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CDK2/cyclinA inhibitors: Targeting the cyclinA recruitment site with small molecules derived from peptide leads

Academic Article
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  • Overview
  • Research
  • Identity
  • Additional Document Info
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Overview

authors

  • Castanedo, G.
  • Clark, K.
  • Wang, S.
  • Tsui, Vickie
  • Wong, M.
  • Nicholas, J.
  • Wickramasinghe, D.
  • Marsters, Jr., J. C.
  • Sutherlin, D.

publication date

  • March 2006

journal

  • Bioorganic & Medicinal Chemistry Letters  Journal

subject areas

  • Amino Acid Substitution
  • Cyclin A
  • Cyclin-Dependent Kinase 2
  • Drug Design
  • Enzyme Inhibitors
  • Guanidine
  • Humans
  • Models, Molecular
  • Peptide Fragments
  • Protein Conformation
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Research

keywords

  • CDK2/cyclinA
  • guanidine replacement
  • protein-protein interaction inhibitor
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Identity

International Standard Serial Number (ISSN)

  • 0960-894X

Digital Object Identifier (DOI)

  • 10.1016/j.bmcl.2005.12.004

PubMed ID

  • 16384702
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Additional Document Info

start page

  • 1716

end page

  • 1720

volume

  • 16

issue

  • 6

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