recent publications
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academic article
- Leibowitz, M. D., Fievet, C., Hennuyer, N., Peinado-Onsurbe, J., Duez, H., Berger, J., Cullinan, C. A., Sparrow, C. P., Baffic, J., Berger, G. D., Santini, C., Marquis, R. W., et al. Activation of PPARdelta alters lipid metabolism in db/db mice FEBS Letters 2000 473:333-336 DOI:10.1016/s0014-5793(00)01554-4 PMID:10818235
- Johnson, B. A., Wilson, E. M., Li, Y., Moller, D. E., Smith, R. G., Zhou, G. C. Ligand-induced stabilization of PPARgamma monitored by NMR spectroscopy: implications for nuclear receptor activation Journal of Molecular Biology 2000 298:187-194 DOI:10.1006/jmbi.2000.3636 PMID:10764590
- Zhang, B., Salituro, G., Szalkowski, D., Li, Z. H., Zhang, Y., Royo, I., Vilella, D., Diez, M. T., Pelaez, F., Ruby, C., Kendall, R. L., Mao, X. Z., et al. Discovery of a small molecule insulin mimetic with antidiabetic activity in mice Science 1999 284:974-977 DOI:10.1126/science.284.5416.974 PMID:10320380
- Elbrecht, A., Chen, Y. L., Adams, A., Berger, J., Griffin, P., Klatt, T., Zhang, B., Menke, J., Zhou, G. C., Smith, R. G., Moller, D. E. L-764406 is a partial agonist of human peroxisome proliferator-activated receptor gamma. The role of Cys313 in ligand binding Journal of Biological Chemistry 1999 274:7913-7922 DOI:10.1074/jbc.274.12.7913 PMID:10075686
- Berger, J., Leibowitz, M. D., Doebber, T. W., Elbrecht, A., Zhang, B., Zhou, G. C., Biswas, C., Cullinan, C. A., Hayes, N. S., Li, Y., Tanen, M., Ventre, J., et al. Novel peroxisome proliferator-activated receptor (PPAR) gamma and PPARdelta ligands produce distinct biological effects Journal of Biological Chemistry 1999 274:6718-6725 DOI:10.1074/jbc.274.10.6718 PMID:10037770
- Zhou, G. C., Cummings, R., Li, Y., Mitra, S., Wilkinson, H. A., Elbrecht, A., Hermes, J. D., Schaeffer, J. M., Smith, R. G., Moller, D. E. Nuclear receptors have distinct affinities for coactivators: characterization by fluorescence resonance energy transfer Molecular Endocrinology 1998 12:1594-1604 DOI:10.1210/me.12.10.1594 PMID:9773982
- Ding, V. D. H., Moller, D. E., Feeney, W. P., Didolkar, V., Nakhla, A. M., Rhodes, L., Rosner, W., Smith, R. G. Sex hormone-binding globulin mediates prostate androgen receptor action via a novel signaling pathway Endocrinology 1998 139:213-218 DOI:10.1210/en.139.1.213 PMID:9421417