendamycin - investigative studies on the preparation of the CDE beta-carboline ring-system and AB quinoline-5,8-quinone ring-system | 1985 | 10.1021/jo00350a069 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote321884 | AcademicArticle | Preparation of optically-active, functionalized cis-delta-6-1-octalones | 1985 | 10.1021/jo00211a024 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote246072 | AcademicArticle | Regioselectivity of the intermolecular Diels-Alder reaction of acyl nitroso-compounds (C-nitrosocarbonyl compounds) and nitrosoformates (O-nitrosocarbonyl compounds) - preparation of functionalized cis-delta-6-1-octalones | 1985 | 10.1021/jo00211a025 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote31052 | AcademicArticle | A detailed, convenient preparation of dimethyl "1,2,4,5-tetrazine-3,6-dicarboxylate | 1985 | 10.1021/jo00225a076 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n45212 | AcademicArticle | Regioselectivity in the intermolecular Diels-Alder reaction of acyl nitroso compounds (C-nitrosocarbonyl compounds) and nitrosoformates (O-nitrosocarbonyl compounds) | 1984 | 10.1021/jo00195a057 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote380280 | AcademicArticle | Palladium (0) mediated beta-carboline synthesis - preparation of the CDE ring-system of lavendamycin | 1984 | http://vivo.scripps.edu/individual/endnote225462 | ||
http://vivo.scripps.edu/individual/endnote268550 | AcademicArticle | Total syntheses of azafluoranthene alkaloids: rufescine and imeluteine | 1984 | 10.1021/jo00195a035 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote60623 | AcademicArticle | Effective, thermal 3-carbon + 2-carbon cycloaddition for cyclopentenone formation - formal 1,3-dipolar cycloaddition of cyclopropenone ketals | 1984 | 10.1021/ja00315a065 | http://vivo.scripps.edu/individual/endnote181842 | |
http://vivo.scripps.edu/individual/endnote84558 | AcademicArticle | Thermal, 3-carbon + 2-atom cycloaddition of cyclopropenone ketals with carbon-heteroatom double-bonds - butenolide, furan, and gamma-keto ester preparation | 1984 | 10.1016/s0040-4039(01)91394-2 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote161185 | AcademicArticle | Inverse electron demand Diels-Alder reactions of 3-carbomethoxy-2-pyrones - controlled introduction of oxygenated aromatics - benzene, phenol, catechol, resorcinol, and pyrogallol annulation - regiospecific total synthesis of sendaverine and a preparation of 6,7-benzomorphans | 1984 | 10.1021/jo00195a033 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote275780 | AcademicArticle | Thermal cycloaddition of dimethyl "1,2,4,5-tetrazine-3,6-dicarboxylate with electron-rich olefins - 1,2-diazine and pyrrole introduction - preparation of octamethylporphin (OMP) | 1984 | 10.1021/jo00197a015 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote26571 | AcademicArticle | Effective, thermal one-carbon + 2-carbon cycloaddition of cyclopropenone ketals with electron deficient olefins - cyclopropane formation | 1984 | 10.1016/s0040-4039(01)91393-0 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote143477 | AcademicArticle | Regiospecific total synthesis of juncusol | 1984 | 10.1021/jo00195a034 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote161688 | AcademicArticle | Intramolecular diels-alder reactions of 1,2-diazines - general indoline synthesis - studies on the preparation of the central and right-hand segments of cc-1065 | 1984 | 10.1021/jo00186a032 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote173664 | AcademicArticle | Direct introduction of nitriles via use of unstable reissert intermediates - convenient procedures for the preparation of 2-cyanoquinolines and 1-cyanoisoquinolines | 1984 | 10.1021/jo00195a036 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/e7n301118 | AcademicArticle | Formal total synthesis of streptonigrin | 1983 | 10.1021/jo00152a049 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote372016 | AcademicArticle | Inverse electron demand Diels-Alder reactions of 3-carbomethoxy-2-pyrones - controlled introduction of oxygenated aromatics - benzene, phenol, catechol, resorcinol, pyrogallol annulation | 1983 | 10.1016/s0040-4039(01)99816-8 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote369173 | AcademicArticle | Diels-Alder reactions of azadienes | 1983 | 10.1016/s0040-4020(01)92154-4 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/endnote42403 | AcademicArticle | 1,2,4-triazine preparation via thermal cycloaddition of dimethyl 1,2,4,5-tetrazine-3,6-dicarboxylate with aryl thioimidates | 1983 | 10.1016/s0040-4039(00)85941-9 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote242354 | AcademicArticle | Diels-Alder reaction of heterocyclic azadienes. 