Publication list

publication_uri type publication_title year doi pmid journal_uri
http://vivo.scripps.edu/individual/e2n132419 AcademicArticle C1-CBP-vancomycin: Impact of a vancomycin C-terminus trimethylammonium cation on pharmacological properties and insights into its newly introduced mechanism of action 2020 10.1021/acs.joc.9b02314 31670958 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e2n371614 AcademicArticle Next-Generation Total Synthesis of Vancomycin 2020 10.1021/jacs.0c07433 32885969 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n317190 AcademicArticle Precise Targeted Cleavage of a r(CUG) Repeat Expansion in Cells by Using a Small-Molecule-Deglycobleomycin Conjugate 2020 10.1021/acschembio.0c00036 http://vivo.scripps.edu/individual/endnote153903
http://vivo.scripps.edu/individual/e2n108497 AcademicArticle Vancomycin C-Terminus Guanidine Modifications and Further Insights into an Added Mechanism of Action Imparted by a Peripheral Structural Modification 2020 10.1021/acsinfecdis.0c00258 32598127 http://vivo.scripps.edu/individual/e2n233249
http://vivo.scripps.edu/individual/e2n181332 AcademicArticle Total synthesis and stereochemical assignment of streptide 2019 10.1021/jacs.9b09067 31577142 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n373958 AcademicArticle A small molecule drug conjugate (SMDC) of DUPA and a duocarmycin built on the solid phase 2019 10.1039/c9md00279k http://vivo.scripps.edu/individual/endnote55555
http://vivo.scripps.edu/individual/e2n170510 AcademicArticle N-acyl pyrazoles: effective and tunable inhibitors of serine hydrolases 2019 10.1016/j.bmc.2019.03.020 30879861 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/e2n319448 AcademicArticle Ultra-potent vinblastine analogues improve on-target activity of the parent microtubulin-targeting compound 2019 10.1016/j.bmcl.2019.03.036 30952593 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n321823 AcademicArticle Triarylaminium radical cation promoted coupling of catharanthine with vindoline: diastereospecific synthesis of anhydrovinblastine and reaction scope 2019 10.1021/jacs.9b06968 31442047 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n72523 AcademicArticle Exploration of the site-specific nature and generalizability of a trimethylammonium salt modification on vancomycin: A-ring derivatives 2019 10.1016/j.tet.2019.02.008 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/e2n91509 AcademicArticle SAR studies of 4-acyl-1,6-dialkylpiperazin-2-one arenavirus cell entry inhibitors 2019 10.1016/j.bmcl.2019.08.024 31537423 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n185220 AcademicArticle Resveratrol trimer enhances gene delivery to hematopoietic stem cells by reducing antiviral restriction at endosomes 2019 10.1182/blood.2019000040 31416800 http://vivo.scripps.edu/individual/endnote304227
http://vivo.scripps.edu/individual/e2n193601 AcademicArticle Structural basis of TLR2/TLR1 activation by the synthetic agonist diprovocim 2019 10.1021/acs.jmedchem.8b01583 30829478 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e2n185787 AcademicArticle Inverse electron demand Diels-Alder reactions of heterocyclic azadienes, 1-aza-1,3-butadienes, cyclopropenone ketals and related systems. A retrospective 2019 10.1021/acs.joc.9b00834 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e2n71244 AcademicArticle Synthesis, characterization, and rapid cycloadditions of 5-nitro-1,2,3-triazine 2018 10.1021/acs.orglett.8b00825 29659291 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/e2n131232 AcademicArticle Diprovocims: A new and exceptionally potent class of toll-like receptor agonists 2018 10.1021/jacs.8b09223 30272974 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n132606 AcademicArticle Duocarmycin SA, a potent antitumor antibiotic, sensitizes glioblastoma cells to proton radiation 2018 10.1016/j.bmcl.2018.04.008 29650288 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n195020 AcademicArticle Adjuvant effect of the novel TLR1/TLR2 agonist Diprovocim synergizes with anti-PD-L1 to eliminate melanoma in mice 2018 10.1073/pnas.1809232115 30150374 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/e2n54849 AcademicArticle High expression of class III β-tubulin has no impact on functional cancer cell growth inhibition of a series of key vinblastine analogs 2018 10.1016/j.bmcl.2018.02.006 29439899 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n61286 AcademicArticle N-terminus alkylation of vancomycin: ligand binding affinity, antimicrobial activity, and site-specific nature of quaternary trimethylammonium salt modification 2018 10.1021/acsinfecdis.8b00152 30067012 http://vivo.scripps.edu/individual/e2n233249
http://vivo.scripps.edu/individual/e2n250703 AcademicArticle Peripheral modifications of [Ψ[CH2NH]Tpg4]vancomycin with added synergistic mechanisms of action provide durable and potent antibiotics 2017 10.1073/pnas.1704125114 28559345 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/e2n251033 AcademicArticle Design of benzoxathiazin-3-one 1,1-dioxides as a new class of irreversible serine hydrolase inhibitors: Discovery of a uniquely selective PNPLA4 inhibitor 2017 10.1021/jacs.7602985 28498651 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n143800 AcademicArticle Direct synthesis of β-aminoenals through reaction of 1,2,3-triazine with secondary amines 2017 10.1021/acs.orglett.7b01543 28657329 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/e2n239190 AcademicArticle Vinblastine 20 ' amides: synthetic analogues that maintain or improve potency and simultaneously overcome Pgp-derived efflux and resistance 2017 10.1021/acs.jmedchem.7b00958 28857558 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e2n261608 AcademicArticle The difference a single atom can make: synthesis and design at the chemistry-biology interface 2017 10.1021/acs.joc.7b02088 28945374 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e2n66041 AcademicArticle Total synthesis of a key series of vinblastines modified at C4 that define the importance and surprising trends in activity 2017 10.1039/c6sc04146a 28194270 http://vivo.scripps.edu/individual/endnote149552
http://vivo.scripps.edu/individual/e2n61617 AcademicArticle Total syntheses of vancomycin-related glycopeptide antibiotics and key analogues 2017 10.1021/acs.chemrev.6b00820 28437097 http://vivo.scripps.edu/individual/endnote51983
http://vivo.scripps.edu/individual/e2n281853 AcademicArticle FAAH inhibitor OL-135 disrupts contextual, but not auditory, fear conditioning in rats 2016 10.1016/j.bbr.2016.04.014 27083303 http://vivo.scripps.edu/individual/endnote70642
http://vivo.scripps.edu/individual/e2n137683 AcademicArticle Synthesis of a potent vinblastine: rationally designed added benign complexity 2016 10.1021/jacs.6b04330 27356080 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n144750 AcademicArticle Small-molecule fusion inhibitors bind the pH-sensing stable signal peptide-GP2 subunit interface of the Lassa virus Envelope glycoprotein 2016 10.1128/jvi.00597-16 27194767 http://vivo.scripps.edu/individual/endnote197644
http://vivo.scripps.edu/individual/e2n53616 AcademicArticle Synthesis and evaluation of duocarmycin SA analogs incorporating the methyl 1,2,8,8a-tetrahydrocyclopropa c imidazolo 4,5-e indol-4-one-6-carboxylat e (CImI) alkylation subunit 2016 10.1016/j.bmc.2016.04.050 27221071 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/e2n122422 AcademicArticle TLR4/MD-2 activation by a synthetic agonist with no similarity to LPS 2016 10.1073/pnas.1525639113 26831104 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/e2n330271 AcademicArticle Tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition cascade of 1,3,4-oxadiazoles: initial scope and applications 2016 10.1021/acs.accounts.5b00510 26813287 http://vivo.scripps.edu/individual/endnote122847
http://vivo.scripps.edu/individual/e2n254668 AcademicArticle Ultrapotent vinblastines in which added molecular complexity further disrupts the target tubulin dimer-dimer interface 2016 10.1073/pnas.1611405113 27512044 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/e2n305180 AcademicArticle Catalysis of heterocyclic azadiene cycloaddition reactions by solvent hydrogen bonding: concise total synthesis of methoxatin 2016 10.1021/jacs.6b05438 27571404 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n14106 AcademicArticle Discovery and structure-activity relationships of the neoseptins: a new class of toll-like receptor-4 (TLR4) agonists 2016 10.1021/acs.jmedchem.6b00177 27050713 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e2n252643 AcademicArticle Total synthesis of (-)-vindoline and (+)-4-epi-vindoline based on a 1,3,4-oxadiazole tandem intramolecular 4+2 / 3+2 cycloaddition cascade initiated by an allene dienophile 2015 10.1021/acs.orglett.5b02818 26457536 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/e2n330409 AcademicArticle A five-membered lactone prodrug of CBI-based analogs of the duocarmycins 2015 10.1016/j.tetlet.2014.11.038 26069351 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/e2n171836 AcademicArticle Comprehensive analysis of structure-activity relationships of a-ketoheterocycles as sn-1-diacylglycerol lipase a inhibitors 2015 10.1021/acs.jmedchem.5b01627 26584396 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e2n330974 AcademicArticle Total synthesis of vinblastine, related natural products, and key analogues and development of inspired methodology suitable for the systematic study of their structure-function properties 2015 10.1021/ar500400w 25586069 http://vivo.scripps.edu/individual/endnote122847
http://vivo.scripps.edu/individual/e2n98348 AcademicArticle Target-based screen against a periplasmic serine protease that regulates intrabacterial pH homeostasis in Mycobacterium tuberculosis 2015 10.1021/cb500746z 25457457 http://vivo.scripps.edu/individual/endnote153903
http://vivo.scripps.edu/individual/e2n229404 AcademicArticle Total synthesis of (-)-kopsinine and ent-(+)-kopsinine 2015 10.1016/j.tet.2014.07.094 26074629 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/e2n267911 AcademicArticle Cycloadditions of 1,2,3-triazines bearing C5-electron donating substituents: robust pyrimidine synthesis 2015 10.1021/acs.orglett.5b01870 26172042 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/e2n147302 AcademicArticle Total syntheses and initial evaluation of [?[C(-S)NH]Tpg(4)]vancomycin, [?[C(-NH)NH]Tpg(4)]vancomycin, [?[CH2NH]Tpg(4)]vancomycin, and their (4-Chlorobiphenyl)methyl derivatives: synergistic binding pocket and peripheral modifications for the glycopeptide antibiotics 2015 10.1021/jacs.5b01008 25750995 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n173008 AcademicArticle Total synthesis of dihydrolysergic acid and dihydrolysergol: development of a divergent synthetic strategy applicable to rapid assembly of D-ring analogs 2015 10.1016/j.tet.2015.05.093 26273113 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/e2n309155 AcademicArticle When sugar is not so sweet 2015 10.1126/science.aad3298 http://vivo.scripps.edu/individual/endnote276633
http://vivo.scripps.edu/individual/e10n5254 AcademicArticle Insights into the mechanism of streptonigrin-induced protein arginine deiminase inactivation 2014 10.1016/j.bmc.2013.12.064 24440480 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/e11n218192 AcademicArticle Design, synthesis, and characterization of alpha-ketoheterocycles that additionally target the cytosolic port Cys269 of fatty acid amide hydrolase 2014 10.1021/jm401820q 24456116 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e11n28879 AcademicArticle Total syntheses of (-)-kopsifoline D and (-)-deoxoapodine: divergent total synthesis via late-stage key strategic bond formation 2014 10.1021/ja500548e 24499015 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e11n53454 AcademicArticle Total syntheses of (-)-pyrimidoblamic acid and P-3A 2014 10.1021/ja412298c 24410439 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e12n212983 AcademicArticle alpha-Ketoheterocycle inhibitors of fatty acid amide hydrolase: exploration of conformational constraints in the acyl side chain 2014 10.1016/j.bmc.2014.03.013 24690529 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/e14n12278 AcademicArticle Enzymatic glycosylation of vancomycin aglycon: completion of a total synthesis of vancomycin and N- and C-terminus substituent effects of the aglycon substrate 2014 10.1021/ol501568t 24954524 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/e14n54464 AcademicArticle Discovery libraries targeting the major enzyme classes: the serine hydrolases 2014 10.1016/j.bmcl.2014.06.063 25037918 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e14n33648 AcademicArticle Inhibition of adenovirus replication by a trisubstituted piperazin-2-one derivative 2014 10.1016/j.antiviral.2014.05.010 24907427 http://vivo.scripps.edu/individual/endnote251700
http://vivo.scripps.edu/individual/e2n259165 AcademicArticle Total synthesis of Psi C(=NH)NH Tpg(4) vancomycin and its ((4)-chlorobiphenyl)methyl derivative: impact of peripheral modifications on vancomycin analogues redesigned for dual D-Ala-D-Ala and D-Ala-D-Lac binding 2014 10.1021/ja507009a 25211770 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n187406 AcademicArticle Asymmetric synthesis of a CBI-based cyclic N-acyl O-amino phenol duocarmycin prodrug 2014 10.1021/jo501839x 25247380 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e2n52915 AcademicArticle Cycloadditions of noncomplementary substituted 1,2,3-triazines 2014 10.1021/ol502436n 25222918 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/e1n6514 AcademicArticle A remarkable series of vinblastine analogues displaying enhanced activity and an unprecedented tubulin binding steric tolerance: C20' urea derivatives 2013 10.1021/jm3015684 23244701 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e1n121557 AcademicArticle Rational design of fatty acid amide hydrolase inhibitors that act by covalently bonding to two active site residues 2013 10.1021/ja4014997 23581831 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e3n124417 AcademicArticle Probing the role of the vancomycin E-ring aryl chloride: selective divergent synthesis and evaluation of alternatively substituted E-ring analogues 2013 10.1021/jm4004494 23617725 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e3n283144 AcademicArticle Efficacious cyclic N-acyl O-amino phenol duocarmycin prodrugs 2013 10.1021/jm400413r 23627265 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/e4n127234 AcademicArticle NMR-assisted computational studies of peptidomimetic inhibitors bound in the hydrophobic pocket of HIV-1 glycoprotein 41 2013 10.1007/s10822-013-9662-6 23893342 http://vivo.scripps.edu/individual/endnote51058
http://vivo.scripps.edu/individual/e4n287897 AcademicArticle Biological and structural evaluation of 10R- and 10S-methylthio-DDACTHF reveals a new role for sulfur in inhibition of glycinamide ribonucleotide transformylase 2013 10.1021/bi4005182 23869564 http://vivo.scripps.edu/individual/endnote165634
http://vivo.scripps.edu/individual/e4n72372 AcademicArticle Investigation into the functional impact of the vancomycin C-ring aryl chloride 2013 10.1016/j.bmcl.2013.06.080 23880541 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e6n70136 AcademicArticle Transannular Diels-Alder/1,3-dipolar cycloaddition cascade of 1,3,4-oxadiazoles: total synthesis of a unique set of vinblastine analogues 2013 10.1021/oI402549n 24087969 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/e6n376933 AcademicArticle Potent vinblastine C20' ureas displaying additionally improved activity against a vinblastine-resistant cancer cell line 2013 10.1021/ml400281w 24223237 http://vivo.scripps.edu/individual/endnote225139
http://vivo.scripps.edu/individual/e6n2464 AcademicArticle Evaluation of a reductively activated duocarmycin prodrug against murine and human solid cancers 2013 10.4161/cbt.24348 23760495 http://vivo.scripps.edu/individual/endnote374839
http://vivo.scripps.edu/individual/e8n253951 AcademicArticle A fundamental relationship between hydrophobic properties and biological activity for the duocarmycin class of DNA-alkylating antitumor drugs: hydrophobic-binding-driven bonding 2013 10.1021/jm400665c 23944748 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/enote10848 AcademicArticle A Pd(0)-mediated indole (macro)cyclization reaction 2013 10.1021/ja3121394 23298368 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/enote337642 AcademicArticle Total synthesis of kopsinine 2013 10.1021/ol303573f 23391149 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/enote74874 AcademicArticle Total synthesis and evaluation of vinblastine analogues containing systematic deep-seated modifications in the vindoline subunit ring system: Core redesign 2013 10.1021/jm3014376 23252481 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/enote245789 AcademicArticle Hypervalent iodine(III)-promoted intermolecular C-C coupling of vindoline with β-ketoesters and related substrates 2013 10.1021/ol400135n 23421318 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/enote202853 AcademicArticle A novel, unusually efficacious duocarmycin carbamate prodrug that releases no residual byproduct 2012 10.1021/jm300330b 22650244 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/enote26088 AcademicArticle Total synthesis of [Psi[C(═S)NH]Tpg4]vancomycin aglycon, [Psi[C(═NH)NH]Tpg4]vancomycin aglycon, and related key compounds: reengineering vancomycin for dual D-Ala-D-Ala and D-Ala-D-Lac binding 2012 10.1021/ja209937s 22188323 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/enote227473 AcademicArticle Fe(III)/NaBH4-mediated free radical hydrofluorination of unactivated alkenes 2012 10.1021/ja3063716 22860624 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/enote308105 AcademicArticle The fatty acid amide hydrolase (FAAH) inhibitor PF-3845 acts in the nervous system to reverse LPS-induced tactile allodynia in mice 2012 10.1111/j.1476-5381.2011.01445.x 21506952 http://vivo.scripps.edu/individual/endnote298379
