subject area of
- Discovery of 3,5-substituted 6-azaindazoles as potent pan-Pim inhibitors Academic Article
- Discovery of 5-azaindazole (GNE-955) as a potent pan-pim inhibitor with optimized bioavailability Academic Article
- Discovery of novel pyrazolo[1,5-a]pyrimidines as potent pan-Pim inhibitors by structure- and property-based drug design Academic Article
- High-throughput kinase profiling: A more efficient approach toward the discovery of new kinase inhibitors Academic Article
- USP7 small-molecule inhibitors interfere with ubiquitin binding Academic Article