2. Catalytic Diels-Alder reaction of in situ generated enamines with 1,2,4-triazines: general pyridine annulation | 1982 | 10.1021/jo00344a031 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote233434 | AcademicArticle | Regiospecific total synthesis of juncusol | 1982 | 10.1016/s0040-4039(00)85652-x | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote266303 | AcademicArticle | Inverse electron demand diels-alder reaction of 3-carbomethoxy-2-pyrones with 1,1-dimethoxyethylene - a simple and mild method of aryl annulation | 1982 | 10.1016/s0040-4039(00)85651-8 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote195921 | AcademicArticle | Thermal cycloaddition of 1,3,5-triazine with enamines - regiospecific pyrimidine annulation | 1982 | 10.1021/jo00134a034 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote1836 | AcademicArticle | Synthetic analgesics - preparation of racemic 6,7-benzomorphans | 1982 | 10.1016/s0040-4039(00)85653-1 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote294737 | AcademicArticle | Pyridine construction via thermal cycloaddition of 1,2,4-triazines with enamines - studies on the preparation of the bi-aryl CD rings of streptonigrin | 1982 | 10.1021/jo00140a035 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote121295 | AcademicArticle | Preparation of 3-methyl-4-vinyl-1,2,5-oxadiazole and 3-methyl-4-vinyl-1,2,5-thiadiazole | 1981 | 10.1002/jhet.5570180636 | http://vivo.scripps.edu/individual/endnote355769 | |
http://vivo.scripps.edu/individual/endnote365275 | AcademicArticle | Preparation of (R)-(+) and (S)-(-)-4-iodo-1,2-epoxybutane (R)-(2-iodoethyl)oxirane and (S)-(2-iodoethyl)oxirane , useful chiral synthons | 1981 | 10.1021/jo00319a034 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote166728 | AcademicArticle | Diels-alder reaction of heterocyclic azadienes .1. Thermal cycloaddition of 1,2,4-triazine with enamines - simple preparation of substituted pyridines | 1981 | 10.1021/jo00323a044 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote227070 | AcademicArticle | A simplified isoquinoline synthesis | 1981 | 10.1016/s0040-4020(01)93272-7 | http://vivo.scripps.edu/individual/endnote9731 | |
http://vivo.scripps.edu/individual/endnote41494 | AcademicArticle | A simple and convenient phenol annelation | 1980 | 10.1021/jo01312a044 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/n25725 | Thesis | I. New annulation processes ; II. Studies directed toward a biomimetic syntheic approach to prostaglandins | 1980 | |||
http://vivo.scripps.edu/individual/endnote342187 | AcademicArticle | Convenient preparation of 2-substituted benzothiazoles | 1978 | 10.1021/jo00405a050 | http://vivo.scripps.edu/individual/endnote171323 | |
http://vivo.scripps.edu/individual/endnote137289 | AcademicArticle | Concerning the stereochemistry of 9-methyl-Δ1-3-octalone | 1978 | 10.1016/S0040-4039(01)88970-X | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote156107 | AcademicArticle | New annulation processes for fused and spiro rings based on chemistry of benzothiazoles | 1978 | http://vivo.scripps.edu/individual/endnote225462 | ||
http://vivo.scripps.edu/individual/endnote8088 | AcademicArticle | Application of benzothiazoles to carbon-carbon bond formation in organic-synthesis | 1978 | http://vivo.scripps.edu/individual/endnote225462 | ||
http://vivo.scripps.edu/individual/endnote160204 | AcademicArticle | Oxidative cationic cyclization reactions effected by pyridinium chlorochromate | 1978 | 10.1016/S0040-4039(01)94800-2 | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote54448 | AcademicArticle | New and unusually flexible scheme for annulation to form fused cyclohexenone units | 1978 | 10.1016/S0040-4039(01)85680-X | http://vivo.scripps.edu/individual/endnote225462 | |
http://vivo.scripps.edu/individual/endnote22302 | AcademicArticle | Benzothiazoles as carbonyl equivalents | 1978 | http://vivo.scripps.edu/individual/endnote225462 | ||
http://vivo.scripps.edu/individual/endnote284510 | AcademicArticle | Synthesis and chiroptical properties of some asymmetric planar cisoid dienes | 1976 | 10.1016/0040-4020(76)80042-7 | http://vivo.scripps.edu/individual/endnote9731 |