subject area of
- 8-Hydroxyquinoline and hydroxamic acid inhibitors of botulinum neurotoxin BoNT/A Academic Article
- A cyclic peptide-polymer probe for the detection of Clostridium botulinum neurotoxin serotype A Academic Article
- A high-throughput-compatible FRET-based platform for identification and characterization of botulinum neurotoxin light chain modulators Academic Article
- A structural perspective of the sequence variability within botulinum neurotoxin subtypes a1-a4 Academic Article
- Active-site mutagenesis of tetanus neurotoxin implicates tyr-375 and glu-271 in metalloproteolytic activity Academic Article
- An in vitro and in vivo disconnect uncovered through high-throughput identification of botulinum neurotoxin A antagonists Academic Article
- Antibody mapping to domains of botulinum neurotoxin serotype A in the complexed and uncomplexed forms Academic Article
- Benzoquinones as inhibitors of botulinum neurotoxin serotype A Academic Article
- Benzylidene cyclopentenediones: First irreversible inhibitors against botulinum neurotoxin A's zinc endopeptidase Academic Article
- Biophysical characterization of the stability of the 150-kilodalton botulinum toxin, the nontoxic component, and the 900-kilodalton botulinum toxin complex species Academic Article
- Botulinum neurotoxin a protease: Discovery of natural product exosite inhibitors Academic Article
- Botulinum neurotoxin subtype A2 enters neuronal cells faster than subtype A1 Academic Article
- Chirality holds the key for potent inhibition of the botulinum neurotoxin serotype A protease Academic Article
- Crystal structure of botulinum neuro-toxin type a and implications for toxicity Academic Article
- Crystal structure of botulinum neurotoxin type a in complex with the cell surface co-receptor gt1b - insight into the toxin-neuron interaction Academic Article
- Dynamics and number of trans-SNARE complexes determine nascent fusion pore properties Academic Article
- Effects of hydroxamate metalloendoprotease inhibitors on botulinum neurotoxin a poisoned mouse neuromuscular junctions Academic Article
- Evaluation of adamantane hydroxamates as botulinum neurotoxin inhibitors: Synthesis, crystallography, modeling, kinetic and cellular based studies Academic Article
- Examination of α-exosite inhibitors against Botulinum neurotoxin A protease through structure-activity relationship studies of chicoric acid Academic Article
- High-throughput screening technologies for botulinum neurotoxins Academic Article
- Identification of a potent botulinum neurotoxin a protease inhibitor using in situ lead identification chemistry Academic Article
- Identification of clinically viable quinolinol inhibitors of botulinum neurotoxin A light chain Academic Article
- Identification of fibroblast growth factor receptor 3 (FGFR3) as a protein receptor for botulinum neurotoxin serotype A (BoNT/A) Academic Article
- Inhibition of botulinum neurotoxin BoNT/A Academic Article
- Investigating novel therapeutic targets and molecular mechanisms to treat botulinum neurotoxin a intoxication Academic Article
- Light chain of botulinum neurotoxin serotype A: Structural resolution of a catalytic intermediate Academic Article
- Lycopodium clavatum exine microcapsules enable safe oral delivery of 3,4-diaminopyridine for treatment of botulinum neurotoxin A intoxication Academic Article
- Molecular evolution of antibody cross-reactivity for two subtypes of type a botulinum neurotoxin Academic Article
- Monitoring botulinum neurotoxin a activity with peptide-functionalized quantum dot resonance energy transfer sensors Academic Article
- Probing BoNT/A protease exosites: implications for inhibitor design and light chain longevity Academic Article
- Purification, modeling, and analysis of botulinum neurotoxin subtype a5 (bont/a5) from clostridium botulinum strain a661222 Academic Article
- Recombinant expression and purification of the botulinum neurotoxin type a translocation domain Academic Article
- Reexamining hydroxamate inhibitors of botulinum neurotoxin serotype a: Extending towards the beta-exosite Academic Article
- Selection and characterization of a human monoclonal neutralizing antibody for clostridium Botulinum Neurotoxin serotype B Academic Article
- Structural basis of cell surface receptor recognition by botulinum neurotoxin B Academic Article
- Structural characterization of three novel hydroxamate-based zinc chelating inhibitors of the clostridium botulinum serotype a neurotoxin light chain metalloprotease reveals a compact binding site resulting from 60/70 loop flexibility Academic Article
- Superactivation of the botulinum neurotoxin serotype A light chain metalloprotease: A new wrinkle in botulinum neurotoxin Academic Article
- Synthesis and evaluation of library of betulin derivatives against the botulinum neurotoxin A protease Academic Article
- Synthesis and structure-activity relationships of second-generation hydroxamate botulinum neurotoxin A protease inhibitors Academic Article
- Synthesis, characterization and development of a high-throughput methodology for the discovery of botulinum neurotoxin A inhibitors Academic Article
- Synthesis/biological evaluation of hydroxamic acids and their prodrugs as inhibitors for Botulinum neurotoxin A light chain Academic Article
- Synthetic substrate for application in both high and low throughput assays for botulinum neurotoxin B protease inhibitors Academic Article
- Tandem fluorescent proteins as enhanced FRET-based substrates for botulinum neurotoxin activity Academic Article
- Targeting botulinum A cellular toxicity: a prodrug approach Academic Article
- The use of small molecules to investigate molecular mechanisms and therapeutic targets for treatment of botulinum neurotoxin A intoxication Academic Article
- Toosendanin: Synthesis of the AB-ring and investigations of its anti-botulinum properties (part II) Academic Article
- Toward the discovery of dual inhibitors for botulinum neurotoxin A: concomitant targeting of endocytosis and light chain protease activity Academic Article
- Vitamin B-2-mediated cellular photoinhibition of botulinum neurotoxin A Academic Article