http://vivo.scripps.edu/individual/enote47534 AcademicArticle New insights into the mechanism and an expanded scope of the Fe(III)-mediated vinblastine coupling reaction 2012 10.1021/ja306229x 22856867 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/enote11607 AcademicArticle Silver(I)-promoted conversion of thioamides to amidines: divergent synthesis of a key series of vancomycin aglycon residue 4 amidines that clarify binding behavior to model ligands 2012 10.1021/ja302808p 22568755 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/enote19581 AcademicArticle Divergent total syntheses of (-)-aspidospermine and (+)-spegazzinine 2012 10.1021/ol300599p 22480368 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/enote249169 AcademicArticle Iron(III)/NaBH4-mediated additions to unactivated alkenes: synthesis of novel 20'-vinblastine analogues 2012 10.1021/ol300173v 22369097 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/enote22938 AcademicArticle Discovery of HIV fusion inhibitors targeting gp41 using a comprehensive α-helix mimetic library 2012 10.1016/j.bmcl.2012.02.062 22424973 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/enote194170 AcademicArticle α-Ketoheterocycle-based inhibitors of Fatty Acid Amide Hydrolase (FAAH) 2012 10.1021/cn2001206 22639704 http://vivo.scripps.edu/individual/endnote309398
http://vivo.scripps.edu/individual/enote97165 AcademicArticle Redesign of glycopeptide antibiotics: back to the future 2012 10.1021/cb300007j 22330049 http://vivo.scripps.edu/individual/endnote153903
http://vivo.scripps.edu/individual/enote134419 AcademicArticle Comprehensive peptidomimetic libraries targeting protein-protein interactions 2012 10.1021/ar300025n 22799570 http://vivo.scripps.edu/individual/endnote122847
http://vivo.scripps.edu/individual/e2n350794 AcademicArticle Tetrahedron Young Investigator Award 2011: Carolyn R. Bertozzi 2011 10.1016/j.bmcl.2011.08.013 21840475 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n169388 AcademicArticle Recent advances in medicinal chemistry 2011 10.1016/j.bmcl.2011.04.019 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote198465 AcademicArticle Reversible competitive α-ketoheterocycle inhibitors of fatty acid amide hydrolase containing additional conformational constraints in the acyl side chain: orally active, long-acting analgesics 2011 10.1021/jm101597x 21428410 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote338926 AcademicArticle Scope of the inverse electron demand Diels-Alder reactions of 1,2,3-triazine 2011 10.1021/ol2007428 21488676 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/endnote304212 AcademicArticle A redesigned vancomycin engineered for dual D-Ala-D-ala And D-Ala-D-Lac binding exhibits potent antimicrobial activity against vancomycin-resistant bacteria 2011 10.1021/ja207142h 21823662 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote18737 AcademicArticle Inverse electron demand Diels-Alder reactions of 1,2,3-triazines: Pronounced substituent effects on reactivity and cycloaddition scope 2011 10.1021/ja204856a 21736324 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote59552 AcademicArticle 10 '-fluorovinblastine and 10 '-fluorovincristine: synthesis of a key series of modified vinca alkaloids 2011 10.1021/ml200236a 22247789 http://vivo.scripps.edu/individual/endnote225139
http://vivo.scripps.edu/individual/endnote93884 AcademicArticle Design, synthesis, and validation of a β-turn mimetic library targeting protein-protein and peptide-receptor interactions 2011 10.1021/ja201878v 21609016 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote167443 AcademicArticle The discovery and development of inhibitors of fatty acid amide hydrolase (FAAH) 2011 10.1016/j.bmcl.2011.06.096 21764305 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote45392 AcademicArticle A specific interaction of small molecule entry inhibitors with the envelope glycoprotein complex of the Junin hemorrhagic fever arenavirus 2011 10.1074/jbc.M110.196428 21159779 http://vivo.scripps.edu/individual/endnote308813
http://vivo.scripps.edu/individual/endnote326586 AcademicArticle Asymmetric synthesis of 1,2,9,9a-tetrahydrocyclopropa[c]benzo[e]indol-4-one (CBI) 2011 10.1021/jo102136w 21192653 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote385145 AcademicArticle Synthesis and stereochemical determination of complestatin A and B (neuroprotectin A and B) 2011 10.1021/ja208570q 21991993 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote188397 AcademicArticle Fluoride-mediated capture of a noncovalent bound state of a reversible covalent enzyme inhibitor: X-ray crystallographic analysis of an exceptionally potent α-ketoheterocycle inhibitor of fatty acid amide hydrolase 2011 10.1021/ja110877y 21355555 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n63311 Report Optimization and characterization of a pan protein arginine deiminase (PAD) inhibitor 2010 23833800 http://vivo.scripps.edu/individual/e2n193384
http://vivo.scripps.edu/individual/e7n125296 AcademicArticle Methods to characterize the effect of DNA-modifying compounds on nucleosomal DNA 2010 10.1007/978-1-60327-418-0_11 19997884 http://vivo.scripps.edu/individual/enote13799
http://vivo.scripps.edu/individual/endnote59228 AcademicArticle Total synthesis, assignment of the relative and absolute stereochemistry, and structural reassignment of phostriecin (aka Sultriecin) 2010 10.1021/ja9097252 20108904 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote179882 AcademicArticle Intramolecular 1+2 and 3+2 cycloaddition reactions of cyclopropenone ketals 2010 10.1021/ja103933n 20527885 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote130386 AcademicArticle Total synthesis of (+)-fendleridine (aspidoalbidine) and (+)-1-acetylaspidoalbidine 2010 10.1021/ja908819q 20148585 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote116035 AcademicArticle Synthesis and evaluation of duocarmycin SA analogs incorporating the methyl 1,2,8,8a-tetrahydrocyclopropa[c]oxazolo[2,3-e]indol-4-one-6-carboxylate (COI) alkylation subunit 2010 10.1016/j.bmcl.2010.01.145 20171886 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote27945 AcademicArticle Total synthesis and evaluation of a key series of C5-substituted vinblastine derivatives 2010 10.1021/ja1027748 20518465 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote191718 AcademicArticle Fatty acid amide signaling molecules 2010 10.1016/j.bmcl.2010.08.048 20817522 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote350214 AcademicArticle Synthesis and evaluation of selected key methyl ether derivatives of vancomycin aglycon 2010 10.1021/jm100946e 20853900 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote95806 AcademicArticle Identification of broad-based HIV-1 protease inhibitors from combinatorial libraries 2010 10.1042/bj20091645 20507280 http://vivo.scripps.edu/individual/endnote277207
http://vivo.scripps.edu/individual/endnote346786 AcademicArticle X-ray crystallographic analysis of alpha-ketoheterocycle inhibitors bound to a humanized variant of fatty acid amide hydrolase 2010 10.1021/jm9012196 19924997 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote970 AcademicArticle Catharanthine C16 substituent effects on the biomimetic coupling with vindoline: preparation and evaluation of a key series of vinblastine analogues 2010 10.1016/j.bmcl.2010.09.091 20932748 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote214314 AcademicArticle Synthesis and evaluation of a series of C5'-substituted duocarmycin SA analogs 2010 10.1016/j.bmcl.2010.03.078 20381346 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote271946 AcademicArticle Total synthesis and evaluation of phostriecin and key structural analogues 2010 10.1021/jo1010203 20669916 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote273289 AcademicArticle Asymmetric total synthesis of vindorosine, vindoline, and key vinblastine analogues 2010 10.1021/ja106284s 20809620 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote132574 AcademicArticle Total synthesis of lycogarubin C and lycogalic acid 2010 10.1021/ol100146b 20148525 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/endnote227188 AcademicArticle Asymmetric total synthesis of vindoline 2010 10.1021/ja910695e 20187641 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote207911 AcademicArticle Synthesis and characterization of a cyclobutane duocarmycin derivative incorporating the 1,2,10,11-tetrahydro-9H-cyclobuta[c]benzo[e]indol-4-one (CbBI) alkylation subunit 2010 10.1021/ja106986f 20839806 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote152852 AcademicArticle Small molecule peptidomimetic inhibitors of importin α/β mediated nuclear transport 2010 10.1016/j.bmc.2010.08.038 20869252 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote345470 AcademicArticle Total synthesis of complestatin: development of a Pd(0)-mediated indole annulation for macrocyclization 2010 10.1021/ja102304p 20469945 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote12499 AcademicArticle Design, synthesis, and evaluation of duocarmycin O-amino phenol prodrugs subject to tunable reductive activation 2010 10.1021/jm1010397 20942408 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote225419 AcademicArticle Intramolecular Diels-Alder reactions of cyclopropenone ketals 2010 10.1021/ol101375a 20614867 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/endnote70870 AcademicArticle Binding and inactivation mechanism of a humanized fatty acid amide hydrolase by alpha-ketoheterocycle inhibitors revealed from cocrystal structures 2009 10.1021/ja902694n 19722626 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote240008 AcademicArticle Synthesis and preliminary evaluation of duocarmycin analogues incorporating the 1,2,11,11a-tetrahydrocyclopropa c naphtho 2,3-e indol-4-one (CNI) and 1,2,11,11a-tetrahydrocyclopropa c naphtho 1,2-e indol-4-one (iso-CNI) alkylation subunits 2009 10.1016/j.tet.2009.02.065 20161204 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/endnote245024 AcademicArticle Total synthesis of chloropeptin II (complestatin) and chloropeptin I 2009 10.1021/ja907193b 19839632 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote168002 AcademicArticle Blockade of endocannabinoid-degrading enzymes attenuates neuropathic pain 2009 10.1124/jpet.109.155465 19502530 http://vivo.scripps.edu/individual/endnote398496
http://vivo.scripps.edu/individual/endnote330326 AcademicArticle Characterization of lassa virus cell entry inhibitors: Determination of the active enantiomer by asymmetric synthesis 2009 10.1016/j.bmcl.2009.04.098 19428249 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote13131 AcademicArticle Structure-activity relationship studies of fostriecin, cytostatin, and key analogs, with PP1, PP2A, PP5, and( beta12-beta13)-chimeras (PP1/PP2A and PP5/PP2A), provide further insight into the inhibitory actions of fostriecin family inhibitors 2009 10.1124/jpet.109.155630 19592665 http://vivo.scripps.edu/individual/endnote398496
http://vivo.scripps.edu/individual/endnote178581 AcademicArticle Synthesis and evaluation of vancomycin aglycon analogues that bear modifications in the N-terminal D-leucyl amino acid 2009 10.1021/jm801549b 19209892 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote358052 AcademicArticle Synthesis of the chlorofusin cyclic peptide 2009 10.1016/j.tet.2008.09.029 20047009 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/endnote251334 AcademicArticle Functional and biochemical analysis of a key series of ramoplanin analogues 2009 10.1016/j.bmcl.2009.09.001 19783144 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote247413 AcademicArticle Total synthesis and evaluation of iso-duocarmycin SA and iso-yatakemycin 2009 10.1021/ja808108q 19154178 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote98126 AcademicArticle Total synthesis of vinblastine, vincristine, related natural products, and key structural analogues 2009 10.1021/ja809842b 19292450 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote208457 AcademicArticle Design, synthesis, and evaluation of an α-helix mimetic library targeting protein-protein interactions 2009 10.1021/ja810025g 19334711 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote83423 AcademicArticle Total synthesis of vindoline and related alkaloids 2009 10.5059/yukigoseikyokaishi.67.123 http://vivo.scripps.edu/individual/endnote219041
http://vivo.scripps.edu/individual/endnote207343 AcademicArticle Small molecule inhibitors of Myc/Max dimerization and Myc-induced cell transformation 2009 10.1016/j.bmcl.2009.09.044 19800226 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote163987 AcademicArticle The isolation, total synthesis and structure elucidation of chlorofusin, a natural product inhibitor of the p53-mDM2 protein-protein interaction 2009 10.1039/b821676b 19642417 http://vivo.scripps.edu/individual/endnote292459
http://vivo.scripps.edu/individual/endnote12643 AcademicArticle Discovery of inhibitors of aberrant gene transcription from libraries of DNA binding molecules: Inhibition of LEF-1-mediated gene transcription and oncogenic transformation 2009 10.1021/ja809083d 19216569 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote236543 AcademicArticle Evaluation of chlorofusin, its seven chromophore diastereomers, and key analogues 2009 10.1016/j.tetlet.2009.01.081 20161293 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote308874 AcademicArticle Fundamental relationships between structure, reactivity, and biological activity for the duocarmycins and CC-1065 2009 10.1021/jm9006214 19639994 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote37487 AcademicArticle Synthesis and evaluation of a thio analogue of duocarmycin SA 2009 10.1016/j.bmcl.2009.10.063 19879753 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote183205 AcademicArticle Endocannabinoid modulation of scratching response in an acute allergenic model: a new prospective neural therapeutic target for pruritus 2009 10.1124/jpet.108.150136 19168707 http://vivo.scripps.edu/individual/endnote398496
http://vivo.scripps.edu/individual/endnote310690 AcademicArticle CSI-FID: high throughput label-free detection of DNA binding molecules 2009 10.1016/j.bmcl.2009.04.097 19435662 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote208131 AcademicArticle Direct coupling of catharanthine and vindoline to provide vinblastine: Total synthesis of (+)- and ent-(-)-vinblastine 2008 10.1021/ja078192m 18081297 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote164175 AcademicArticle Unique small molecule entry inhibitors of hemorrhagic fever arenaviruses 2008 10.1074/jbc.M802089200 18474596 http://vivo.scripps.edu/individual/endnote308813
http://vivo.scripps.edu/individual/endnote320240 AcademicArticle Structural features of the (+)-Yatakemycin/d(GACTAATTGAC)-(GTCAATTAGTC) complex: Quantum mechanical calculation of NMR parameters as a tool for the characterization of ligand/DNA Interactions 2008 10.1002/ejoc.200701212 http://vivo.scripps.edu/individual/endnote282598
http://vivo.scripps.edu/individual/endnote230198 AcademicArticle Correlation of inhibitor effects on enzyme activity and thermal stability for the integral membrane protein fatty acid amide hydrolase 2008 10.1016/j.bmcl.2008.06.086 18644727 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote9193 AcademicArticle Yatakemycin: Total synthesis, DNA alkylation, and biological properties 2008 10.1039/b705665f 18389136 http://vivo.scripps.edu/individual/endnote292459
http://vivo.scripps.edu/individual/endnote277167 AcademicArticle Glycinamide ribonucleotide transformylase (GAR Tfase) as a target for cancer therapy 2008 10.1358/dof.2008.33.11.1247542 http://vivo.scripps.edu/individual/endnote288580
http://vivo.scripps.edu/individual/endnote37163 AcademicArticle Disruption of the MYC transcriptional function by a small-molecule antagonist of MYC/MAX dimerization 2008 18288422 http://vivo.scripps.edu/individual/endnote100285
http://vivo.scripps.edu/individual/endnote115125 AcademicArticle Optimization of the central heterocycle of alpha-ketoheterocycle inhibitors of fatty acid amide hydrolase 2008 10.1021/jm800136b 18630870 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote286204 AcademicArticle Asymmetric synthesis of inhibitors of glycinamide ribonucleotide transformylase 2008 10.1021/jm800555h 18686942 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote121561 AcademicArticle An additional spirocyclization for duocarmycin SA 2008 10.1021/ja806593w 19554689 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote184462 AcademicArticle Optimization of alpha-ketooxazole inhibitors of fatty acid amide hydrolase 2008 10.1021/jm701210y 18247553 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote371316 AcademicArticle Exploration of a fundamental substituent effect of α-ketoheterocycle enzyme inhibitors: Potent and selective inhibitors of fatty acid amide hydrolase 2008 10.1016/j.bmcl.2008.06.084 18639454 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote59043 AcademicArticle Total synthesis of chlorofusin, its seven chromophore diastereomers, and key partial structures 2008 10.1021/ja8012819 18712872 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote179836 AcademicArticle Structure-based design, synthesis, evaluation, and crystal structures of transition state analogue inhibitors of inosine monophosphate cyclohydrolase 2007 10.1074/jbc.M607293200 17324932 http://vivo.scripps.edu/individual/endnote308813
