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Botulinum Toxins, Type A

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  • 8-Hydroxyquinoline and hydroxamic acid inhibitors of botulinum neurotoxin BoNT/A  Academic Article
  • A cyclic peptide-polymer probe for the detection of Clostridium botulinum neurotoxin serotype A  Academic Article
  • A high-throughput-compatible FRET-based platform for identification and characterization of botulinum neurotoxin light chain modulators  Academic Article
  • A structural perspective of the sequence variability within botulinum neurotoxin subtypes a1-a4  Academic Article
  • Active-site mutagenesis of tetanus neurotoxin implicates tyr-375 and glu-271 in metalloproteolytic activity  Academic Article
  • An in vitro and in vivo disconnect uncovered through high-throughput identification of botulinum neurotoxin A antagonists  Academic Article
  • Antibody mapping to domains of botulinum neurotoxin serotype A in the complexed and uncomplexed forms  Academic Article
  • Benzoquinones as inhibitors of botulinum neurotoxin serotype A  Academic Article
  • Benzylidene cyclopentenediones: First irreversible inhibitors against botulinum neurotoxin A's zinc endopeptidase  Academic Article
  • Biophysical characterization of the stability of the 150-kilodalton botulinum toxin, the nontoxic component, and the 900-kilodalton botulinum toxin complex species  Academic Article
  • Botulinum neurotoxin a protease: Discovery of natural product exosite inhibitors  Academic Article
  • Botulinum neurotoxin subtype A2 enters neuronal cells faster than subtype A1  Academic Article
  • Chirality holds the key for potent inhibition of the botulinum neurotoxin serotype A protease  Academic Article
  • Crystal structure of botulinum neuro-toxin type a and implications for toxicity  Academic Article
  • Crystal structure of botulinum neurotoxin type a in complex with the cell surface co-receptor gt1b - insight into the toxin-neuron interaction  Academic Article
  • Dynamics and number of trans-SNARE complexes determine nascent fusion pore properties  Academic Article
  • Effects of hydroxamate metalloendoprotease inhibitors on botulinum neurotoxin a poisoned mouse neuromuscular junctions  Academic Article
  • Evaluation of adamantane hydroxamates as botulinum neurotoxin inhibitors: Synthesis, crystallography, modeling, kinetic and cellular based studies  Academic Article
  • Examination of α-exosite inhibitors against Botulinum neurotoxin A protease through structure-activity relationship studies of chicoric acid  Academic Article
  • High-throughput screening technologies for botulinum neurotoxins  Academic Article
  • Identification of a potent botulinum neurotoxin a protease inhibitor using in situ lead identification chemistry  Academic Article
  • Identification of clinically viable quinolinol inhibitors of botulinum neurotoxin A light chain  Academic Article
  • Identification of fibroblast growth factor receptor 3 (FGFR3) as a protein receptor for botulinum neurotoxin serotype A (BoNT/A)  Academic Article
  • Inhibition of botulinum neurotoxin BoNT/A  Academic Article
  • Investigating novel therapeutic targets and molecular mechanisms to treat botulinum neurotoxin a intoxication  Academic Article
  • Light chain of botulinum neurotoxin serotype A: Structural resolution of a catalytic intermediate  Academic Article
  • Lycopodium clavatum exine microcapsules enable safe oral delivery of 3,4-diaminopyridine for treatment of botulinum neurotoxin A intoxication  Academic Article
  • Molecular evolution of antibody cross-reactivity for two subtypes of type a botulinum neurotoxin  Academic Article
  • Monitoring botulinum neurotoxin a activity with peptide-functionalized quantum dot resonance energy transfer sensors  Academic Article
  • Probing BoNT/A protease exosites: implications for inhibitor design and light chain longevity  Academic Article
  • Purification, modeling, and analysis of botulinum neurotoxin subtype a5 (bont/a5) from clostridium botulinum strain a661222  Academic Article
  • Recombinant expression and purification of the botulinum neurotoxin type a translocation domain  Academic Article
  • Reexamining hydroxamate inhibitors of botulinum neurotoxin serotype a: Extending towards the beta-exosite  Academic Article
  • Selection and characterization of a human monoclonal neutralizing antibody for clostridium Botulinum Neurotoxin serotype B  Academic Article
  • Structural basis of cell surface receptor recognition by botulinum neurotoxin B  Academic Article
  • Structural characterization of three novel hydroxamate-based zinc chelating inhibitors of the clostridium botulinum serotype a neurotoxin light chain metalloprotease reveals a compact binding site resulting from 60/70 loop flexibility  Academic Article
  • Superactivation of the botulinum neurotoxin serotype A light chain metalloprotease: A new wrinkle in botulinum neurotoxin  Academic Article
  • Synthesis and evaluation of library of betulin derivatives against the botulinum neurotoxin A protease  Academic Article
  • Synthesis and structure-activity relationships of second-generation hydroxamate botulinum neurotoxin A protease inhibitors  Academic Article
  • Synthesis, characterization and development of a high-throughput methodology for the discovery of botulinum neurotoxin A inhibitors  Academic Article
  • Synthesis/biological evaluation of hydroxamic acids and their prodrugs as inhibitors for Botulinum neurotoxin A light chain  Academic Article
  • Synthetic substrate for application in both high and low throughput assays for botulinum neurotoxin B protease inhibitors  Academic Article
  • Tandem fluorescent proteins as enhanced FRET-based substrates for botulinum neurotoxin activity  Academic Article
  • Targeting botulinum A cellular toxicity: a prodrug approach  Academic Article
  • The use of small molecules to investigate molecular mechanisms and therapeutic targets for treatment of botulinum neurotoxin A intoxication  Academic Article
  • Toosendanin: Synthesis of the AB-ring and investigations of its anti-botulinum properties (part II)  Academic Article
  • Toward the discovery of dual inhibitors for botulinum neurotoxin A: concomitant targeting of endocytosis and light chain protease activity  Academic Article
  • Vitamin B-2-mediated cellular photoinhibition of botulinum neurotoxin A  Academic Article

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