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GNE-781, a highly advanced potent and selective bromodomain inhibitor of cyclic adenosine monophosphate response element binding protein, binding protein (CBP)

Academic Article
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  • Identity
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Overview

authors

  • Romero, F. A.
  • Murray, J.
  • Lai, K. W.
  • Tsui, Vickie
  • Albrecht, B. K.
  • An, L.
  • Beresini, M. H.
  • de Leon Boenig, G.
  • Bronner, S. M.
  • Chan, E. W.
  • Chen, K.
  • Chen, Z.
  • Choo, E. F.
  • Clagg, K.
  • Clark, K.
  • Crawford, T. D.
  • Cyr, P.
  • Nagata, D. D.
  • Gascoigne, K. E.
  • Grogan, J. L.
  • Hatzivassiliou, G.
  • Huang, W.
  • Hunsaker, T. L.
  • Kaufman, S.
  • Koenig, S. G.
  • Li, R.
  • Li, Y.
  • Liang, X.
  • Liao, J.
  • Liu, W.
  • Ly, J.
  • Maher, J.
  • Masui, C.
  • Merchant, M.
  • Ran, Y. Q.
  • Taylor, A. M.
  • Wai, J.
  • Wang, F.
  • Wei, X.
  • Yu, D.
  • Zhu, B. Y.
  • Zhu, X.
  • Magnuson, S.

publication date

  • November 2017

journal

  • Journal of Medicinal Chemistry  Journal

subject areas

  • Animals
  • Antineoplastic Agents
  • CREB-Binding Protein
  • Dogs
  • Female
  • Forkhead Transcription Factors
  • HEK293 Cells
  • Humans
  • Macaca fascicularis
  • Male
  • Mice
  • Protein Domains
  • Proto-Oncogene Proteins c-myc
  • Pyrazoles
  • Pyridines
  • RNA
  • Rats, Sprague-Dawley
  • Structure-Activity Relationship
  • Xenograft Model Antitumor Assays
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Identity

International Standard Serial Number (ISSN)

  • 0022-2623

Digital Object Identifier (DOI)

  • 10.1021/acs.jmedchem.7b00796

PubMed ID

  • 28892380
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Additional Document Info

start page

  • 9162

end page

  • 9183

volume

  • 60

issue

  • 22

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