http://vivo.scripps.edu/individual/endnote267198 AcademicArticle Potent and selective alpha-ketoheterocycle-based inhibitors of the anandamide and oleamide catabolizing enzyme, fatty acid amide hydrolase 2007 10.1021/jm0611509 17279740 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote62332 AcademicArticle Alanine scan of [L-Dap2]ramoplanin A2 aglycon:  Assessment of the importance of each residue 2007 10.1021/ja068573k 17592838 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote198424 AcademicArticle Structure-activity relationships of alpha-ketooxazole inhibitors of fatty acid amide hydrolase 2007 10.1021/jm061414r 17559203 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote65252 AcademicArticle A unique class of duocarmycin and CC-1065 analogues subject to reductive activation 2007 10.1021/ja075398e 18020335 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote206989 AcademicArticle An in vitro and in vivo disconnect uncovered through high-throughput identification of botulinum neurotoxin A antagonists 2007 10.1073/pnas.0611213104 17293454 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote324261 AcademicArticle Total synthesis, stereochemical reassignment, and absolute configuration of chlorofusin 2007 10.1021/ja073264v 17637057 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote200449 AcademicArticle Systematic exploration of the structural features of yatakemycin impacting DNA alkylation and biological activity 2007 10.1021/ja072777z 17691783 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote190245 AcademicArticle Total synthesis of (-)- and ent-(+)-4-desacetoxy-5-desethylvindoline 2007 10.3987/COM-06-S(K)8 http://vivo.scripps.edu/individual/endnote14559
http://vivo.scripps.edu/individual/endnote337664 AcademicArticle Rational design, synthesis, and evaluation of key analogues of CC-1065 and the duocarmycins 2007 10.1021/ja073989z 17948994 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote258157 AcademicArticle Delineation of a fundamental alpha-ketoheterocycle substituent effect for use in the design of enzyme inhibitors 2006 10.1021/ja064522b 17061864 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote5493 AcademicArticle Total synthesis of (-)- and ent-(+)-vindorosine: Tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition of 1,3,4-oxadiazoles 2006 10.1002/anie.200503024 16355429 http://vivo.scripps.edu/individual/endnote319084
http://vivo.scripps.edu/individual/endnote244550 AcademicArticle Total synthesis of cytostatin 2006 10.3987/COM-06-S(W)13 http://vivo.scripps.edu/individual/endnote14559
http://vivo.scripps.edu/individual/endnote182395 AcademicArticle Asymmetric total synthesis of (+)- and ent-(-)-yatakemycin and duocarmycin SA: evaluation of yatakemycin key partial structures and its unnatural enantiomer 2006 10.1021/ja064228j 17147378 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote203649 AcademicArticle Discovery of a potent, nonpolyglutamatable inhibitor of glycinamide ribonucleotide transformylase 2006 10.1021/jm0601147 16686541 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote66316 AcademicArticle The mechanism of action of ramoplanin and enduracidin 2006 10.1039/b515328j 16880924 http://vivo.scripps.edu/individual/endnote93661
http://vivo.scripps.edu/individual/endnote246390 AcademicArticle Total synthesis of (-)- and ent-(+)-vindoline and related alkaloids 2006 10.1021/ja061256t 16895428 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote206198 AcademicArticle Total synthesis and evaluation of [Ψ[CH(2)NH]Tpg(4)]vancomycin aglycon: reengineering vancomycin for dual D-Ala-D-Ala and D-Ala-D-Lac binding 2006 10.1021/ja0572912 16506767 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote159164 AcademicArticle Diastereoselective Diels-Alder reactions of N-sulfonyl-1-aza-1,3-butadienes with optically active enol ethers: An asymmetric variant of the 1-azadiene Diels-Alder reaction 2006 10.1021/ja0571646 16492042 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote17487 AcademicArticle Total synthesis of piericidin A1 and B1 and key analogues 2006 10.1021/ja0632862 16953619 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote187884 AcademicArticle Alkylation of duplex DNA in nucleosome core particles by duocarmycin SA and yatakemycin 2006 10.1038/nchembio761 16415862 http://vivo.scripps.edu/individual/endnote16708
http://vivo.scripps.edu/individual/endnote19183 AcademicArticle Two novel 1,2,4,5-tetrazines that participate in inverse electron demand Diels-Alder reactions with an unexpected regioselectivity 2006 10.1021/jo051832o 16388634 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote394364 AcademicArticle Intramolecular Diels-Alder/1,3-dipolar cycloaddition cascade of 1,3,4-oxadiazoles 2006 10.1021/ja0612549 16895427 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote19249 AcademicArticle Total synthesis and evaluation of cytostatin, its C10-C11 diastereomers, and additional key analogues: Impact on PP2A inhibition 2006 10.1021/ja066477d 17177422 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n328144 AcademicArticle Bioorganic & Medicinal Chemistry Letters Symposia-in-Print 2005 10.1016/j.bmcl.2005.07.002 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote136021 AcademicArticle Discovery of a potent, selective, and efficacious class of reversible alpha-ketoheterocycle inhibitors of fatty acid amide hydrolase effective as analgesics 2005 10.1021/jm049614v 15771430 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote120777 AcademicArticle Chemistry and biology of ramoplanin: A lipoglycodepsipeptide with potent antibiotic activity 2005 10.1021/cr030106n 15700952 http://vivo.scripps.edu/individual/endnote51983
http://vivo.scripps.edu/individual/endnote258061 AcademicArticle Elucidation of fatty acid amide hydrolase inhibition by potent alpha-ketoheterocycle derivatives from Monte Carlo simulations 2005 10.1021/ja055438j 16332087 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote287545 AcademicArticle Design, synthesis, and biological evaluation of 10-methanesulfonyl-DDACTHF, 10-methanesulfonyl-5-DACTHF, and 10-methylthio-DDACTHF as potent inhibitors of GAR Tfase and the de novo purine biosynthetic pathway 2005 10.1016/j.bmc.2004.12.004 15848770 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote289349 AcademicArticle Synthesis and biological evaluation of α- and γ-carboxamide derivatives of 10-CF3CO-DDACTHF 2005 10.1016/j.bme.2004.11.050 15848771 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote125136 AcademicArticle Discovery of an exceptionally potent and selective class of fatty acid amide hydrolase inhibitors enlisting proteome-wide selectivity screening: concurrent optimization of enzyme inhibitor potency and selectivity 2005 10.1016/j.bmcl.2004.12.085 15713400 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote67107 AcademicArticle Heterocyclic sulfoxide and sulfone inhibitors of fatty acid amide hydrolase 2005 10.1016/j.bmcl.2004.10.025 15582420 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote92329 AcademicArticle Total synthesis of piericidin A1 and B1 2005 10.1021/ja055041f 16277503 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote63204 AcademicArticle Discovery of aicar tfase inhibitors that disrupt requisite enzyme dimerization 2005 10.1016/j.bcml.2005.03.094 15911265 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote50866 AcademicArticle Potent reversal of multidrug resistance by ningalins and its use in drug combinations against human colon carcinoma xenograft in nude mice 2005 10.1007/s00280-005-1019-y 15875185 http://vivo.scripps.edu/individual/endnote235495
http://vivo.scripps.edu/individual/endnote291060 AcademicArticle Synthesis and biological evaluation of N-{4- 5-(2,4-diamino-6-oxo-1,6-dihydropyrimidin-5-yl)-2-(2,2,2-trifluoro acetyl)pentyl)benzoyl}-L-glutamic acid as a potential inhibitor of GAR Tfase and the de novo purine biosynthetic pathway 2005 10.1016/j.bme.2004.11.049 15848772 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote294251 AcademicArticle Total synthesis of (-)- and ent-(+)-vindoline 2005 10.1021/o1051975x 16178578 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/endnote238354 AcademicArticle Total synthesis of ningalin D 2005 10.1021/ja0526416 16045367 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote251755 AcademicArticle Total synthesis of natural (-)- and ent-(+)-4-desacetoxy-6,7-dihydrovindorosine and natural and ent-minovine: Oxadiazole tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition reaction 2005 10.1021/ol050017s 15704939 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/endnote9036 AcademicArticle Sequence-selective DNA recognition: natural products and nature's lessons 2004 10.1016/j.chembiol.2003.08.012 15610844 http://vivo.scripps.edu/individual/endnote342045
http://vivo.scripps.edu/individual/endnote304860 AcademicArticle A fluorescent intercalator displacement assay for establishing DNA binding selectivity and affinity 2004 10.1021/ar030113y 14730995 http://vivo.scripps.edu/individual/endnote122847
http://vivo.scripps.edu/individual/endnote144263 AcademicArticle A powerful selection assay for mixture libraries of DNA alkylating agents 2004 10.1021/ja0477930 15281804 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote76671 AcademicArticle Total synthesis, structure revision, and absolute configuration of (+)-yatakemycin 2004 10.1021/ja0472735 15237994 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote8937 AcademicArticle Total synthesis and examination of three key analogues of ramoplanin: a lipoglycodepsipeptide with potent antibiotic activity 2004 10.1021/ja039671y 14746470 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote282893 AcademicArticle Dissecting ramoplanin: mechanistic analysis of synthetic ramoplanin analogues as a guide to the design of improved antibiotics 2004 10.1021/ja047879t 15198592 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote79055 AcademicArticle A human single-chain antibody specific for integrin alpha(3)beta(1) capable of cell internalization and delivery of antitumor agents 2004 10.1016/j.chembiol.2004.04.018 15271348 http://vivo.scripps.edu/individual/endnote342045
http://vivo.scripps.edu/individual/endnote173920 AcademicArticle Establishing the parabolic relationship between reactivity and activity for derivatives and analogues of the duocarmycin and CC-1065 alkylation subunits 2004 10.1021/ja038162t 14709069 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote332968 AcademicArticle Reversible inhibitors of fatty acid amide hydrolase that promote analgesia: evidence for an unprecedented combination of potency and selectivity 2004 10.1124/jpet.104.069401 15229230 http://vivo.scripps.edu/individual/endnote398496
http://vivo.scripps.edu/individual/endnote310066 AcademicArticle Total synthesis and structure of the ramoplanin A1 and A3 aglycons: two minor components of the ramoplanin complex 2004 10.1073/pnas.0401419101 15175429 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote267028 AcademicArticle Effective asymmetric synthesis of 1,2,9,9a-tetrahydrocyclopropa c benzo e indol-4-one (cbi) 2004 10.1021/jo035465x 15049620 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote296935 AcademicArticle Energetic preferences for alpha,beta versus beta,gamma unsaturation 2004 10.1021/jo049365y 15287795 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote288887 AcademicArticle Synthesis and evaluation of N-aryl and N-alkenyl CBI derivatives 2004 10.1016/j.bmc.2004.08.032 15498660 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote231971 AcademicArticle Total synthesis of the ristocetin aglycon 2004 10.1021/ja039795a 15053621 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote301033 AcademicArticle Multidrug resistance reversal activity of permethyl ningalin B amide derivatives 2004 10.1016/j.bmcl.2004.10.002 15546712 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote352787 AcademicArticle Synthesis of the chlorofusin cyclic peptide: assignment of the asparagine stereochemistry 2003 10.1021/ol036083g 14682761 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/endnote93713 AcademicArticle Comprehensive high-resolution analysis of hairpin polyamides utilizing a fluorescent intercalator displacement (FID) assay 2003 10.1016/s0968-0896(03)00455-3 13129584 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote357622 AcademicArticle Synthesis and inverse electron demand Diels-Alder reactions of 3,6-bis(3,4-dimethoxybenzoyl)-1,2,4,5-tetrazine 2003 10.1021/jo020713v 12713365 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote35698 AcademicArticle Multidrug resistance reversal activity of key ningalin analogues 2003 10.1016/s0960-894x(03)00294-4 12729663 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote62339 AcademicArticle 10-(2-benzoxazolcarbonyl)-5,10-dideaza-acyclic-5,6,7,8-tetrahydrofolic acid: a potential inhibitor of GAR transformylase and AICAR transformylase 2003 10.1016/s0968-0896(03)00457-7 13129586 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote201679 AcademicArticle Synthesis of the (S,S,S)-diastereomer of the 15-membered biaryl ring system of RP 66453 2003 10.1016/s0040-4039(03)00856-6 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote160952 AcademicArticle NMR structure of the (+)-CPI-indole/d(GACTAATTGAC)-d(GTCAATTAGTC) covalent complex 2003 10.1002/cbic.200300642 14613110 http://vivo.scripps.edu/individual/e2n264100
http://vivo.scripps.edu/individual/endnote89489 AcademicArticle A new and improved method for deglycosidation of glycopeptide antibiotics exemplified with vancomycin, ristocetin, and ramoplanin 2003 10.1016/s0960-894x(03)00051-9 12643936 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote108126 AcademicArticle High-resolution assessment of protein DNA binding affinity and selectivity utilizing a fluorescent intercalator displacement (FID) assay 2003 10.1016/j.bmcl.2003.06.002 14552784 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote399934 AcademicArticle Synthesis of isochrysohermidin-distamycin hybrids 2003 10.1021/jo034326c 12816485 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote165310 AcademicArticle Synthesis and evaluation of methyl ether derivatives of the vancomycin, teicoplanin, and ristocetin aglycon methyl esters 2003 10.1016/s0960-894x(03)00513-4 14611861 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote43335 AcademicArticle Determination of binding affinities of triplex forming oligonucleotides using a fluorescent intercalator displacement (FID) assay 2003 10.1016/j.bmcl.2003.07.005 14552783 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote63515 AcademicArticle Solution-phase synthesis of combinatorial libraries designed to modulate protein-protein or protein-DNA interactions 2003 10.1016/s0968-0896(03)00031-2 12659745 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote206837 AcademicArticle Discovering potent and selective reversible inhibitors of enzymes in complex proteomes 2003 10.1038/nbt826 12740587 http://vivo.scripps.edu/individual/endnote208688
http://vivo.scripps.edu/individual/endnote7829 AcademicArticle Fundamental role of the fostriecin unsaturated lactone and implications for selective protein phosphatase inhibition 2003 10.1021/ja038672n 14677930 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote210880 AcademicArticle Synthesis and X-ray analysis of an unprecedented and stable 2-aza-4,4-spirocyclopropacyclohexadienone 2003 10.1021/ol035000t 12841785 http://vivo.scripps.edu/individual/endnote341245
http://vivo.scripps.edu/individual/endnote163232 AcademicArticle DNA alkylation properties of yatakemycin 2003 10.1021/ja035984h 12952479 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote147585 AcademicArticle Design, synthesis and biological evaluation of 10-CF3CO-DDACTHF analogues and derivatives as inhibitors of GAR Tfase and the de novo purine biosynthetic pathway 2003 10.1016/s0968-0896(03)00458-9 13129587 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote292242 AcademicArticle Total synthesis of the ramoplanin a2 and ramoplanose aglycon 2003 10.1021/ja0212314 12580615 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote275708 AcademicArticle Establishment of substituent effects in the DNA binding subunit of CBI analogues of the duocarmycins and CC-1065 2003 10.1016/s0968-0896(03)00194-9 12901927 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote180327 AcademicArticle Synthesis and evaluation of duocarmycin and CC-1065 analogues incorporating the 1,2,9,9a-tetrahydrocyclopropa c benz e -3-azaindol-4-one (CBA) alkylation subunit 2003 10.1021/jo035119f 14604371 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote172922 AcademicArticle Design, synthesis, and biological evaluation of simplified alpha-keto heterocycle, trifluoromethyl ketone, and formyl substituted folate analogues as potential inhibitors of GAR transformylase and AICAR transformylase 2003 10.1016/s0968-0896(03)00456-5 13129585 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote359072 AcademicArticle Rational design, synthesis, evaluation, and crystal structure of a potent inhibitor of human GAR Tfase: 10-(trifluoroacetyl)-5,10-dideazaacyclic-5,6,7,8-tetrahydrofolic acid 2003 10.1021/bi034219c 12755606 http://vivo.scripps.edu/individual/endnote165634
http://vivo.scripps.edu/individual/endnote79506 AcademicArticle Solution-phase combinatorial libraries: modulating cellular signaling by targeting protein-protein or protein-DNA interactions 2003 10.1002/anie.200300574 14502729 http://vivo.scripps.edu/individual/endnote319084
