recent publications

• academic article

  • Yang, M. G., Dhar, T. G. M., Xiao, Z., Xiao, H. Y., Duan, J. J. W., Jiang, B., Galella, M. A., Cunningham, M., Wang, J., Habte, S., Shuster, D., McIntyre, K. W., et al. Improving the pharmacokinetic and CYP inhibition profiles of azaxanthene-based glucocorticoid receptor modulators-identification of (S)-5-(2-(9-fluoro-2-(4-(2-hydroxypropan-2-yl)phenyl)-5H-chromeno[2,3-b]pyridin-5-yl)-2-methylpropanamido)-N-(tetrahydro-2H-pyran-4-yl)-1,3,4-thiadiazole-2-carboxamide (BMS-341) Journal of Medicinal Chemistry  2015 58:4278-4290  DOI:10.1021/acs.jmedchem.5b00257  PMID:25905990