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• Cryo-EM structure of hexameric yeast Lon protease (PIM1) highlights the importance of conserved structural elements  Academic Article
• Discovery of 3,5-substituted 6-azaindazoles as potent pan-Pim inhibitors  Academic Article
• Discovery of 5-azaindazole (GNE-955) as a potent pan-pim inhibitor with optimized bioavailability  Academic Article
• Discovery of novel pyrazolo[1,5-a]pyrimidines as potent pan-Pim inhibitors by structure- and property-based drug design  Academic Article
• High-throughput kinase profiling: A more efficient approach toward the discovery of new kinase inhibitors  Academic Article
• USP7 small-molecule inhibitors interfere with ubiquitin binding  Academic Article