http://vivo.scripps.edu/individual/endnote331747 AcademicArticle Partitioning the loss in vancomycin binding affinity for D-Ala-D-Lac into lost H-bond and repulsive lone pair contributions 2003 10.1021/ja035901x 12889959 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote343214 AcademicArticle Small-molecule antagonists of Myc/Max dimerization inhibit Myc-induced transformation of chicken embryo fibroblasts 2002 10.1073/pnas.062036999 11891322 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote4164 AcademicArticle Preparation of the 14-membered L,L-cycloisodityrosine subunit of RP 66453 2002 10.1016/s0040-4039(01)02194-3 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote262372 AcademicArticle Erythropoietin mimetics derived from solution phase combinatorial libraries 2002 10.1021/ja0118789 11804483 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote94295 AcademicArticle Synthesis and DNA binding properties of iminodiacetic acid-linked polyamides: characterization of cooperative extended 2 : 1 side-by-side parallel binding 2002 10.1021/ja026588m 12207521 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote322034 AcademicArticle Mechanisms of in situ activation for DNA-targeting antitumor agents 2002 10.1021/cr010046q 12105933 http://vivo.scripps.edu/individual/endnote51983
http://vivo.scripps.edu/individual/endnote109717 AcademicArticle Synthesis and evaluation of vancomycin and vancomycin aglycon analogues that bear modifications in the residue 3 asparagine 2002 10.1016/s0960-894x(02)00130-0 11965380 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote317615 AcademicArticle Inhibitors of cell migration that inhibit intracellular paxillin/alpha a binding: A well-documented use of positional scanning libraries 2002 10.1016/s1074-5521(02)00246-6 12445772 http://vivo.scripps.edu/individual/endnote342045
http://vivo.scripps.edu/individual/endnote314513 AcademicArticle Solution-phase parallel synthesis of a pharmacophore library of hun-7293 analogues: a general chemical mutagenesis approach to defining structure-function properties of naturally occurring cyclic (depsi)peptides 2002 10.1021/ja020166v 11996584 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote276137 AcademicArticle Synthesis and DNA binding properties of saturated distamycin analogues 2002 10.1016/s0960-894x(02)00467-5 12182879 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote73363 AcademicArticle Fostriecin: Chemistry and biology 2002 12369868 http://vivo.scripps.edu/individual/endnote178003
http://vivo.scripps.edu/individual/endnote46956 AcademicArticle Total synthesis of anhydrolycorinone utilizing sequential intramolecular Diels-Alder reactions of a 1,3,4-oxadiazole 2002 10.1021/jo030437k 12375965 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote188582 AcademicArticle Total synthesis of the ramoplanin a2 and ramoplanose aglycon 2002 10.1021/ja020237q 11996568 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote114633 AcademicArticle Intramolecular Diels-Alder and tandem intramolecular Diels-Alder/1,3-dipolar cycloaddition reactions of 1,3,4-oxadiazoles 2002 10.1021/ja027533n 12236743 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote384272 AcademicArticle Crystal structures of human GAR Tfase at low and high pH and with substrate β-GAR 2002 10.1021/bi020522m 12450384 http://vivo.scripps.edu/individual/endnote165634
http://vivo.scripps.edu/individual/endnote268759 AcademicArticle The DNA phosphate backbone is not involved in catalysis of the duocarmycin and CC-1065 DNA alkylation reaction 2002 10.1016/s0960-894x(01)00740-5 11814783 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote34329 AcademicArticle 10-formyl-5,10-dideaza-acyclic-5,6,7,8-tetrahydrofolic acid (10-formyl-DDACTHF): a potent cytotoxic agent acting by selective inhibition of human GAR Tfase and the de novo purine biosynthetic pathway 2002 10.1016/s0968-0896(02)00102-5 12057663 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote41441 AcademicArticle Total synthesis of (+)-camptothecin 2002 10.1016/s0040-4020(02)00633-6 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/endnote279320 AcademicArticle Hairpin versus extended DNA binding of a substituted beta-alanine linked polyamide 2002 10.1021/ja0122039 11878968 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote21263 AcademicArticle Total syntheses of thiocoraline and be-22179 and assessment of their DNA binding and biological properties 2001 10.1021/ja003602r 11456568 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote121063 AcademicArticle Synthesis and evaluation of a series of C3-substituted CBI analogues of CC-1065 and the duocarmycins 2001 10.1021/jo010309g 11463270 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote384073 AcademicArticle Synthesis, chemical properties, and biological evaluation of CC-1065 and duocarmycin analogues incorporating the 5-methoxycarbonyl-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one alkylation subunit 2001 10.1021/jo001772g 11281757 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote203640 AcademicArticle Disruption of matrix metalloproteinase 2 binding to integrin alpha(v)beta(3) by an organic molecule inhibits angiogenesis and tumor growth in vivo 2001 10.1073/pnas.011343298 11134507 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote249578 AcademicArticle Identification of a novel class of small-molecule antiangiogenic agents through the screening of combinatorial libraries which function by inhibiting the binding and localization of proteinase MMP2 to integrin alpha(V)beta(3) 2001 10.1021/ja003579+ 11456699 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote286887 AcademicArticle Alpha-Keto heterocycle inhibitors of fatty acid amide hydrolase: carbonyl group modification and alpha-substitution 2001 10.1016/s0960-894x(01)00211-6 11412972 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote70838 AcademicArticle Substituent effects within the DNA binding subunit of CBI analogues of the duocarmycins and CC-1065 2001 10.1016/s0960-894x(01)00372-9 11454471 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote4989 AcademicArticle Thiazole orange as the fluorescent intercalator in a high resolution fid assay for determining DNA binding affinity and sequence selectivity of small molecules 2001 10.1016/s0968-0896(01)00243-7 11553493 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote277003 AcademicArticle Metal cation complexation and activation of reversed CPyi analogues of CC-1065 and duocarmycin SA: Partitioning the effects of binding and catalysis 2001 10.1021/ja010769r 11562212 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote242915 AcademicArticle Cytokine receptor dimerization and activation: prospects for small molecule agonists 2001 10.1016/s0968-0896(00)00276-5 11310589 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote225790 AcademicArticle Parallel synthesis and evaluation of 132 (+)-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (CBI) analogues of CC-1065 and the duocarmycins defining the contribution of the DNA-binding domain 2001 10.1021/jo010454u 11578217 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote138294 AcademicArticle A simple, high-resolution method for establishing DNA binding affinity and sequence selectivity 2001 10.1021/ja010041a 11414820 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote124062 AcademicArticle First and second generation total synthesis of the teicoplanin aglycon 2001 10.1021/ja003835i 11456806 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote111578 AcademicArticle Recent advances in bioorganic and medicinal chemistry. Preface. 2001 10.1016/s0960-894x(01)00337-7 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote286284 AcademicArticle Vancomycin, teicoplanin, and ramoplanin: Synthetic and mechanistic studies 2001 10.1002/med.1014 11579438 http://vivo.scripps.edu/individual/endnote50744
http://vivo.scripps.edu/individual/endnote216314 AcademicArticle Asymmetric total synthesis of ent-(-)-roseophilin: Assignment of absolute configuration 2001 10.1021/ja011271s 11525659 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote128105 AcademicArticle Unexpected formation of an epoxide-derived multisubstrate adduct inhibitor on the active site of GAR transformylase 2001 10.1021/bi011482+ 11695901 http://vivo.scripps.edu/individual/endnote165634
http://vivo.scripps.edu/individual/endnote47587 AcademicArticle Behavioral evidence for the interaction of oleamide with multiple neurotransmitter systems 2001 11561096 http://vivo.scripps.edu/individual/endnote398496
http://vivo.scripps.edu/individual/endnote151661 AcademicArticle Alternative synthesis and thermal atropisomerism of a fully functionalized DEFG ring system of teicoplanin 2001 10.1016/s0040-4039(01)01199-6 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote374953 AcademicArticle Total synthesis of fostriecin (CI-920) 2001 10.1021/ja010195q 11457179 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote89251 AcademicArticle Total syntheses of thiocoraline and be-22179: Establishment of relative and absolute stereochemistry 2000 10.1021/ja0001660 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote182597 AcademicArticle Synthesis and evaluation of 1,2,8, 8a-Tetrahydrocyclopropa[c]pyrrolo[3,2-e]indol-4(5H)-one, the parent alkylation subunit of CC-1065 and the duocarmycins: impact of the alkylation subunit substituents and its implications for DNA alkylation catalysis 2000 10.1021/jo000297j 10866627 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote357589 AcademicArticle Development of a solution-phase synthesis of minor groove binding bis-intercalators based on triostin A suitable for combinatorial synthesis 2000 10.1021/jo000382r 10987932 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote116495 AcademicArticle Total synthesis of distamycin A and 2640 analogues: A solution-phase combinatorial approach to the discovery of new, bioactive DNA binding agents and development of a rapid, high-throughput screen for determining relative DNA binding affinity or DNA binding sequence selectivity 2000 10.1021/ja994192d http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote151989 AcademicArticle Design, synthesis, and biological evaluation of fluoronitrophenyl substituted folate analogues as potential inhibitors of GAR transformylase and AICAR transformylase 2000 10.1016/s0960-894x(00)00271-7 10888335 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote74082 AcademicArticle Exceptionally potent inhibitors of fatty acid amide hydrolase: the enzyme responsible for degradation of endogenous oleamide and anandamide 2000 10.1073/pnas.97.10.5044 10805767 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote185537 AcademicArticle Total synthesis of the rubrolone aglycon 2000 10.1021/ja002997b http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote265356 AcademicArticle Fatty acid amide hydrolase substrate specificity 2000 10.1016/s0960-894x(00)00528-x 11128635 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote129079 AcademicArticle Two comparisons of the performance of positional scanning and deletion synthesis for the identification of active constituents in mixture combinatorial libraries 2000 10.1021/jo9916481 10814111 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote229545 AcademicArticle Assessment of solution-phase positional scanning libraries based on distamycin A for the discovery of new DNA binding agents 2000 10.1016/s0968-0896(00)00137-1 11003149 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote266305 AcademicArticle Synthesis and evaluation of a novel bleomycin A(2) analogue: Continuing assessment of the linker domain 2000 10.1016/s0040-4039(00)01633-6 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote217191 AcademicArticle Asymmetric synthesis of orthogonally protected L-threo-beta-hydroxyasparagine 2000 10.1021/jo000628s 11052134 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote317012 AcademicArticle A new class of highly cytotoxic diketopiperazines 2000 10.1016/s0960-894x(00)00152-9 10843206 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote162686 AcademicArticle Selective metal cation activation of a DNA alkylating agent: Synthesis and evaluation of methyl 1,2,9,9a-Tetrahydrocyclopropa c pyrido 3,2-e indol-4-one-7-carboxylate (CPyl) 2000 10.1021/jo000177b 10866626 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote351894 AcademicArticle Conformationally restricted analogues designed for selective inhibition of GAR Tfase versus thymidylate synthase or dihydrofolate reductase 2000 10.1016/s0968-0896(00)00051-1 10882019 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote20485 AcademicArticle The structural basis for in situ activation of DNA alkylation by duocarmycin sa 2000 10.1006/jmbi.2000.3887 10903864 http://vivo.scripps.edu/individual/endnote261742
http://vivo.scripps.edu/individual/endnote369655 AcademicArticle Thermal atropisomerism of teicoplanin aglycon derivatives: Preparation of the P,P,P and M,P,P atropisomers of the teicoplanin aglycon via selective equilibration of the DE ring system 2000 10.1021/ja002376i http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote149655 AcademicArticle Bifunctional alkylating agents derived from duocarmycin SA: Potent antitumor activity with altered sequence selectivity 2000 10.1016/s0960-894x(00)00042-1 10743956 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote233289 AcademicArticle Total synthesis of the teicoplanin aglycon 2000 10.1021/ja001663j http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote176668 AcademicArticle Synthesis and evaluation of aza HUN-7293 2000 10.1016/s0960-894x(00)00336-x 10937737 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote12566 AcademicArticle Total synthesis of ningalin B utilizing a heterocyclic azadiene Diels-Alder reaction and discovery of a new class of potent multidrug resistant (MDR) reversal agents 2000 10.1021/jo9916535 10789460 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote123072 AcademicArticle Total synthesis of Amaryllidaceae alkaloids utilizing sequential intramolecular heterocyclic azadiene Diels-Alder reactions of an unsymmetrical 1,2,4,5-tetrazine 2000 10.1021/jo0012546 11149859 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote239483 AcademicArticle A new method of in situ activation for a novel class of DNA alkylating agents: tunable metal cation complexation and activation 2000 10.1021/ja000653f http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote112830 AcademicArticle Non-amide-based combinatorial libraries derived from N-BOC-iminodiacetic acid: solution-phase synthesis of piperazinone libraries with activity against LEF-1/β-catenin-mediated transcription 2000 10.1002/1522-2675(20000809)83:8<1825::aid-hlca1825>3.0.co;2-4 http://vivo.scripps.edu/individual/endnote350717
http://vivo.scripps.edu/individual/endnote187932 AcademicArticle Total synthesis and comparative evaluation of luzopeptin A-C and quinoxapeptin A-C 1999 10.1021/ja993019e http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote279965 AcademicArticle A novel class of CC-1065 and duocarmycin analogues subject to mitomycin-related reductive activation 1999 10.1021/jo991301y 11674758 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote348860 AcademicArticle Total synthesis of luzopeptins A-C 1999 10.1021/ja983925b http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote225088 AcademicArticle CBI prodrug analogs of CC-1065 and the duocarmycins 1999 http://vivo.scripps.edu/individual/endnote215025
http://vivo.scripps.edu/individual/endnote353539 AcademicArticle Shape-dependent catalysis: Insights into the source of catalysis for the CC-1065 and duocarmycin DNA alkylation reaction 1999 10.1021/ar9800946 http://vivo.scripps.edu/individual/endnote122847
http://vivo.scripps.edu/individual/endnote45497 AcademicArticle N-acylglycine amidation: implications for the biosynthesis of fatty acid primary amides 1999 10.1021/bi982255j 10079066 http://vivo.scripps.edu/individual/endnote165634
http://vivo.scripps.edu/individual/endnote168914 AcademicArticle Total synthesis of quinoxapeptin A-C: Establishment of absolute stereochemistry 1999 10.1002/(sici)1521-3773(19990816)38:16<2424::aid-anie2424>3.0.co;2-9 10458810 http://vivo.scripps.edu/individual/endnote319084
