recent publications
-
academic article
- Velcicky, J., Mathison, C. J. N., Nikulin, V., Pflieger, D., Epple, R., Azimioara, M., Cow, C., Michellys, P. Y., Rigollier, P., Beisner, D. R., Bodendorf, U., Guerini, D., et al. Discovery of Orally active hydroxyethylamine based SPPL2a inhibitors ACS Medicinal Chemistry Letters 2019 10:887-892 DOI:10.1021/acsmedchemlett.9b00044 PMID:31223443 PMCID:PMC6580379
- Khare, S., Nagle, A. S., Biggart, A., Lai, Y. H., Liang, F., Davis, L. C., Barnes, S. W., Mathison, C. J. N., Myburgh, E., Gao, M. Y., Gillespie, J. R., Liu, X., et al. Proteasome inhibition for treatment of leishmaniasis, Chagas disease and sleeping sickness Nature 2016 537:229-233 DOI:10.1038/nature19339 PMID:27501246 PMCID:PMC5161665
- Nagle, A. S., Khare, S., Kumar, A. B., Supek, F., Buchynskyy, A., Mathison, C. J. N., Chennamaneni, N. K., Pendem, N., Buckner, F. S., Gelb, M. H., Molteni, V. Recent developments in drug discovery for leishmaniasis and human African trypanosomiasis Chemical Reviews 2014 114:11305-11347 DOI:10.1021/cr500365f PMID:25365529
-
Nicolaou, K. C.*, Mathison, C. J. N.*
Synthesis of imides, N-acyl vinylogous carbamates and ureas, and nitriles by oxidation of amides and amines with Dess-Martin periodinane
Angewandte Chemie-International Edition
2005
44:5992-5997
DOI:10.1002/anie.200501853
PMID:16124020
(* = equal contribution)
-
Nicolaou, K. C., Montagnon, T., Vassilikogiannakis, G., Mathison, C. J. N.
The total synthesis of coleophomones B, C, and D
Journal of the American Chemical Society
2005
127:8872-8888
DOI:10.1021/ja0509984
PMID:15954796
- Bourdon, L. H., Fairfax, D. J., Martin, G. S., Mathison, C. J., Zhichkin, P. An enantioselective synthesis of nitrogen protected 3-arylserine esters Tetrahedron-Asymmetry 2004 15:3485-3487 DOI:10.1016/j.tetasy.2004.10.005
-
Nicolaou, K. C.*, Mathison, C. J. N.*, Montagnon, T.
o-Iodoxybenzoic acid (IBX) as a viable reagent in the manipulation of nitrogen- and sulfur-containing substrates: scope, generality, and mechanism of IBX-mediated amine oxidations and dithiane deprotections
Journal of the American Chemical Society
2004
126:5192-5201
DOI:10.1021/ja0400382
PMID:15099102
(* = equal contribution)
- Laitar, D. S., Mathison, C. J. N., Davis, W. M., Sadighi, J. P. Copper(I) complexes of a heavily fluorinated beta-diketiminate ligand: Synthesis, electronic properties, and intramolecular aerobic hydroxylation Inorganic Chemistry 2003 42:7354-7356 DOI:10.1021/ic035056j PMID:14606823
-
Nicolaou, K. C.*, Mathison, C. J. N.*, Montagnon, T.
New reactions of IBX: Oxidation of nitrogen- and sulfur-containing substrates to afford useful synthetic intermediates
Angewandte Chemie-International Edition
2003
42:4077-4082
DOI:10.1002/anie.200352076
PMID:12973775
(* = equal contribution)