http://vivo.scripps.edu/individual/endnote228432 AcademicArticle Total synthesis of the vancomycin aglycon 1999 10.1021/ja992577q http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote176165 AcademicArticle Trifluoromethyl ketone inhibitors of fatty acid amide hydrolase: a probe of structural and conformational features contributing to inhibition 1999 10.1016/s0960-894x(98)00734-3 10021942 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote377764 AcademicArticle Total synthesis of phomazarin 1999 10.1021/ja983631q http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote184660 AcademicArticle Total synthesis of HUN-7293 1999 10.1021/ja990918u http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote170614 AcademicArticle Solution phase combinatorial synthesis of biaryl libraries employing heterogeneous conditions for catalysis and isolation with size exclusion chromatography for purification 1999 10.1021/jo982234v http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote96922 AcademicArticle Resolution of a CPzl precursor, synthesis and biological evaluation of (+) and (-)-NBoc-CPzl: a further validation of the relationship between chemical solvolytic stability and cytotoxicity 1999 10.1016/s0960-894x(99)00533-8 10560730 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote218088 AcademicArticle Arachidonic acid amide inhibitors of gap junction cell-cell communication 1999 10.1016/s0960-894x(99)00148-1 10328303 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote341174 AcademicArticle Convergent solution-phase combinatorial synthesis with multiplication of diversity through rigid biaryl and diarylacetylene couplings 1999 10.1021/jo990639p http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote247939 AcademicArticle Vancomycin CD and DE macrocyclization and atropisomerism studies 1999 10.1021/jo980880o 11674087 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote171910 AcademicArticle Are the duocarmycin and CC-1065 DNA alkylation reactions acid-catalyzed? Solvolysis pH-rate profiles suggest they are not 1999 10.1021/jo990762g 11674637 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote62791 AcademicArticle Diastereoselective total synthesis of the vancomycin aglycon with ordered atropisomer equilibrations 1999 10.1021/ja990189i http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote35031 AcademicArticle Synthesis and evaluation of duocarmycin and CC-1065 analogues containing modifications in the subunit linking amide 1999 10.1021/jo990452y http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote226505 AcademicArticle Binding-induced activation of DNA alkylation by duocarmycin SA: Insights from the structure of an indole derivative-DNA adduct 1999 10.1021/ja983556j http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote72941 AcademicArticle Total syntheses of ningalin A, lamellarin O, lukianol A, and permethyl storniamide A utilizing heterocyclic azadiene Diels-Alder reactions 1999 10.1021/ja982078+ http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote84645 AcademicArticle New insights into inhibitor design from the crystal structure and NMR studies of escherichia coli GAR and 10-formyl-5,8,10-trideazafolic acid 1999 10.1021/bi991888a 10606510 http://vivo.scripps.edu/individual/endnote165634
http://vivo.scripps.edu/individual/endnote223713 AcademicArticle Bleomycin: synthetic and mechanistic studies 1999 10.1002/(sici)1521-3773(19990215)38:4<448::aid-anie448>3.0.co;2-w http://vivo.scripps.edu/individual/endnote319084
http://vivo.scripps.edu/individual/endnote321743 AcademicArticle DNA binding properties of key sandramycin analogues: systematic examination of the intercalation chromophore 1999 10.1016/s0968-0896(98)00206-5 10218823 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/e2n367672 AcademicArticle Combinatorial chemistry 1998 10.1016/s0960-894x(98)90007-5 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e7n84380 AcademicArticle The first synthesis of a daphnane diterpene: the enantiocontrolled total synthesis of (+)-resiniferatoxin 1998 http://vivo.scripps.edu/individual/e7n18490
http://vivo.scripps.edu/individual/endnote150799 AcademicArticle Thermal atropisomerism of aglucovancomycin derivatives: preparation of (M,M,M)- and (P,M,M)-aglucovancomycins 1998 10.1021/ja981928i http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote398787 AcademicArticle Solution-phase combinatorial synthesis: Convergent multiplication of diversity via the olefin metathesis reaction 1998 10.1016/s0040-4020(98)00128-8 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/endnote82992 AcademicArticle Synthesis of acyclic precursors to (3S,4S)-4-hydroxy-2,3,4,5-tetrahydro-pyridazine-3-carboxylic acid and incorporation into a luzopeptin/quinoxapeptin dipeptide 1998 10.1021/jo980765d 11672282 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote371226 AcademicArticle Heterocyclic and acyclic azadiene Diels-Alder reactions: total synthesis of nothapodytine B 1998 10.1002/jhet.5570350502 http://vivo.scripps.edu/individual/endnote355769
http://vivo.scripps.edu/individual/endnote211351 AcademicArticle An endogenous sleep-inducing compound is a novel competitive inhibitor of fatty acid amide hydrolase 1998 10.1016/s0960-894x(98)00073-0 9871570 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote322623 AcademicArticle Chemical requirements for inhibition of gap junction communication by the biologically active lipid oleamide 1998 10.1073/pnas.95.9.4810 9560184 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote139070 AcademicArticle Higher order iminodiacetic acid libraries for probing protein-protein interactions 1998 10.1016/s0960-894x(98)00423-5 9873538 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote3246 AcademicArticle Design, synthesis, and evaluation of potential GAR and AICAR transformylase inhibitors 1998 10.1016/s0968-0896(98)00040-6 9681131 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote233392 AcademicArticle Synthesis and evaluation of a carbocyclic analogue of the CC-1065 and duocarmycin alkylation subunits: role of the vinylogous amide and implications on DNA alkylation catalysis 1998 10.1021/jo981698q http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote195891 AcademicArticle Synthesis of the vancomycin CDE ring system 1998 10.1016/s0960-894x(98)00110-3 9871529 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote103386 AcademicArticle Regioselective inverse electron demand Diels-Alder reactions of N-acyl 6-amino-3-(methylthio)-1,2,4,5-tetrazines 1998 10.1021/jo980795g 11672266 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote240228 AcademicArticle NMR studies of Co.deglycoBleomycin A2 green and its complex with d(CCAGGCCTGG) 1998 10.1021/ja972125i http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote282523 AcademicArticle Assessment of the role of the bleomycin A(2) pyrimidoblamic acid C4 amino group 1998 10.1021/ja971889v http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote258490 AcademicArticle Critical role of the linking amide in CC-1065 and the duocarmycins: implications on the source of DNA alkylation catalysis 1998 10.1021/ja9818093 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote249563 AcademicArticle Structural requirements for 5-HT2A and 5-HT1A serotonin receptor potentiation by the biologically active lipid oleamide 1998 10.1073/pnas.95.8.4102 9539697 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote216022 AcademicArticle Synthesis of key sandramycin analogs: Systematic examination of the intercalation chromophore 1998 10.1016/s0968-0896(97)10014-1 9502108 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote312787 AcademicArticle Definition of the effect and role of the bleomycin A(2) valerate substituents: preorganization of a rigid, compact conformation implicated in sequence-selective DNA cleavage 1998 10.1021/ja9816640 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote25122 AcademicArticle A systematic evaluation of the bleomycin A(2) L-threonine side chain: its role in preorganization of a compact conformation implicated in sequence-selective DNA cleavage 1998 10.1021/ja9816638 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote140851 AcademicArticle Oleamide: an endogenous sleep-inducing lipid and prototypical member of a new class of biological signaling molecules 1998 10197045 http://vivo.scripps.edu/individual/endnote248220
http://vivo.scripps.edu/individual/endnote196859 AcademicArticle Higher order iminodiacetic acid libraries for probing protein-protein interactions 1998 10.1016/s0968-0896(98)00128-x 9784874 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote164535 AcademicArticle Synthesis of CC-1065 and duocarmycin analogs via intramolecular aryl radical cyclization of a tethered vinyl chloride 1998 10.1016/s0040-4039(98)00232-9 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote388085 AcademicArticle Multistep convergent solution-phase combinatorial synthesis and deletion synthesis deconvolution 1998 10.1021/ja9803557 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote47504 AcademicArticle Total synthesis of nothapodytine B and (-)-mappicine 1998 10.1021/ja973007y http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e7n368030 AcademicArticle Solution structures of Co·Bleomycin A2 green and its complex with d(CCAGGCCTGG)​2 1997 http://vivo.scripps.edu/individual/e7n18490
http://vivo.scripps.edu/individual/endnote63378 AcademicArticle Total synthesis of (+)-duocarmycin A, epi-(+)-duocarmycin A and their unnatural enantiomers: assessment of chemical and biological properties 1997 10.1021/ja962431g http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote9779 AcademicArticle pH dependence of the rate of DNA alkylation for (+)-duocarmycin SA and (+)-CCBI-TMI 1997 10.1016/s0960-894x(96)00605-1 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote351599 AcademicArticle Applications of free radicals in organic synthesis 1997 http://vivo.scripps.edu/individual/endnote235588
http://vivo.scripps.edu/individual/endnote57934 AcademicArticle Determination of the relative and absolute stereochemistry of fostriecin (CL-920) 1997 10.1021/jo962166h http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote343313 AcademicArticle CC-1065/duocarmycin and bleomycin A(2) hybrid agents: lack of enhancement of DNA alkylation by attachment to noncomplementary DNA binding subunits 1997 10.1016/s0968-0896(96)00237-4 9061188 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote267204 AcademicArticle Preparation and inverse electron demand diels-alder reactions of 3-methoxy-6-methylthio-1,2,4,5-tetrazine 1997 10.1016/s0040-4039(97)00751-x http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote46694 AcademicArticle Solution-phase combinatorial synthesis via the olefin metathesis reaction 1997 10.1016/s0960-894x(97)00043-7 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote17378 AcademicArticle 10-formyl-5,8,10-trideazafolic acid (10-formyl-TDAF): a potent inhibitor of glycinamide ribonucleotide transformylase 1997 10.1016/s0968-0896(97)00120-x 9354237 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote168316 AcademicArticle Multisubstrate analogue based on 5,8,10-trideazafolate 1997 10.1016/s0968-0896(97)00124-7 9354241 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote266407 AcademicArticle Synthesis and evaluation of CC-1065 and duocarmycin analogues incorporating the iso-CI and iso-CBI alkylation subunits: impact of relocation of the C-4 carbonyl 1997 10.1021/jo971686p http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote72606 AcademicArticle Synthesis of (9R,12S)- and (9S,12S)-cycloisodityrosine and their N-methyl derivatives 1997 10.1021/jo961346o 11671510 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote228294 AcademicArticle Abenzyl 10-formyl-trideazafolic acid (abenzyl 10-formyl-TDAF): an effective inhibitor of glycinamide ribonucleotide transformylase 1997 10.1016/s0968-0896(97)00123-5 9354240 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote170972 AcademicArticle Catalysis of the CC-1065 and duocarmycin DNA alkylation reaction: DNA binding induced conformational change in the agent results in activation 1997 10.1016/s0968-0896(96)00238-6 9061191 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote347473 AcademicArticle Synthesis of the vancomycin CD and DE ring systems 1997 10.1021/jo970560p http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote396213 AcademicArticle An exceptionally potent analog of sandramycin 1997 10.1016/s0960-894x(97)00129-7 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote265865 AcademicArticle N-methyl threonine analogues of deglycobleomycin A(2): Synthesis and evaluation 1997 10.1016/s0968-0896(97)00107-7 9313863 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote122835 AcademicArticle Duocarmycin SA shortened, simplified, and extended agents: A systematic examination of the role of the DNA binding subunit 1997 10.1021/ja9637208 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote322661 AcademicArticle CC-1065 and the duocarmycins: Synthetic studies 1997 10.1021/cr960095g 11848889 http://vivo.scripps.edu/individual/endnote51983
http://vivo.scripps.edu/individual/endnote129480 AcademicArticle Functionalized analogues of 5,8,10-trideazafolate: Development of an enzyme-assembled tight binding inhibitor of GAR Tfase and a potential irreversible inhibitor of AICAR Tfase 1997 10.1016/s0968-0896(97)00122-3 9354239 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote22856 AcademicArticle High resolution solution structure of a DNA duplex alkylated by the antitumor agent duocarmycin SA 1997 10.1006/jmbi.1997.1223 9299351 http://vivo.scripps.edu/individual/endnote261742
http://vivo.scripps.edu/individual/endnote395585 AcademicArticle Functionalized analogues of 5,8,10-trideazafolate as potential inhibitors of gar tfase or aicar tfase 1997 10.1016/s0968-0896(97)00121-1 9354238 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote270306 AcademicArticle The sleep-inducing lipid oleamide deconvolutes gap junction communication and calcium wave transmission in glial cells 1997 10.1083/jcb.139.7.1785 9412472 http://vivo.scripps.edu/individual/endnote322298
http://vivo.scripps.edu/individual/endnote52885 AcademicArticle Synthesis and evaluation of CC-1065 and duocarmycin analogs incorporating the 1,2,3,4,11,11a-hexahydrocyclopropa c naphtho 2,1-b azepin-6-one (CNA) alkylation subunit: Structural features that govern reactivity and reaction regioselectivity 1997 10.1021/jo9707085 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote180172 AcademicArticle Thermal atropisomerism of fully functionalized vancomycin CD, DE, and CDE ring systems 1997 10.1016/s0960-894x(97)10182-2 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote122948 AcademicArticle Asymmetric synthesis of the CBI alkylation subunit of the CC-1065 and duocarmycin analogs 1997 http://vivo.scripps.edu/individual/endnote302592
http://vivo.scripps.edu/individual/endnote183242 AcademicArticle Reversed and sandwiched analogs of duocarmycin SA: Establishment of the origin of the sequence-selective alkylation of DNA and new insights into the source of catalysis 1997 10.1021/ja9637210 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote203700 AcademicArticle Generation of targeted C-2-symmetrical compound libraries by solution-phase combinatorial chemistry 1997 10.1016/s0960-894x(97)00330-2 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e2n232667 AcademicArticle Editorial 1996 10.1016/s0960-894x(96)90241-3 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e7n301280 AcademicArticle Cycloaddition reactions of azadienes, cyclopropenone ketals, and related systems: scope and applications 1996 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/e7n121566 AcademicArticle Alternative synthesis of the cycloisodityrosine subunit of deoxybouvardin, RA-VII, and related agents: reassignment of the stereochemistry of prior intermediates 1996 10.1021/jo9604144 11667262 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n289723 AcademicArticle Control of chemoselectivity in catalytic rhodium carbenoid reactions through ligand modification. Comments 1996 http://vivo.scripps.edu/individual/e7n180816
http://vivo.scripps.edu/individual/endnote220512 AcademicArticle A comparative study of the solvolysis reactivity, regioselectivity, and stereochemistry of the duocarmycin A and SA alkylation subunits 1996 10.1016/0960-894x(96)00346-0 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote339406 AcademicArticle Synthesis, chemical properties, and preliminary evaluation of substituted CBI analogs of CC-1065 and the duocarmycins incorporating the 7-cyano-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one alkylation subunit: Hammett quantitation of the magnitude of electronic effects on functional reactivity 1996 10.1021/jo9605298 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote117425 AcademicArticle Molecular characterization of an enzyme that degrades neuromodulatory fatty-acid amides 1996 10.1038/384083a0 8900284 http://vivo.scripps.edu/individual/endnote351395
http://vivo.scripps.edu/individual/endnote360112 AcademicArticle Structure determination of an endogenous sleep-inducing lipid, cis-9-octadecenamide (oleamide): A synthetic approach to the chemical analysis of trace quantities of a natural product 1996 10.1021/ja9532345 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote187755 AcademicArticle Demonstration and definition of the noncovalent binding selectivity of agents related to CC-1065 by an affinity cleavage agent: Noncovalent binding coincidental with alkylation 1996 10.1016/0968-0896(96)00073-9 8818235 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote182195 AcademicArticle Examination of the role of the duocarmycin SA methoxy substituents: Identification of the minimum, fully potent DNA binding subunit 1996 10.1016/0960-894x(96)00401-5 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote19802 AcademicArticle Inhibition of oleamide hydrolase catalyzed hydrolysis of the endogenous sleep-inducing lipid cis-9-octadecenamide 1996 10.1021/ja954064z http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote26390 AcademicArticle CC-1065 and the duocarmycins: understanding their biological function through mechanistic studies 1996 10.1002/anie.199614381 http://vivo.scripps.edu/individual/endnote319084
http://vivo.scripps.edu/individual/endnote63617 AcademicArticle Synthesis of (9S,12S)-cycloisodityrosine and its unnatural (9R,12S)-diastereomer 1996 10.1016/0960-894x(96)00179-5 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote30964 AcademicArticle (-)-Sandramycin: total synthesis and characterization of DNA binding properties 1996 10.1021/ja952799y http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote238056 AcademicArticle Novel solution phase strategy for the synthesis of chemical libraries containing small organic molecules 1996 10.1021/ja9530681 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote137025 AcademicArticle Key analogues of the tetrapeptide subunit of RA-VII and deoxybouvardin 1996 10.1016/0968-0896(96)00151-4 8931929 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote172529 AcademicArticle Synthesis and evaluation of deglycobleomycin A(2) analogues containing a tertiary N-methyl amide and simple ester replacement for the L-histidine secondary amide: Direct functional characterization of the requirement for secondary amide metal complexation 1996 10.1016/0968-0896(95)00183-2 8814877 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote18327 AcademicArticle Synthesis and evaluation of potential N-pi and N-sigma metal chelation sites within the beta-hydroxy-L-histidine subunit of bleomycin A(2): Functional characterization of imidazole N-pi metal complexation 1996 10.1016/0968-0896(95)00184-0 8814878 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote394540 AcademicArticle A solution-phase strategy for the synthesis of chemical libraries containing small organic molecules: a universal and dipeptide mimetic template 1996 10.1016/0968-0896(96)00069-7 8804539 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote289638 AcademicArticle Synthesis, X-ray structure, and properties of fluorocyclopropane analogs of the duocarmycins incorporating the 9,9-difluoro-1,2,9,9a-tetrahydrocyclopropa c benzo e indol-4-one (F2CBI) alkylation subunit 1996 10.1021/ja961888n http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote29742 AcademicArticle Azadiene Diels-Alder reactions: scope and applications. Total synthesis of natural and ent-fredericamycin A 1996 10.1002/jhet.5570330508 http://vivo.scripps.edu/individual/endnote355769
http://vivo.scripps.edu/individual/endnote307756 AcademicArticle Synthesis of (r)-(4-methoxy-3,5-dihydroxyphenyl)glycine derivatives: The central amino acid of vancomycin and related agents 1996 10.1021/jo960085f http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote267683 AcademicArticle Enantioselective total synthesis of (+)-duocarmycin A, epi-(+)-duocarmycin a, and their unnatural enantiomers 1996 10.1021/ja953777e http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote202999 AcademicArticle Generalized dipeptidomimetic template: solution phase parallel synthesis of combinatorial libraries 1996 10.1021/ja9539711 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote82719 AcademicArticle Synthesis and properties of substituted CBI analogs of CC-1065 and the duocarmycins incorporating the 7-methoxy-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (MCBI) alkylation subunit: magnitude of electronic effects on the functional reactivity 1996 10.1021/jo952033g 11667041 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote149972 AcademicArticle A Hammett correlation for CC-1065 and duocarmycin analogs: magnitude of substituent electronic effects on functional reactivity 1996 10.1016/0960-894x(96)00093-5 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e7n179688 AcademicArticle Total synthesis of (+)- and ent-(-)-duocarmycin SA 1995 http://vivo.scripps.edu/individual/e7n257080
http://vivo.scripps.edu/individual/endnote180960 AcademicArticle A modified friedlander condensation for the synthesis of 3-hydroxyquinoline-2-carboxylates 1995 10.1021/jo00127a055 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote322928 AcademicArticle CC-1065 CBI analogs - an example of enhancement of DNA alkylation efficiency through introduction of stabilizing electrostatic interactions 1995 10.1016/0968-0896(95)00048-l 7582940 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote329599 AcademicArticle Diastereoselective dieckmann condensation suitable for introduction of the duocarmycin A C6 center - development of a divergent strategy for the total synthesis of duocarmycins A and SA 1995 10.1016/0968-0896(94)00147-u 8612048 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote183158 AcademicArticle An unusually facile SNAr 14-membered biaryl ether macrocyclization reaction suitable for preparation of the cycloisodityrosine subunit of bouvardin, deoxybouvardin and related agents 1995 10.1016/0960-894x(95)00192-v http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote343252 AcademicArticle Chemical characterization of a family of brain lipids that induce sleep 1995 10.1126/science.7770779 7770779 http://vivo.scripps.edu/individual/endnote276633
http://vivo.scripps.edu/individual/endnote132861 AcademicArticle Key synthetic analogs of bleomycin A(2) that directly address the effect and role of the disaccharide - demannosylbleomycin A(2) and alpha-D-mannopyranosyldeglycobleomycin A(2) 1995 10.1021/ja00133a008 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote142239 AcademicArticle Key analogs of the tetrapeptide subunit of RA-VII and deoxybouvardin 1995 10.1016/0968-0896(95)00141-7 8770383 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote367504 AcademicArticle CBI-CDPBO1 and CBI-CDPBI1 - CC-1065 analogs containing deep-seated modifications in the DNA-binding subunit 1995 10.1016/0968-0896(95)00066-p 7582954 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote245376 AcademicArticle Second definitive test of proposed models for the origin of the CC-1065 and duocarmycin DNA alkylation selectivity 1995 10.1021/ja00109a035 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote121527 AcademicArticle An efficient synthesis of 1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (CBI) - an enhanced and simplified analog of the CC-1065 and duocarmycin alkylation subunits 1995 10.1021/jo00110a034 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote247922 AcademicArticle DNA alkylation properties of CC-1065 and duocarmycin analogs incorporating the 2,3,10,10a-tetrahydrocyclopropa d benzo f quinol-5-one alkylation subunit - identification of subtle structural features that contribute to the regioselectivity of the adenine N3 alkylation reaction 1995 10.1021/ja00152a004 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote211094 AcademicArticle Synthesis and evaluation of the fully functionalized bleomycin A(2) metal-binding domain-containing the 2-O-(3-O-carbamoyl-alpha-D-mannopyranosyl)-alpha-L-gulopyranosyl disaccharide 1995 10.1021/ja00133a007 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote347005 AcademicArticle Total synthesis of natural and ent-fredericamycin-a 1995 10.1021/ja00153a004 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote353147 AcademicArticle 1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one (CBI) analogs of CC-1065 and the duocarmycins: synthesis and evaluation 1995 10.1016/0968-0896(95)00130-9 8634824 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote42726 AcademicArticle CC-1065 and the duocarmycins - unraveling the keys to a new class of naturally derived DNA alkylating-agents 1995 10.1073/pnas.92.9.3642 7731958 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote3861 AcademicArticle Synthesis of key analogs of bleomycin A(2) that permit a systematic evaluation of the linker region - identification of an exceptionally prominent role for the L-threonine substituent 1995 10.1016/0968-0896(95)00113-u 8564421 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote374345 AcademicArticle N-desmethyl derivatives of deoxybouvardin and RA-VII: synthesis and evaluation 1995 10.1021/ja00133a010 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote54399 AcademicArticle The duocarmycins: synthetic and mechanistic studies 1995 10.1021/ar00049a004 http://vivo.scripps.edu/individual/endnote122847
http://vivo.scripps.edu/individual/endnote395760 AcademicArticle Solution-phase conformational studies of the cyclic peptide RA-VII: lithium-chloride perturbation of the conformational equilibria 1995 10.1021/ja00133a009 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote239998 AcademicArticle Total synthesis of granditropone, grandirubrine, imerubrine, and isoimerubrine 1995 10.1021/ja00155a009 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote114077 AcademicArticle Synthesis of appropriately functionalized vancomycin CD and DE ring systems 1995 10.1016/0960-894x(95)00543-9 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/e7n266715 AcademicArticle Design, synthesis and evaluation of bouvardin, deoxybouvardin and RA-I-XIV pharmacophore analogs 1994 10.1016/s0968-0896(00)82005-2 7922127 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/e7n387665 AcademicArticle Control of chemoselectivity in catalytic rhodium carbenoid reactions through ligand modification 1994 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/e7n364678 AcademicArticle Molecular basis for sequence selective DNA alkylation by (+)- and ent-(-)-CC-1065 and related agents: alkylation site models that accommodate the offset AT-rich adenine N3 alkylation selectivity 1994 10.1016/S0968-0896(00)82007-6 7922122 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote264892 AcademicArticle Cerebrodiene: A brain lipid isolated from sleep-deprived cats 1994 10.1073/pnas.91.20.9505 7937797 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote233050 AcademicArticle Total synthesis of bleomycin A(2) and related agents .4. Synthesis of the disaccharide subunit - 2-O-(3-O-carbamoyl-alpha-D-mannopyranosyl)-L-gulopyranose and completion of the total synthesis of bleomycin a(2) 1994 10.1021/ja00092a014 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote216390 AcademicArticle P-quinonemethide analog of the CC-1065 and duocarmycin alkylation subunits 1994 10.1021/jo00096a043 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote319634 AcademicArticle Diels-Alder reactions of cyclopropenone ketals - a concise tropolone annulation applicable to rubrolone-C ring introduction 1994 10.1021/jo00091a040 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote16486 AcademicArticle Total synthesis and biological properties of novel antineoplastic (chloromethyl)furanoindolines - an asymmetric hydroboration mediated synthesis of the alkylation subunits 1994 10.1021/jm00028a005 8295210 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote144893 AcademicArticle Design, synthesis, and evaluation of DNA minor-groove binding-agents - the duocarmycins 1994 10.1351/pac199466040837 http://vivo.scripps.edu/individual/endnote313708
http://vivo.scripps.edu/individual/endnote287904 AcademicArticle Chemical and structural comparison of N-BOC-CBQ and N-BOC-CBI - identification and structural origin of an unappreciated but productive stability of the CC-1065 and duocarmycin SA alkylation subunits 1994 10.1021/ja00093a067 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote167157 AcademicArticle (+)- and ent-(-)-duocarmycin SA and (+)- and ent-(-)-N-BOC-DSA DNA alkylation properties - alkylation site models that accommodate the offset AT-rich adenine N3 alkylation selectivity of the enantiomeric agents 1994 10.1021/ja00084a004 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote289851 AcademicArticle CBI-TMI - synthesis and evaluation of a key analog of the duocarmycins - validation of a direct relationship between chemical solvolytic stability and cytotoxic potency and confirmation of the structural features responsible for the distinguishing behavior of enantiomeric pairs of agents 1994 10.1021/ja00097a006 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote102790 AcademicArticle Crossing extreme mechanistic barriers by antibody catalysis: Syn elimination to a cis olefin 1994 10.1021/ja00092a080 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote30738 AcademicArticle Role of the CC-1065 and duocarmycin N-2 substituent - validation of a direct relationship between solvolysis chemical-stability and in-vitro biological potency 1994 10.1021/ja00091a088 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote237484 AcademicArticle Total synthesis of bouvardin, O-methylbouvardin, and O-methyl-N-9-desmethylbouvardin 1994 10.1021/ja00098a015 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote380868 AcademicArticle Design, synthesis, and evaluation of CC-1065 and duocarmycin analogs incorporating the 2,3,10,10a-tetrahydro-1H-cyclopropa d benzo f quinol-5-one (CBQ) alkylation subunit - identification and structural origin of subtle stereoelectronic features that govern reactivity and regioselectivity 1994 10.1021/ja00104a013 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote242802 AcademicArticle Total synthesis of bleomycin-A(2) and related agents .1. Synthesis and DNA-binding properties of the extended C-terminus - tripeptide-S, tetrapeptide-S, pentapeptide-S, and related agents 1994 10.1021/ja00092a011 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote118365 AcademicArticle Total syntheses of (+)-p-3a, epi-(-)-p-3a, and (-)-desacetamido p-3a 1994 10.1021/ja00080a010 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote45569 AcademicArticle Synthesis of a functionalized rigid bicyclo[2.2.1]heptane: a useful hapten for eliciting catalytic antibodies 1994 10.1021/jo00096a064 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote66318 AcademicArticle Induction of endonucleolytic DNA fragmentation and apoptosis by the duocarmycins 1994 10.1016/s0960-894x(01)80168-2 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote115977 AcademicArticle Inverse electron demand Diels-Alder reactions of heterocyclic azadienes - 4+2 -cycloaddition reaction of amidines with 1,3,5-triazines 1994 10.1021/jo00096a044 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote41313 AcademicArticle Total synthesis of bleomycin-A(2) and related agents .2. Synthesis of (-)-pyrimidoblamic acid, epi-(+)-pyrimidoblamic acid, (+)-desacetamidopyrimidoblamic acid, and (-)-descarboxamidopyrimidoblamic acid 1994 10.1021/ja00092a012 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote273598 AcademicArticle Total synthesis of bleomycin-A(2) and related agents .3. Synthesis and comparative-evaluation of deglycobleomycin-A(2), epideglycobleomycin-A(2), deglycobleomycin-A(1), and desacetamidodeglycobleomycin, descarboxamidodeglycobleomycin, desmethyldeglycobleomycin, and desimidazolyldeglycobleomycin-A(2) 1994 10.1021/ja00092a013 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e7n378082 AcademicArticle Evaluation of functional analogs of CC-1065 and the duocarmycins incorporating the cross-linking 9a-chloromethyl-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-on e (C2BI) alkylation subunit 1993 10.1016/S0968-0896(00)82100-8 8081835 http://vivo.scripps.edu/individual/endnote193708
http://vivo.scripps.edu/individual/endnote188912 AcademicArticle Vancomycin and ristocetin models - synthesis via the Ullmann macrocyclization reaction 1993 10.1021/jo00058a024 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote53013 AcademicArticle 4pi participation of 1-aza-1,3-butadienes in [4 + 2] cycloaddition reactions: intramolecular Diels-Alder reactions of alpha,beta-unsaturated N-sulfonylimines 1993 10.1021/jo00060a022 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote260958 AcademicArticle Design, synthesis, and evaluation of DNA minor-groove binding-agents 1993 10.1351/pac199365061123 http://vivo.scripps.edu/individual/endnote313708
http://vivo.scripps.edu/individual/endnote366526 AcademicArticle Singlet oxygen oxidation of bipyrroles - total synthesis of d,l-isochrysohermidin and meso-isochrysohermidin 1993 10.1021/ja00071a069 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote72459 AcademicArticle (-)-sandramycin - total synthesis and preliminary DNA-binding properties 1993 10.1021/ja00077a082 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote66520 AcademicArticle CDPI3-enediyne and CDPI3-EDTA conjugates - a new class of DNA cleaving agents 1993 10.1021/jo00063a019 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote345558 AcademicArticle Studies on the synthesis of bleomycin-A(2) - observations on a diastereoselective imine addition-reaction for C2-acetamido side-chain introduction 1993 10.1016/0040-4039(93)85008-k http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote266906 AcademicArticle D, l- and meso-isochrysohermidin - total synthesis and interstrand DNA cross-linking 1993 10.1021/ja00077a046 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote9911 AcademicArticle Total synthesis of streptonigrone 1993 10.1021/ja00076a035 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote115780 AcademicArticle Total synthesis of (-)-pyrimidoblamic acid and deglycobleomycin A2 1993 10.1002/anie.199302731 http://vivo.scripps.edu/individual/endnote319084
http://vivo.scripps.edu/individual/endnote397602 AcademicArticle Total synthesis and preliminary evaluation of (+)-duocarmycin and ent-(-)-duocarmycin SA 1993 10.1021/ja00073a019 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote282808 AcademicArticle Reversibility of the duocarmycin-A and SA DNA alkylation reaction 1993 10.1021/ja00074a093 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote293730 AcademicArticle K-13 and OF4949 - evaluation of key partial structures and pharmacophore delineation 1993 10.1016/s0960-894x(01)80885-4 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote222276 AcademicArticle Total synthesis of cycloisodityrosine, RA-VII, deoxybouvardin, and N29-desmethyl-RA-VII - identification of the pharmacophore and reversal of the subunit functional roles 1993 10.1021/ja00062a004 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote42248 AcademicArticle Total synthesis of (+)-piperazinomycin 1993 10.1021/ja00077a047 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e7n385159 AcademicArticle Preparation and Diels-Alder reaction of a reactive, electron-deficient heterocyclic azadiene: dimethyl 1,2,4,5-tetrazine-3,6-dicarboxylate. 1,2-Diazine and pyrrole introduction 1992 http://vivo.scripps.edu/individual/endnote12246
http://vivo.scripps.edu/individual/e7n334975 AcademicArticle Total synthesis of (+)-duocarmycin SA 1992 10.1021/ja00051a045 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e7n71158 AcademicArticle Synthesis of N29-desmethyl RA-VII. Identification of the pharmacophore of RA-I-VII and deoxybouvardin and reassignment of the subunit functional roles 1992 10.1021/jo00031a001 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n326895 AcademicArticle Synthesis of tri- and tetrapeptide S: the extended C-terminus of bleomycin A2 1992 10.1021/jo00042a003 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n284662 AcademicArticle Synthesis of desacetamidopyrimidoblamic acid and deglyco desacetamidobleomycin A2 1992 10.1021/jo00042a004 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n373535 AcademicArticle Design, synthesis, and evaluation of functional analogs of CC-1065 and the duocarmycins: a study of structural features effecting DNA binding selectivity 1992 http://vivo.scripps.edu/individual/e7n385337
http://vivo.scripps.edu/individual/e7n187986 AcademicArticle Synthesis of desacetamido P-3A: 1,3,5-triazine .fwdarw. pyrimidine heteroaromatic azadiene Diels-Alder reaction 1992 10.1021/jo00032a001 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote29754 AcademicArticle DNA alkylation properties of enhanced functional analogs of cc-1065 incorporating the 1,2,9,9a-tetrahydrocyclopropa 1,2-c benz 1,2-e indol-4-one (cbi) alkylation subunit 1992 10.1021/ja00040a001 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote386103 AcademicArticle P-3A and (-)-desacetamido P-3A - demonstration and study of their effective functional cleavage of duplex DNA 1992 10.1016/s0960-894x(00)80449-7 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote132393 AcademicArticle Acyl radicals - intermolecular and intramolecular alkene addition-reactions 1992 10.1021/jo00031a021 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote198417 AcademicArticle A convenient and general preparation of n-sulfonylimines 1992 10.1021/jo00043a047 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote267978 AcademicArticle Deglyco GABA,gly-desacetamidobleomycin-A2 - a simplified synthetic model for bleomycin-A2 1992 10.1016/s0960-894x(01)81076-3 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote107076 AcademicArticle A concise synthesis of the fredericamycin-a DEF ring-system - 4+2 cycloaddition reactions of 1-aza-1,3-butadienes 1992 10.1021/jo00040a044 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote566 AcademicArticle Functional analogs of CC-1065 and the duocarmycins incorporating the 9A-(chloromethyl)-1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (C2BI) alkylation subunit - synthesis and preliminary DNA alkylation studies 1992 10.1021/ja00050a012 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote160953 AcademicArticle An improved synthesis of 1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (CBI) - a simplified analog of the CC-1065 alkylation subunit 1992 10.1021/jo00036a023 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote311521 AcademicArticle A simple method for the purification and isolation of bleomycin-A2 1992 10.1016/s0960-894x(00)80597-1 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote185465 AcademicArticle DNA alkylation properties of enhanced functional analogs of CC-1065 incorporating the 1,2,9,9a-tetrahydrocyclopropa[1,2-c]benz[1,2-e]indol-4-one (CBI) alkylation subunit 1992 10.1016/s0960-894x(00)80407-2 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote113320 AcademicArticle Synthesis of the lower subunit of rhizoxin 1992 10.1021/jo00034a010 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote192783 AcademicArticle CC-1065 partial structures - enhancement of noncovalent affinity for DNA minor groove binding through introduction of stabilizing electrostatic interactions 1992 10.1021/jo00030a042 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n393042 AcademicArticle Total synthesis of calicheamicinone: a solution to the problem of the elusive urethane 1991 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/e7n251533 AcademicArticle Recent advances in bioorganic chemistry. Preface 1991 10.1016/s0040-4020(01)81771-3 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/e7n81503 AcademicArticle Solution structure of FKBP, a rotamase enzyme and receptor for FK506 and rapamycin. Atomic structure of FKBP-FK506, an immunophilin-immunosuppressant complex 1991 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/e7n109651 AcademicArticle Duocarmycins: a new class of sequence selective DNA minor groove alkylating agents 1991 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/endnote344314 AcademicArticle Singlet oxygen mediated oxidative decarboxylation of pyrrole-2-carboxylic acids 1991 10.1021/jo00024a045 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote270484 AcademicArticle Inverse electron demand Diels-Alder reactions of N-sulfonyl alpha,beta-unsaturated imines - a general-approach to implementation of the 4-pi participation of 1-aza-1,3-butadienes in Diels-Alder reactions 1991 10.1021/ja00005a040 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote158004 AcademicArticle Design and synthesis of a conformational analog of deoxybouvardin 1991 10.1021/jo00018a035 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote319162 AcademicArticle Intramolecular Ullmann condensation reaction - an effective approach to macrocyclic diaryl ethers 1991 10.1021/jo00005a020 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote41555 AcademicArticle Isolation and characterization of the duocarmycin adenine DNA adduct 1991 10.1021/ja00017a042 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote83430 AcademicArticle A potent, simple derivative of an analog of the CC-1065 alkylation subunit 1991 10.1016/s0960-894x(01)81090-8 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote101550 AcademicArticle Diels-Alder reactions of N-sulfonyl-1-aza-1,3-butadienes: Development of a synthetic approach to the streptonigrone C ring 1991 10.1021/jo00002a077 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote388201 AcademicArticle Evaluation of bouvardin, deoxybouvardin, and RA-I - RA-VII partial structures - reassignment of the pharmacophore 1991 10.1016/s0960-894x(01)80815-5 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote196335 AcademicArticle Demonstration of a pronounced effect of noncovalent binding selectivity on the (+)-CC-1065 DNA alkylation and identification of the pharmacophore of the alkylation subunit 1991 10.1073/pnas.88.4.1431 1847523 http://vivo.scripps.edu/individual/endnote71945
http://vivo.scripps.edu/individual/endnote213657 AcademicArticle Total synthesis of (+/-)-cis-trikentrin-A and (+/-)-trans-trikentrin-A - Diels-Alder reactions of heteroaromatic azadienes 1991 10.1021/ja00011a026 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote126154 AcademicArticle (+)-CC-1065 DNA alkylation - observation of an unexpected relationship between cyclopropane electrophile reactivity and the intensity of DNA alkylation 1991 10.1021/ja00007a077 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote141476 AcademicArticle Total synthesis of deoxybouvardin and RA-VII - macrocyclization via an intramolecular Ullmann reaction 1991 10.1021/ja00004a062 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote140285 AcademicArticle Synthesis and preliminary evaluation of the fredericamycin-A ABCDE ring-system 1991 10.1021/jo00006a029 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote60386 AcademicArticle Total synthesis of combretastatin D-2 - intramolecular ullmann macrocyclization reaction 1991 10.1021/jo00013a024 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote137621 AcademicArticle (+)-CC-1065 DNA alkylation - key studies demonstrating a noncovalent binding selectivity contribution to the alkylation selectivity 1991 10.1021/ja00010a046 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote398001 AcademicArticle Synthesis and preliminary evaluation of (+)-CBI-indole2 - an enhanced functional analog of (+)-CC-1065 1991 10.1016/s0960-894x(00)80243-7 http://vivo.scripps.edu/individual/endnote119710
http://vivo.scripps.edu/individual/endnote312063 AcademicArticle Studies on the synthesis of rubrolone: 4π participation of O-alkyl α,β-unsaturated oximes in intramolecular [4 + 2] cycloaddition reactions 1991 10.1016/0040-4039(91)80554-j http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote46782 AcademicArticle An alternative and convenient strategy for generation of substantial quantities of singly 5-32P-end-labeled double-stranded DNA for binding-studies - development of a protocol for examination of functional features of (+)-CC-1065 and the duocarmycins that contribute to their sequence-selective DNA alkylation properties 1991 10.1016/s0040-4020(01)81798-1 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/e2n15447 AcademicArticle Tandem free-radical ring expansion and 5-exo-dig 5-hexynyl radical cyclization: a useful approach to fused bicyclic carbocycles 1990 10.1021/jo00307a010 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n237859 AcademicArticle Use of methylenecyclopropanone ketals for cyclopentane synthesis. A new efficient thermal [3 + 2] cycloaddition 1990 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/e7n51727 AcademicArticle Polyethylene-bound soluble recoverable palladium(0) catalysts 1990 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/e7n124651 AcademicArticle Photolytic reactions of chromium aminocarbene complexes. Conversion of amides to α-amino acids 1990 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/e7n209698 AcademicArticle Room-temperature, endo-specific 1-aza-1,3-butadiene Diels-Alder reactions: acceleration of the LUMOdiene-controlled [4 + 2] cycloaddition reactions through noncomplementary aza diene substitution 1990 10.1021/jo00297a006 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n108806 AcademicArticle Synthesis and preliminary evaluation of agents incorporating the pharmacophore of the duocarmycin/pyrindamycin alkylation subunit: identification of the CC-1065/duocarmycin common pharmacophore 1990 10.1021/jo00302a002 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n262907 AcademicArticle The absolute configuration and synthesis of natural (-)-dolastatin 10 1990 http://vivo.scripps.edu/individual/e7n47566
http://vivo.scripps.edu/individual/e7n280569 AcademicArticle Diels-Alder reactions of 1-aza-1,3-butadienes: room temperature, endo-selective LUMOdiene-controlled [4 + 2] cycloaddition reactions of N-sulfonyl-4-(ethoxycarbonyl)-1-aza-1,3-butadienes 1990 10.1021/jo00307a009 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote266256 AcademicArticle Synthesis of N-(tert-butyloxycarbonyl)-CBI, CBI, CBI-CBI1, and CBI-CDPI2 - enhanced functional analogs of CC-1065 incorporating the 1,2,9,9a-tetrahydrocyclopropa c benz e indol-4-one (CBI) left-hand subunit 1990 10.1021/jo00310a013 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote310433 AcademicArticle Regiocontrolled nucleophilic-addition to selectively activated para-quinone diimines - alternative preparation of a key intermediate employed in the preparation of the CC-1065 left-hand subunit 1990 10.1021/jo00291a059 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote174449 AcademicArticle Synthesis and evaluation of aborted and extended CC-1065 functional analogs - (+)-CPI-PDE-1, and (-)-CPI-PDE-1, (+)-CPI-PDE-1, and (-)-CPI-CDPI1, and (+/-)-CPI-PDE-i1, (+)-CPI-PDE-i1, and (-)-CPI-CDPI3 - preparation of key partial structures and definition of an additional functional-role of the CC-1065 central and right-hand subunits 1990 10.1021/ja00168a002 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote78406 AcademicArticle Tandem free-radical alkene addition-reactions of acyl radicals 1990 10.1021/ja00166a043 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote279273 AcademicArticle Synthesis and preliminary evaluation of agents incorporating the pharmacophore of the duocarmycin pyrindamycin alkylation subunit - identification of the cc-1065 duocarmycin common pharmacophore 1990 10.1021/jo00302a002 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote47805 AcademicArticle Duocarmycin pyrindamycin DNA alkylation properties and identification, synthesis, and evaluation of agents incorporating the pharmacophore of the duocarmycin pyrindamycin alkylation subunit - identification of the CC-1065-duocarmycin common pharmacophore 1990 10.1021/ja00180a048 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote322347 AcademicArticle Design and total synthesis of a conformational analog of bouvardin deoxybouvardin 1990 http://vivo.scripps.edu/individual/endnote302592
http://vivo.scripps.edu/individual/endnote62204 AcademicArticle Resolution of a CBI precursor and incorporation into the synthesis of (+)-CBI, (+)-CBI-CDPI1, (+)-CBI-CDPI2 - enhanced functional analogs of (+)-CC-1065 - a critical-appraisal of a proposed relationship between electrophile reactivity, DNA-binding properties, and cytotoxic potency 1990 10.1016/s0040-4039(00)94629-x http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote149493 AcademicArticle Intramolecular acyl radical alkene addition-reactions - macrocyclization reactions 1990 10.1021/ja00166a044 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote13515 AcademicArticle Diels-Alder reactions of azadienes: scope and applications 1990 10.1002/bscb.19900990902 http://vivo.scripps.edu/individual/endnote204561
http://vivo.scripps.edu/individual/endnote235650 AcademicArticle Studies of the total synthesis of fredericamycin-A - preparation of key partial structures and development of an intermolecular alkyne chromium carbene complex benzannulation cyclization approach to the ABCD(E) ring-system 1990 10.1021/jo00293a043 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote84827 AcademicArticle Total synthesis of L,L-isodityrosine and isodityrosine-derived agents - K-13, OF4949-III, and OF4949-IV 1990 10.1021/jo00311a019 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote186396 AcademicArticle A demonstration of the intrinsic importance of stabilizing hydrophobic binding and noncovalent van der Waals contacts dominant in the noncovalent CC-1065/b-DNA binding 1990 10.1016/0009-2797(90)90107-x 2406033 http://vivo.scripps.edu/individual/endnote187913
http://vivo.scripps.edu/individual/endnote354821 AcademicArticle Synthesis of n-(phenylsulfonyl)-CI, N-((tert-butyloxy)carbonyl)-CI, CI-CDPI1, and CI-CDPI2 - CC-1065 functional analogs incorporating the parent 1,2,7,7a-tetrahydrocycloprop 1,2-c indol-4-one (CI) left-hand subunit 1990 10.1021/ja00169a034 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e2n323346 AcademicArticle Total synthesis of (.+-.)-N-(phenylsulfonyl)- and (.+-.)-N-(tert-butyloxycarbonyl)-CI, (.+-.)-CI-CDPI1, and (.+-.)-CI-CDPI2: CC-1065 functional analogs incorporating the parent 1,2,7,7a-tetrahydrocycloprop[1,2-c]indol-4-one (CI) left-hand subunit 1989 10.1021/jo00267a004 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n296998 AcademicArticle Total synthesis of K-13 1989 10.1021/jo00272a003 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n270787 AcademicArticle Diels-Alder reactions of heterocyclic azadienes: development of a strategy for the total synthesis of streptonigrin, lavendamycin, and synthetic quinoline-5,8-quinones 1989 10.1016/B978-0-08-092429-8.50006-4 http://vivo.scripps.edu/individual/e7n271124
http://vivo.scripps.edu/individual/e7n69344 AcademicArticle Phenylselenoesters as effective precursors of acyl radicals for use in intermolecular alkene addition reactions 1989 10.1021/jo00269a001 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n252223 AcademicArticle Recent applications of the inverse electron demand Diels-Alder reaction 1989 http://vivo.scripps.edu/individual/e7n163765
http://vivo.scripps.edu/individual/endnote1433 AcademicArticle A general-solution to implementing the 4-p participation of 1-aza-1,3-butadienes in Diels-Alder reactions - inverse electron demand Diels-Alder reactions of alpha,beta-unsaturated n-benzenesulfonyl imines 1989 10.1021/ja00186a067 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote173129 AcademicArticle Studies on the total synthesis of fredericamycin-a - development of an intermolecular alkyne-chromium carbene complex cyclization approach to the abcde ring-system 1989 10.1016/s0040-4039(01)93705-0 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote345129 AcademicArticle Synthesis of isodityrosine 1989 10.1016/s0040-4039(01)93709-8 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote43046 AcademicArticle Total synthesis of OF4949-III and OF4949-IV - unusual effects of remote substituents on the rate of macrocyclization reactions 1989 10.1016/s0040-4039(01)93447-1 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote80846 AcademicArticle A study of the scope of the 4+2 cyclo-addition reactions of unactivated 1,3-oxazin-6-ones 1989 10.1021/jo00264a041 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote21719 AcademicArticle Total synthesis and evaluation of (+/-)-N-(tert-butyloxycarbonyl)-CBI, (+/-)-CBI-CDPI1, and (+/-)-CBI-CDPI2 - CC-1065 functional agents incorporating the equivalent 1,2,9,9a-tetrahydrocycloprop 1,2-c benz 1,2-e indol-4-one (CBI) left-hand subunit 1989 10.1021/ja00198a089 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e7n140777 AcademicArticle A divergent de novo synthesis of carbohydrates based on an accelerated inverse electron demand Diels-Alder reaction of 1-oxa-1,3-butadienes 1988 10.1021/jo00259a040 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n148045 AcademicArticle Preparation and inverse-​electron-​demand Diels-​Alder reaction of an electron-​deficient heterocyclic azadiene: triethyl 1,​2,​4-​triazine-​3,​5,​6-​tricarboxylate and 2,​3,​6-​tricarboethoxypyridine 1988 http://vivo.scripps.edu/individual/endnote12246
http://vivo.scripps.edu/individual/e7n26376 AcademicArticle Accelerated inverse electron demand Diels-Alder reactions of 1-oxa-1,3-butadienes: [4 + 2] cycloaddition reactions of beta,gamma-unsaturated alpha-keto esters 1988 10.1021/jo00249a052 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n192828 AcademicArticle Acyl radicals: functionalized free radicals for intramolecular cyclization reactions 1988 10.1021/jo00249a053 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote246984 AcademicArticle Inverse electron demand Diels-Alder reactions of 2,4,6-tris(ethoxycarbonyl)-1,3,5-triazine and 2,4,6-tris(methylthio)-1,3,5-triazine - pyrimidine introduction 1988 10.1016/s0040-4020(01)85973-1 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/endnote252937 AcademicArticle Studies on the total synthesis of bouvardin and deoxybouvardin - cyclic hexapeptide cyclization studies and preparation of key partial structures 1988 10.1021/jo00238a005 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote300165 AcademicArticle Oxidative coupling of methyl 6-hydroxyindole-2-carboxylate with primary amines - preparation of 2-substituted methyl pyrrolo 2,3-e benzoxazole-5-carboxylates 1988 10.1021/jo00256a053 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote24237 AcademicArticle Total synthesis of (+/-)-n-2-(phenylsulfonyl)-cpi, (+/-)-cc-1065, (+)-cc-1065, ent-(-)-cc-1065, and the precise, functional agents (+/-)-cpi-cdpi2, (+)-cpi-cdpi2, and (-)-cpi-cdpi2 (+/-)-(3br-star,4as-star)-deoxy-cc-1065, (+)-(3br,4as)-deoxy-cc-1065, and (-)-(3bs,4ar)-deoxy-cc-1065 1988 10.1021/ja00222a043 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote3953 AcademicArticle Total synthesis of prodigiosin, prodigiosene, and desmethoxyprodigiosin - Diels-Alder reactions of heterocyclic azadienes and development of an effective palladium(II)-promoted 2,2'-bipyrrole coupling procedure 1988 10.1021/jo00242a013 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote232546 AcademicArticle Total synthesis of (+)CPI-CDPI2 and (-)-CPI-CDPI2 - (+)-(3br,4as)-deoxy-CC-1065 and (-)-(3bs,4ar)-deoxy-CC-1065 1988 10.1021/jo00238a042 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote15051 AcademicArticle Preparation and inverse electron demand Diels-Alder reaction of an electron-deficient heterocyclic azadiene - triethyl 1,2,4-triazine-3,5,6-tricarboxylate 1988 http://vivo.scripps.edu/individual/endnote12246
http://vivo.scripps.edu/individual/endnote373062 AcademicArticle Inverse electron demand Diels-Alder reactions of 3,6-bis(methylthio)-1,2,4,5-tetrazine - 1,2-diazine introduction and direct implementation of a divergent 1,2,4,5-tetrazine- 1,2-diazine- benzene (indoline indole) Diels-Alder strategy 1988 10.1021/jo00242a014 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote159208 AcademicArticle Thermal cyclo-addition reactions of pi-delocalized singlet vinylcarbenes - 3-carbon 1,1-dipoles/1,3-dipoles - the thermal 3-carbon + 2-carbon cyclo-addition 1988 10.1021/jo00250a002 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote13343 AcademicArticle Total synthesis of (+)-CC-1065 and ent-(-)-CC-1065 1988 10.1021/ja00212a067 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/e7n112519 AcademicArticle Preparation and inverse electron demand Diels-Alder reaction of an electron-deficient diene: methyl 2-oxo-5,6,7,8-tetrahydro-2H-1-benzopyran-3-carboxylate (2H-1-benzopyran-3-carboxylic acid, 5,6,7,8-tetrahydro-2-oxo-, methyl ester) 1987 http://vivo.scripps.edu/individual/endnote12246
http://vivo.scripps.edu/individual/e7n151037 AcademicArticle Preparation and three-carbon + two-carbon cycloaddition of a cyclopropenone ketal: cyclopropenone 1,3-propanediol ketal (4,8-dioxaspiro[2.5]oct-1-ene) 1987 http://vivo.scripps.edu/individual/endnote12246
http://vivo.scripps.edu/individual/endnote39970 AcademicArticle Activation and coupling of pyrrole-1-carboxylic acid in the formation of pyrrole N-carbonyl compounds - pyrrole-1-carboxylic acid anhydride 1987 10.1021/jo00387a046 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote58429 AcademicArticle Diels-alder reactions of heterocyclic azadienes - total synthesis of pde-i, pde-ii, and pde-i dimer methyl-ester 1987 10.1021/ja00243a027 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote206328 AcademicArticle Selectively protected L-dopa derivatives - application of the benzylic hydroperoxide rearrangement 1987 10.1021/jo00232a044 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote31699 AcademicArticle Further observations on the Lewis acid-catalyzed benzylic hydroperoxide rearrangement - use of a boron-trifluoride hydrogen-peroxide preformed, aged reagent 1987 10.1016/s0040-4039(00)95902-1 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote215926 AcademicArticle Streptonigrin and lavendamycin partial structures. Preparation of 7-amino-2-(2′-pyridyl)quinoline-5,8-quinone-6′-carboxylic acid: a probe for the minimum, potent pharmacophore of the naturally occurring antitumor-antibiotics 1987 10.1002/jhet.5570240504 http://vivo.scripps.edu/individual/endnote355769
http://vivo.scripps.edu/individual/endnote118849 AcademicArticle Streptonigrin and lavendamycin partial structures - probes for the minimum, potent pharmacophore of streptonigrin, lavendamycin, and synthetic quinoline-5,8-diones 1987 10.1021/jm00393a040 3656364 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote201544 AcademicArticle Indole N-carbonyl compounds - preparation and coupling of indole-1-carboxylic acid anhydride 1987 10.1021/jo00226a044 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote113754 AcademicArticle Total synthesis of prodigiosin 1987 10.1016/s0040-4039(00)95451-0 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote365520 AcademicArticle Studies on the total synthesis of CC-1065 - preparation of a synthetic, simplified 3-carbamoyl-1,2-dihydro-3h-pyrrolo 3,2-e indole dimer/trimer/tetramer (CDPI dimer/trimer/tetramer) and development of methodology for PDE-I dimer methyl-ester formation 1987 10.1021/jo00384a026 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n396489 AcademicArticle Diels-Alder reactions of heterocyclic azadienes: total synthesis of PDE-II methyl ester 1986 10.1021/jo00366a048 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote248573 AcademicArticle Thermal-reactions of cyclopropenone ketals - key mechanistic features and scope of the cycloaddition reactions of delocalized singlet vinylcarbenes - 3-carbon 1,1-dipoles 1,3-dipoles 1986 10.1021/ja00281a041 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote310880 AcademicArticle Benzylic hydroperoxide rearrangement - observations on a viable and convenient alternative to the Baeyer Villiger rearrangement 1986 10.1021/jo00376a079 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote62135 AcademicArticle An improved and divergent introduction of the streptonigrin and lavendamycin quinoline-5,8-quinone AB ring-systems 1986 10.3987/R-1986-04-1067 http://vivo.scripps.edu/individual/endnote14559
http://vivo.scripps.edu/individual/endnote33353 AcademicArticle Diels-Alder reactions of heterocyclic azadienes: scope and applications 1986 10.1021/cr00075a004 http://vivo.scripps.edu/individual/endnote51983
http://vivo.scripps.edu/individual/endnote289061 AcademicArticle Diels-Alder cycloaddition reactions of cyclopropenone ketals: dual participation in inverse electron demand (LUMOdiene controlled) and normal HOMOdiene controlled) Diels-Alder reactions, approaches to the preparation of tropones 1986 10.1016/s0040-4020(01)90567-8 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/endnote88058 AcademicArticle Thermal-reactions of cyclopropenone ketals - application of the cycloaddition reactions of delocalized singlet vinylcarbenes - 3-carbon 1,1-dipoles 1,3-dipoles - an alternative synthesis of deacetamidocolchiceine - formal total synthesis of colchicine 1986 10.1021/ja00281a042 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote390618 AcademicArticle Diels-Alder cycloadditions of rigid dienophiles: a probe for allylic axial substituent control of the pi-facial selectivity in the Diels-Alder reaction 1986 10.1016/s0040-4039(00)84072-1 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/e7n384434 AcademicArticle Thermal, four-carbon + three-carbon cycloaddition reaction of cyclopropenone ketals. Total synthesis of deacetamidocolchiceine: formal total synthesis of colchicine 1985 10.1021/jo00218a042 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote112947 AcademicArticle Inverse electron demand Diels-Alder reactions of heterocyclic azadienes - formal total synthesis of streptonigrin 1985 10.1021/ja00306a024 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote65240 AcademicArticle Antimicrobial and cytotoxic properties of 9,10-dihydrophenanthrenes: structure activity studies on juncusol 1985 10.1021/jm00148a031 4045930 http://vivo.scripps.edu/individual/endnote266962
http://vivo.scripps.edu/individual/endnote282630 AcademicArticle Total synthesis of lavendamycin methyl-ester 1985 10.1021/jo00350a070 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote286000 AcademicArticle Inverse electron demand Diels-Alder reactions of heterocyclic aza dienes - studies on the total synthesis of lavendamycin - investigative studies on the preparation of the CDE beta-carboline ring-system and AB quinoline-5,8-quinone ring-system 1985 10.1021/jo00350a069 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote321884 AcademicArticle Preparation of optically-active, functionalized cis-delta-6-1-octalones 1985 10.1021/jo00211a024 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote246072 AcademicArticle Regioselectivity of the intermolecular Diels-Alder reaction of acyl nitroso-compounds (C-nitrosocarbonyl compounds) and nitrosoformates (O-nitrosocarbonyl compounds) - preparation of functionalized cis-delta-6-1-octalones 1985 10.1021/jo00211a025 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote31052 AcademicArticle A detailed, convenient preparation of dimethyl "1,2,4,5-tetrazine-3,6-dicarboxylate 1985 10.1021/jo00225a076 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n45212 AcademicArticle Regioselectivity in the intermolecular Diels-Alder reaction of acyl nitroso compounds (C-nitrosocarbonyl compounds) and nitrosoformates (O-nitrosocarbonyl compounds) 1984 10.1021/jo00195a057 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote380280 AcademicArticle Palladium (0) mediated beta-carboline synthesis - preparation of the CDE ring-system of lavendamycin 1984 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote268550 AcademicArticle Total syntheses of azafluoranthene alkaloids: rufescine and imeluteine 1984 10.1021/jo00195a035 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote60623 AcademicArticle Effective, thermal 3-carbon + 2-carbon cycloaddition for cyclopentenone formation - formal 1,3-dipolar cycloaddition of cyclopropenone ketals 1984 10.1021/ja00315a065 http://vivo.scripps.edu/individual/endnote181842
http://vivo.scripps.edu/individual/endnote84558 AcademicArticle Thermal, 3-carbon + 2-atom cycloaddition of cyclopropenone ketals with carbon-heteroatom double-bonds - butenolide, furan, and gamma-keto ester preparation 1984 10.1016/s0040-4039(01)91394-2 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote161185 AcademicArticle Inverse electron demand Diels-Alder reactions of 3-carbomethoxy-2-pyrones - controlled introduction of oxygenated aromatics - benzene, phenol, catechol, resorcinol, and pyrogallol annulation - regiospecific total synthesis of sendaverine and a preparation of 6,7-benzomorphans 1984 10.1021/jo00195a033 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote275780 AcademicArticle Thermal cycloaddition of dimethyl "1,2,4,5-tetrazine-3,6-dicarboxylate with electron-rich olefins - 1,2-diazine and pyrrole introduction - preparation of octamethylporphin (OMP) 1984 10.1021/jo00197a015 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote26571 AcademicArticle Effective, thermal one-carbon + 2-carbon cycloaddition of cyclopropenone ketals with electron deficient olefins - cyclopropane formation 1984 10.1016/s0040-4039(01)91393-0 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote143477 AcademicArticle Regiospecific total synthesis of juncusol 1984 10.1021/jo00195a034 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote161688 AcademicArticle Intramolecular diels-alder reactions of 1,2-diazines - general indoline synthesis - studies on the preparation of the central and right-hand segments of cc-1065 1984 10.1021/jo00186a032 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote173664 AcademicArticle Direct introduction of nitriles via use of unstable reissert intermediates - convenient procedures for the preparation of 2-cyanoquinolines and 1-cyanoisoquinolines 1984 10.1021/jo00195a036 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/e7n301118 AcademicArticle Formal total synthesis of streptonigrin 1983 10.1021/jo00152a049 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote372016 AcademicArticle Inverse electron demand Diels-Alder reactions of 3-carbomethoxy-2-pyrones - controlled introduction of oxygenated aromatics - benzene, phenol, catechol, resorcinol, pyrogallol annulation 1983 10.1016/s0040-4039(01)99816-8 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote369173 AcademicArticle Diels-Alder reactions of azadienes 1983 10.1016/s0040-4020(01)92154-4 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/endnote42403 AcademicArticle 1,2,4-triazine preparation via thermal cycloaddition of dimethyl 1,2,4,5-tetrazine-3,6-dicarboxylate with aryl thioimidates 1983 10.1016/s0040-4039(00)85941-9 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote242354 AcademicArticle Diels-Alder reaction of heterocyclic azadienes. 2. Catalytic Diels-Alder reaction of in situ generated enamines with 1,2,4-triazines: general pyridine annulation 1982 10.1021/jo00344a031 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote233434 AcademicArticle Regiospecific total synthesis of juncusol 1982 10.1016/s0040-4039(00)85652-x http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote266303 AcademicArticle Inverse electron demand diels-alder reaction of 3-carbomethoxy-2-pyrones with 1,1-dimethoxyethylene - a simple and mild method of aryl annulation 1982 10.1016/s0040-4039(00)85651-8 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote195921 AcademicArticle Thermal cycloaddition of 1,3,5-triazine with enamines - regiospecific pyrimidine annulation 1982 10.1021/jo00134a034 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote1836 AcademicArticle Synthetic analgesics - preparation of racemic 6,7-benzomorphans 1982 10.1016/s0040-4039(00)85653-1 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote294737 AcademicArticle Pyridine construction via thermal cycloaddition of 1,2,4-triazines with enamines - studies on the preparation of the bi-aryl CD rings of streptonigrin 1982 10.1021/jo00140a035 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote121295 AcademicArticle Preparation of 3-methyl-4-vinyl-1,2,5-oxadiazole and 3-methyl-4-vinyl-1,2,5-thiadiazole 1981 10.1002/jhet.5570180636 http://vivo.scripps.edu/individual/endnote355769
http://vivo.scripps.edu/individual/endnote365275 AcademicArticle Preparation of (R)-(+) and (S)-(-)-4-iodo-1,2-epoxybutane (R)-(2-iodoethyl)oxirane and (S)-(2-iodoethyl)oxirane , useful chiral synthons 1981 10.1021/jo00319a034 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote166728 AcademicArticle Diels-alder reaction of heterocyclic azadienes .1. Thermal cycloaddition of 1,2,4-triazine with enamines - simple preparation of substituted pyridines 1981 10.1021/jo00323a044 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote227070 AcademicArticle A simplified isoquinoline synthesis 1981 10.1016/s0040-4020(01)93272-7 http://vivo.scripps.edu/individual/endnote9731
http://vivo.scripps.edu/individual/endnote41494 AcademicArticle A simple and convenient phenol annelation 1980 10.1021/jo01312a044 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/n25725 Thesis I. New annulation processes ; II. Studies directed toward a biomimetic syntheic approach to prostaglandins 1980
http://vivo.scripps.edu/individual/endnote342187 AcademicArticle Convenient preparation of 2-substituted benzothiazoles 1978 10.1021/jo00405a050 http://vivo.scripps.edu/individual/endnote171323
http://vivo.scripps.edu/individual/endnote137289 AcademicArticle Concerning the stereochemistry of 9-methyl-Δ1-3-octalone 1978 10.1016/S0040-4039(01)88970-X http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote156107 AcademicArticle New annulation processes for fused and spiro rings based on chemistry of benzothiazoles 1978 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote8088 AcademicArticle Application of benzothiazoles to carbon-carbon bond formation in organic-synthesis 1978 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote160204 AcademicArticle Oxidative cationic cyclization reactions effected by pyridinium chlorochromate 1978 10.1016/S0040-4039(01)94800-2 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote54448 AcademicArticle New and unusually flexible scheme for annulation to form fused cyclohexenone units 1978 10.1016/S0040-4039(01)85680-X http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote22302 AcademicArticle Benzothiazoles as carbonyl equivalents 1978 http://vivo.scripps.edu/individual/endnote225462
http://vivo.scripps.edu/individual/endnote284510 AcademicArticle Synthesis and chiroptical properties of some asymmetric planar cisoid dienes 1976 10.1016/0040-4020(76)80042-7 http://vivo.scripps.edu/individual/endnote9731